AU2003271619A1 - Phenol derivatives and their use as rotamase inhibitors - Google Patents

Phenol derivatives and their use as rotamase inhibitors Download PDF

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Publication number
AU2003271619A1
AU2003271619A1 AU2003271619A AU2003271619A AU2003271619A1 AU 2003271619 A1 AU2003271619 A1 AU 2003271619A1 AU 2003271619 A AU2003271619 A AU 2003271619A AU 2003271619 A AU2003271619 A AU 2003271619A AU 2003271619 A1 AU2003271619 A1 AU 2003271619A1
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Australia
Prior art keywords
phenyl
hydroxy
chloro
urea
benzylamino
Prior art date
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Abandoned
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AU2003271619A
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English (en)
Inventor
Claudia Christner
Christoph Gibson
Gerd Hummel
Laurence Jobron
Jochen Knolle
Frank Osterkamp
Dirk Scharn
Mike Schutkowski
Roland Stragies
Thomas Tradler
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Jerini AG
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Jerini AG
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Publication of AU2003271619A1 publication Critical patent/AU2003271619A1/en
Abandoned legal-status Critical Current

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    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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AU2003271619A 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors Abandoned AU2003271619A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20020020987 EP1402888A1 (en) 2002-09-18 2002-09-18 The use of substituted carbocyclic compounds as rotamases inhibitors
EP02020987.0 2002-09-18
PCT/EP2003/010406 WO2004026815A2 (en) 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors

Publications (1)

Publication Number Publication Date
AU2003271619A1 true AU2003271619A1 (en) 2004-04-08

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ID=31970282

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Application Number Title Priority Date Filing Date
AU2003271619A Abandoned AU2003271619A1 (en) 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors

Country Status (14)

Country Link
US (2) US20070054904A1 (https=)
EP (3) EP1402888A1 (https=)
JP (2) JP2005539072A (https=)
KR (1) KR20050053673A (https=)
CN (1) CN100546977C (https=)
AU (1) AU2003271619A1 (https=)
BR (1) BR0314544A (https=)
CA (1) CA2498662A1 (https=)
MX (1) MXPA05003084A (https=)
PL (1) PL374846A1 (https=)
RU (2) RU2005111256A (https=)
SG (1) SG165995A1 (https=)
WO (1) WO2004026815A2 (https=)
ZA (1) ZA200501913B (https=)

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CA2514363A1 (en) * 2003-02-12 2004-08-26 Transtech Pharma, Inc. Substituted azole derivatives as therapeutic agents
US20050026844A1 (en) 2003-04-03 2005-02-03 Regents Of The University Of California Inhibitors for the soluble epoxide hydrolase
WO2005089380A2 (en) 2004-03-16 2005-09-29 The Regents Of The University Of California Reducing nephropathy with inhibitors of soluble epoxide hydrolase and epoxyeicosanoids
PL1701940T3 (pl) * 2003-12-23 2008-11-28 H Lundbeck As Pochodne 2-(1H-indolilosulfanylo)benzyloaminy jako SSRI
CA2554809C (en) * 2004-02-05 2014-04-29 Probiodrug Ag Novel n-alkyl thiourea- and thioamide-substituted imidazolyl inhibitors of glutaminyl cyclase
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
CN1984899B (zh) * 2004-05-12 2011-07-27 先灵公司 Cxcr1和cxcr2趋化因子拮抗剂
AR052308A1 (es) * 2004-07-16 2007-03-14 Lundbeck & Co As H Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto
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EP1402888A1 (en) 2004-03-31
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