PT99064A - Processo para a preparacao de analogos de anel condensado de heterociclos nao aromaticos que contem azoto - Google Patents

Processo para a preparacao de analogos de anel condensado de heterociclos nao aromaticos que contem azoto Download PDF

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Publication number
PT99064A
PT99064A PT99064A PT9906491A PT99064A PT 99064 A PT99064 A PT 99064A PT 99064 A PT99064 A PT 99064A PT 9906491 A PT9906491 A PT 9906491A PT 99064 A PT99064 A PT 99064A
Authority
PT
Portugal
Prior art keywords
alkyl
formula
compound
phenyl
amino
Prior art date
Application number
PT99064A
Other languages
English (en)
Portuguese (pt)
Inventor
Manoj C Desai
Harry R Howard
Terry J Rosen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT99064A publication Critical patent/PT99064A/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Eye Examination Apparatus (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Electroluminescent Light Sources (AREA)
  • Polyoxymethylene Polymers And Polymers With Carbon-To-Carbon Bonds (AREA)
PT99064A 1990-09-28 1991-09-26 Processo para a preparacao de analogos de anel condensado de heterociclos nao aromaticos que contem azoto PT99064A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59042390A 1990-09-28 1990-09-28

Publications (1)

Publication Number Publication Date
PT99064A true PT99064A (pt) 1992-08-31

Family

ID=24362216

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99064A PT99064A (pt) 1990-09-28 1991-09-26 Processo para a preparacao de analogos de anel condensado de heterociclos nao aromaticos que contem azoto

Country Status (22)

Country Link
EP (1) EP0550635B1 (forum.php)
JP (1) JPH0772175B2 (forum.php)
CN (1) CN1060285A (forum.php)
AT (1) ATE121389T1 (forum.php)
AU (1) AU651145B2 (forum.php)
BR (1) BR9106905A (forum.php)
CA (1) CA2089736A1 (forum.php)
CZ (1) CZ387492A3 (forum.php)
DE (1) DE69109125T2 (forum.php)
DK (1) DK0550635T3 (forum.php)
ES (1) ES2071334T3 (forum.php)
FI (1) FI931370A7 (forum.php)
HU (1) HUT68667A (forum.php)
IE (1) IE66042B1 (forum.php)
IL (1) IL99525A0 (forum.php)
MX (1) MX9101274A (forum.php)
NO (1) NO931151L (forum.php)
PT (1) PT99064A (forum.php)
TW (1) TW199144B (forum.php)
WO (1) WO1992006079A1 (forum.php)
YU (1) YU159291A (forum.php)
ZA (1) ZA917744B (forum.php)

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US5387595A (en) * 1992-08-26 1995-02-07 Merck & Co., Inc. Alicyclic compounds as tachykinin receptor antagonists
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DK0675886T3 (da) * 1992-12-10 2000-09-18 Pfizer Aminomethylensubstituerede ikke-aromatiske heterocykler og deres anvendelse som substance P-antagonister
US5830854A (en) * 1992-12-14 1998-11-03 Merck Sharp & Dohme, Limited Method of treating cystic fibrosis using a tachykinin receptor antagonist
US5340826A (en) * 1993-02-04 1994-08-23 Pfizer Inc. Pharmaceutical agents for treatment of urinary incontinence
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US5854262A (en) * 1993-10-07 1998-12-29 Pfizer Inc. Aminomethylene substituted non-aromatic heterocycles and use as substance P antagonists
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Also Published As

Publication number Publication date
AU651145B2 (en) 1994-07-14
EP0550635B1 (en) 1995-04-19
IE913396A1 (en) 1992-04-08
JPH06501267A (ja) 1994-02-10
HUT68667A (en) 1995-07-28
HU9300898D0 (en) 1993-06-28
ZA917744B (en) 1993-03-29
BR9106905A (pt) 1993-08-17
FI931370L (fi) 1993-03-26
DK0550635T3 (da) 1995-09-04
CA2089736A1 (en) 1992-03-29
ATE121389T1 (de) 1995-05-15
MX9101274A (es) 1992-05-04
EP0550635A1 (en) 1993-07-14
FI931370A0 (fi) 1993-03-26
ES2071334T3 (es) 1995-06-16
NO931151D0 (no) 1993-03-26
CZ387492A3 (en) 1994-02-16
DE69109125T2 (de) 1995-09-28
AU8746391A (en) 1992-04-28
TW199144B (forum.php) 1993-02-01
FI931370A7 (fi) 1993-03-26
YU159291A (sh) 1994-01-20
IE66042B1 (en) 1995-12-13
JPH0772175B2 (ja) 1995-08-02
NO931151L (no) 1993-03-26
DE69109125D1 (de) 1995-05-24
WO1992006079A1 (en) 1992-04-16
CN1060285A (zh) 1992-04-15
IL99525A0 (en) 1992-08-18

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