RU2005103618A - Ингибирующие циклооксигеназу-2 (цог-2) производные пиридина - Google Patents

Ингибирующие циклооксигеназу-2 (цог-2) производные пиридина Download PDF

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RU2005103618A
RU2005103618A RU2005103618/04A RU2005103618A RU2005103618A RU 2005103618 A RU2005103618 A RU 2005103618A RU 2005103618/04 A RU2005103618/04 A RU 2005103618/04A RU 2005103618 A RU2005103618 A RU 2005103618A RU 2005103618 A RU2005103618 A RU 2005103618A
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Russia
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alkyl
methyl
group
phenyl
methylsulfonyl
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RU2005103618/04A
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English (en)
Russian (ru)
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Пол БЕСУИК (GB)
Пол БЕСУИК
Сэндип МОДИ (GB)
Сэндип МОДИ
Нил ПЕГГ (GB)
Нил ПЕГГ
Джон СКИДМОР (GB)
Джон Скидмор
Мартин СУОРБРИК (GB)
Мартин СУОРБРИК
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Глаксо Груп Лимитед (GB)
Глаксо Груп Лимитед
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Publication of RU2005103618A publication Critical patent/RU2005103618A/ru

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
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    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Molecular Biology (AREA)
  • Psychology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • AIDS & HIV (AREA)
  • Transplantation (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
RU2005103618/04A 2002-09-16 2003-09-12 Ингибирующие циклооксигеназу-2 (цог-2) производные пиридина RU2005103618A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0221443.5A GB0221443D0 (en) 2002-09-16 2002-09-16 Pyridine derivates
GB0221443.5 2002-09-16

Publications (1)

Publication Number Publication Date
RU2005103618A true RU2005103618A (ru) 2005-10-27

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RU2005103618/04A RU2005103618A (ru) 2002-09-16 2003-09-12 Ингибирующие циклооксигеназу-2 (цог-2) производные пиридина

Country Status (24)

Country Link
US (1) US7446117B2 (enExample)
EP (1) EP1546107B1 (enExample)
JP (1) JP4630063B2 (enExample)
KR (1) KR20050046782A (enExample)
CN (1) CN1681788A (enExample)
AR (1) AR041246A1 (enExample)
AT (1) ATE462694T1 (enExample)
AU (1) AU2003276063A1 (enExample)
BR (1) BR0313718A (enExample)
CA (1) CA2493497A1 (enExample)
DE (1) DE60331931D1 (enExample)
ES (1) ES2343316T3 (enExample)
GB (1) GB0221443D0 (enExample)
IL (1) IL166460A0 (enExample)
IS (1) IS7659A (enExample)
MA (1) MA27436A1 (enExample)
MX (1) MXPA05002886A (enExample)
NO (1) NO20050662L (enExample)
NZ (1) NZ538201A (enExample)
PL (1) PL376023A1 (enExample)
RU (1) RU2005103618A (enExample)
TW (1) TW200404541A (enExample)
WO (1) WO2004024691A1 (enExample)
ZA (1) ZA200501174B (enExample)

Families Citing this family (21)

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DE60305053T2 (de) 2002-08-19 2006-08-31 Glaxo Group Ltd., Greenford Pyrimidinderivate als selektive cox-2-inhibitoren
GB0221443D0 (en) 2002-09-16 2002-10-23 Glaxo Group Ltd Pyridine derivates
WO2005007627A1 (ja) * 2003-07-18 2005-01-27 Nihon Nohyaku Co., Ltd. フェニルピリジン誘導体、その中間体及びこれを有効成分とする除草剤
SI1945632T1 (sl) 2005-11-08 2014-03-31 Vertex Pharmaceuticals Incorporated Heterocikliäśni modulatorji za prenaĺ alce z atp-vezavno kaseto
NZ581259A (en) 2007-05-09 2012-07-27 Vertex Pharma Modulators of cystic fibrosis transmembrane conductance regulator
JP5301557B2 (ja) * 2007-12-04 2013-09-25 エフ．ホフマン−ラ ロシュ アーゲー イソオキサゾロ−ピリジン誘導体
AU2008333845C1 (en) 2007-12-07 2014-01-16 Vertex Pharmaceuticals Incorporated Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3] dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid
SI2639224T1 (sl) * 2007-12-07 2016-12-30 Vertex Pharmaceuticals Incorporated Postopek za pripravo cikloalkilkarboksiamido-piridinskih benzojskih kislin
CN102245573B (zh) 2008-02-28 2013-11-20 沃泰克斯药物股份有限公司 作为cftr调节剂的杂芳基衍生物
WO2010017055A2 (en) 2008-08-06 2010-02-11 Lead Therapeutics, Inc. Dihydropyridophthalazinone inhibitors of poly(adp-ribose)polymerase (parp)
WO2010046780A2 (en) * 2008-10-22 2010-04-29 Institut Pasteur Korea Anti viral compounds
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