KR20050053673A - 로타마제 억제제로서의 페놀유도체 및 이들의 용도 - Google Patents

로타마제 억제제로서의 페놀유도체 및 이들의 용도 Download PDF

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Publication number
KR20050053673A
KR20050053673A KR1020057004693A KR20057004693A KR20050053673A KR 20050053673 A KR20050053673 A KR 20050053673A KR 1020057004693 A KR1020057004693 A KR 1020057004693A KR 20057004693 A KR20057004693 A KR 20057004693A KR 20050053673 A KR20050053673 A KR 20050053673A
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South Korea
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phenyl
hydroxy
chloro
benzylamino
phenol
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KR1020057004693A
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Korean (ko)
Inventor
조첸 크놀레
마이크 스츄트코와스키
게르드 훔멜
토마스 트래드레르
로렌스 조브론
클라우디아 크리스트네르
디르크 스취아른
롤랜드 스트라지에스
크리스토프 지브손
프랭크 오스테르캄프
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제리니 아게
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    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/32Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • C07C275/34Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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    • A61K31/17Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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KR1020057004693A 2002-09-18 2003-09-18 로타마제 억제제로서의 페놀유도체 및 이들의 용도 Ceased KR20050053673A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02020987.0 2002-09-18
EP20020020987 EP1402888A1 (en) 2002-09-18 2002-09-18 The use of substituted carbocyclic compounds as rotamases inhibitors

Publications (1)

Publication Number Publication Date
KR20050053673A true KR20050053673A (ko) 2005-06-08

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KR1020057004693A Ceased KR20050053673A (ko) 2002-09-18 2003-09-18 로타마제 억제제로서의 페놀유도체 및 이들의 용도

Country Status (14)

Country Link
US (2) US20070054904A1 (https=)
EP (3) EP1402888A1 (https=)
JP (2) JP2005539072A (https=)
KR (1) KR20050053673A (https=)
CN (1) CN100546977C (https=)
AU (1) AU2003271619A1 (https=)
BR (1) BR0314544A (https=)
CA (1) CA2498662A1 (https=)
MX (1) MXPA05003084A (https=)
PL (1) PL374846A1 (https=)
RU (2) RU2005111256A (https=)
SG (1) SG165995A1 (https=)
WO (1) WO2004026815A2 (https=)
ZA (1) ZA200501913B (https=)

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JP2006518738A (ja) * 2003-02-12 2006-08-17 トランス テック ファーマ,インコーポレイテッド 治療薬としての置換アゾール誘導体
CA2520763A1 (en) * 2003-04-03 2004-10-21 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
RS50589B (sr) * 2003-12-23 2010-05-07 H. Lundbeck A/S. 2-(1h-indolilsulfanil)-benzil amin derivati kao ssri
US7304086B2 (en) * 2004-02-05 2007-12-04 Probiodrug Ag Inhibitors of glutaminyl cyclase
EP1765311A4 (en) 2004-03-16 2009-04-29 Univ California REDUCTION OF NEPHROPATHY WITH INHIBITORS OF SOLUBLE EPOXY HYDROLASE AND EPOXYEICOSANOIDS
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
WO2005113534A2 (en) * 2004-05-12 2005-12-01 Schering Corporation Cxcr1 and cxcr2 chemokine antagonists
AR052308A1 (es) * 2004-07-16 2007-03-14 Lundbeck & Co As H Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto
US7662910B2 (en) * 2004-10-20 2010-02-16 The Regents Of The University Of California Inhibitors for the soluble epoxide hydrolase
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