OA12522A - Novel tiotropium-containing inhalation powder. - Google Patents

Novel tiotropium-containing inhalation powder. Download PDF

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Publication number
OA12522A
OA12522A OA1200300108A OA1200300108A OA12522A OA 12522 A OA12522 A OA 12522A OA 1200300108 A OA1200300108 A OA 1200300108A OA 1200300108 A OA1200300108 A OA 1200300108A OA 12522 A OA12522 A OA 12522A
Authority
OA
OAPI
Prior art keywords
inhalation
excipient
powder
tiotropium
mixture
Prior art date
Application number
OA1200300108A
Other languages
English (en)
French (fr)
Inventor
Michael Walz
Georg Boeck
Rolf Dorr
Karoline Bechtold-Peters
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659578&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA12522(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of OA12522A publication Critical patent/OA12522A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Otolaryngology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
OA1200300108A 2000-10-12 2001-09-28 Novel tiotropium-containing inhalation powder. OA12522A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050635 2000-10-12

Publications (1)

Publication Number Publication Date
OA12522A true OA12522A (en) 2006-05-30

Family

ID=7659578

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200300108A OA12522A (en) 2000-10-12 2001-09-28 Novel tiotropium-containing inhalation powder.

Country Status (49)

Country Link
US (4) US7070800B2 (nl)
EP (2) EP1292281B1 (nl)
JP (1) JP3870159B2 (nl)
KR (1) KR100488644B1 (nl)
CN (1) CN1210017C (nl)
AP (1) AP1712A (nl)
AR (1) AR031819A1 (nl)
AT (1) ATE275391T1 (nl)
AU (1) AU757008B2 (nl)
BG (1) BG65753B1 (nl)
BR (1) BR0107304A (nl)
CA (1) CA2395653C (nl)
CR (1) CR6937A (nl)
CU (1) CU23284B7 (nl)
CZ (1) CZ301465B6 (nl)
DE (1) DE50103551C5 (nl)
DK (1) DK1292281T3 (nl)
DZ (1) DZ3477A1 (nl)
EA (1) EA004034B1 (nl)
EC (2) ECSP024268A (nl)
EE (1) EE04414B1 (nl)
EG (1) EG24139A (nl)
ES (1) ES2227268T3 (nl)
GE (1) GEP20063865B (nl)
HK (1) HK1051812A1 (nl)
HR (1) HRP20020437B1 (nl)
HU (1) HU226982B1 (nl)
IL (2) IL149984A0 (nl)
IS (1) IS2360B (nl)
MA (1) MA25843A1 (nl)
ME (2) ME00245B (nl)
MX (1) MXPA02005666A (nl)
MY (1) MY123544A (nl)
NO (1) NO331956B1 (nl)
NZ (1) NZ519406A (nl)
OA (1) OA12522A (nl)
PE (1) PE20020577A1 (nl)
PL (1) PL200063B1 (nl)
PT (1) PT1292281E (nl)
RS (1) RS50197B (nl)
SA (1) SA01220460B1 (nl)
SI (1) SI1292281T1 (nl)
SK (1) SK285389B6 (nl)
TR (1) TR200402367T4 (nl)
TW (1) TWI285553B (nl)
UA (1) UA72014C2 (nl)
UY (1) UY26959A1 (nl)
WO (1) WO2002030389A1 (nl)
ZA (1) ZA200204378B (nl)

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