PL374846A1 - New compounds for the inhibition of rotamases and use thereof - Google Patents
New compounds for the inhibition of rotamases and use thereofInfo
- Publication number
- PL374846A1 PL374846A1 PL03374846A PL37484603A PL374846A1 PL 374846 A1 PL374846 A1 PL 374846A1 PL 03374846 A PL03374846 A PL 03374846A PL 37484603 A PL37484603 A PL 37484603A PL 374846 A1 PL374846 A1 PL 374846A1
- Authority
- PL
- Poland
- Prior art keywords
- rotamases
- inhibition
- new compounds
- compounds
- new
- Prior art date
Links
Classifications
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- C—CHEMISTRY; METALLURGY
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- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
- C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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- C07C335/16—Derivatives of thiourea having nitrogen atoms of thiourea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C335/18—Derivatives of thiourea having nitrogen atoms of thiourea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Organic Chemistry (AREA)
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- Epidemiology (AREA)
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- Oncology (AREA)
- Communicable Diseases (AREA)
- Neurology (AREA)
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- Immunology (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Molecular Biology (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Psychology (AREA)
- Gastroenterology & Hepatology (AREA)
- Hospice & Palliative Care (AREA)
- Biotechnology (AREA)
- AIDS & HIV (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP20020020987 EP1402888A1 (en) | 2002-09-18 | 2002-09-18 | The use of substituted carbocyclic compounds as rotamases inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
PL374846A1 true PL374846A1 (en) | 2005-11-14 |
Family
ID=31970282
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL03374846A PL374846A1 (en) | 2002-09-18 | 2003-09-18 | New compounds for the inhibition of rotamases and use thereof |
Country Status (14)
Country | Link |
---|---|
US (2) | US20070054904A1 (xx) |
EP (3) | EP1402888A1 (xx) |
JP (2) | JP2005539072A (xx) |
KR (1) | KR20050053673A (xx) |
CN (1) | CN100546977C (xx) |
AU (1) | AU2003271619A1 (xx) |
BR (1) | BR0314544A (xx) |
CA (1) | CA2498662A1 (xx) |
MX (1) | MXPA05003084A (xx) |
PL (1) | PL374846A1 (xx) |
RU (2) | RU2005111256A (xx) |
SG (1) | SG165995A1 (xx) |
WO (1) | WO2004026815A2 (xx) |
ZA (1) | ZA200501913B (xx) |
Families Citing this family (44)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2006518738A (ja) * | 2003-02-12 | 2006-08-17 | トランス テック ファーマ,インコーポレイテッド | 治療薬としての置換アゾール誘導体 |
AU2004228028B2 (en) | 2003-04-03 | 2009-12-10 | The Regents Of The University Of California | Improved inhibitors for the soluble epoxide hydrolase |
BRPI0417858B1 (pt) * | 2003-12-23 | 2017-10-10 | H. Lundbeck A/S | Derivative compounds of aniline and pharmaceutical composition that understand it |
KR101099206B1 (ko) * | 2004-02-05 | 2011-12-27 | 프로비오드룩 아게 | 신규한 글루타미닐 시클라제 저해제 |
CA2559665A1 (en) | 2004-03-16 | 2005-09-29 | The Regents Of The University Of California | Reducing nephropathy with inhibitors of soluble epoxide hydrolase and epoxyeicosanoids |
US7550499B2 (en) | 2004-05-12 | 2009-06-23 | Bristol-Myers Squibb Company | Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions |
JP2007537272A (ja) * | 2004-05-12 | 2007-12-20 | シェーリング コーポレイション | Cxcr1およびcxcr2ケモカインアンタゴニスト |
AR052308A1 (es) * | 2004-07-16 | 2007-03-14 | Lundbeck & Co As H | Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto |
EP1814875A4 (en) * | 2004-10-20 | 2010-02-17 | Univ California | IMPROVED INHIBITORS OF SOLUBLE HYDROLASE EPOXYDE |
WO2006078621A2 (en) | 2005-01-19 | 2006-07-27 | Bristol-Myers Squibb Company | 2-phenoxy-n- (1, 3 , 4-thiadizol-2-yl) pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders |
EP1888052A2 (en) * | 2005-05-12 | 2008-02-20 | Wisconsin Alumni Research Foundation | Blockade of pin1 prevents cytokine production by activated immune cells |
US7629473B2 (en) * | 2005-06-17 | 2009-12-08 | H. Lundbeck A/S | 2-(1H-indolylsulfanyl)-aryl amine derivatives |
AR054393A1 (es) * | 2005-06-17 | 2007-06-20 | Lundbeck & Co As H | Derivados de benzo(b)furano y benzo(b)tiofeno, composiciones farmaceuticas que los contienen y su uso en la fabricacion de un medicamento para el tratamiento de enfermedades mediadas por la inhibicion de la reabsorcion de neurotransmisores de amina biogenicos. |
WO2007002634A1 (en) | 2005-06-27 | 2007-01-04 | Bristol-Myers Squibb Company | Carbocycle and heterocycle antagonists of p2y1 receptor useful in the treatment of thrombotic conditions |
ATE502924T1 (de) | 2005-06-27 | 2011-04-15 | Bristol Myers Squibb Co | Lineare harnstoffmimetika-antagonisten des p2y1- rezeptors zur behandlung von thromboseleiden |
WO2007002635A2 (en) | 2005-06-27 | 2007-01-04 | Bristol-Myers Squibb Company | C-linked cyclic antagonists of p2y1 receptor useful in the treatment of thrombotic conditions |
AU2006261828A1 (en) | 2005-06-27 | 2007-01-04 | Bristol-Myers Squibb Company | N-linked heterocyclic antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions |
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2002
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2003
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- 2003-09-18 EP EP09007837A patent/EP2100876A3/en not_active Withdrawn
- 2003-09-18 KR KR1020057004693A patent/KR20050053673A/ko not_active Application Discontinuation
- 2003-09-18 PL PL03374846A patent/PL374846A1/xx not_active Application Discontinuation
- 2003-09-18 JP JP2004537125A patent/JP2005539072A/ja not_active Withdrawn
- 2003-09-18 MX MXPA05003084A patent/MXPA05003084A/es not_active Application Discontinuation
- 2003-09-18 BR BR0314544-1A patent/BR0314544A/pt not_active IP Right Cessation
- 2003-09-18 WO PCT/EP2003/010406 patent/WO2004026815A2/en active Application Filing
- 2003-09-18 CN CNB038252651A patent/CN100546977C/zh not_active Expired - Fee Related
- 2003-09-18 EP EP03753427A patent/EP1539683A2/en not_active Ceased
- 2003-09-18 AU AU2003271619A patent/AU2003271619A1/en not_active Abandoned
- 2003-09-18 US US10/528,139 patent/US20070054904A1/en not_active Abandoned
- 2003-09-18 SG SG200702382-3A patent/SG165995A1/en unknown
- 2003-09-18 RU RU2005111256/04A patent/RU2005111256A/ru not_active Application Discontinuation
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2005
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2010
- 2010-09-02 RU RU2010136779/04A patent/RU2010136779A/ru not_active Application Discontinuation
- 2010-09-29 JP JP2010219856A patent/JP2011037869A/ja active Pending
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ZA200501913B (en) | 2005-07-27 |
RU2005111256A (ru) | 2006-10-27 |
EP1539683A2 (en) | 2005-06-15 |
WO2004026815A2 (en) | 2004-04-01 |
US20070054904A1 (en) | 2007-03-08 |
EP1402888A1 (en) | 2004-03-31 |
AU2003271619A1 (en) | 2004-04-08 |
MXPA05003084A (es) | 2005-11-17 |
CA2498662A1 (en) | 2004-04-01 |
SG165995A1 (en) | 2010-11-29 |
CN1701061A (zh) | 2005-11-23 |
JP2011037869A (ja) | 2011-02-24 |
WO2004026815A3 (en) | 2004-12-02 |
KR20050053673A (ko) | 2005-06-08 |
JP2005539072A (ja) | 2005-12-22 |
CN100546977C (zh) | 2009-10-07 |
RU2010136779A (ru) | 2012-03-10 |
EP2100876A2 (en) | 2009-09-16 |
BR0314544A (pt) | 2005-08-16 |
EP2100876A3 (en) | 2010-02-24 |
US20110065760A1 (en) | 2011-03-17 |
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