CN100546977C - 抑制旋转异构酶的新化合物及其应用 - Google Patents

抑制旋转异构酶的新化合物及其应用 Download PDF

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CN100546977C
CN100546977C CNB038252651A CN03825265A CN100546977C CN 100546977 C CN100546977 C CN 100546977C CN B038252651 A CNB038252651 A CN B038252651A CN 03825265 A CN03825265 A CN 03825265A CN 100546977 C CN100546977 C CN 100546977C
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phenyl
hydroxyl
chloro
urea
thiocarbamide
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CN1701061A (zh
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J·克内勒
M·舒特考斯基
G·胡梅尔
T·特拉德勒
L·朱卜龙
C·克里斯特纳
D·沙恩
R·斯特拉齐
C·吉布森
F·奥斯特坎普
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Jerini AG
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CNB038252651A 2002-09-18 2003-09-18 抑制旋转异构酶的新化合物及其应用 Expired - Fee Related CN100546977C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02020987.0 2002-09-18
EP20020020987 EP1402888A1 (en) 2002-09-18 2002-09-18 The use of substituted carbocyclic compounds as rotamases inhibitors

Publications (2)

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CN1701061A CN1701061A (zh) 2005-11-23
CN100546977C true CN100546977C (zh) 2009-10-07

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US (2) US20070054904A1 (https=)
EP (3) EP1402888A1 (https=)
JP (2) JP2005539072A (https=)
KR (1) KR20050053673A (https=)
CN (1) CN100546977C (https=)
AU (1) AU2003271619A1 (https=)
BR (1) BR0314544A (https=)
CA (1) CA2498662A1 (https=)
MX (1) MXPA05003084A (https=)
PL (1) PL374846A1 (https=)
RU (2) RU2005111256A (https=)
SG (1) SG165995A1 (https=)
WO (1) WO2004026815A2 (https=)
ZA (1) ZA200501913B (https=)

Cited By (2)

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CN107417578A (zh) * 2017-08-23 2017-12-01 沈阳海诺威医药科技有限公司 N‑(3,5‑二甲基金刚烷‑1‑基)‑n’‑取代苯基脲类化合物及其制备方法和用途
CN111233692A (zh) * 2020-01-19 2020-06-05 江西农业大学 一种香茅酸酰胺类衍生物及其制备方法与应用

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JP2006518738A (ja) * 2003-02-12 2006-08-17 トランス テック ファーマ,インコーポレイテッド 治療薬としての置換アゾール誘導体
CA2520763A1 (en) * 2003-04-03 2004-10-21 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
RS50589B (sr) * 2003-12-23 2010-05-07 H. Lundbeck A/S. 2-(1h-indolilsulfanil)-benzil amin derivati kao ssri
US7304086B2 (en) * 2004-02-05 2007-12-04 Probiodrug Ag Inhibitors of glutaminyl cyclase
EP1765311A4 (en) 2004-03-16 2009-04-29 Univ California REDUCTION OF NEPHROPATHY WITH INHIBITORS OF SOLUBLE EPOXY HYDROLASE AND EPOXYEICOSANOIDS
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
WO2005113534A2 (en) * 2004-05-12 2005-12-01 Schering Corporation Cxcr1 and cxcr2 chemokine antagonists
AR052308A1 (es) * 2004-07-16 2007-03-14 Lundbeck & Co As H Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto
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