NO343370B1 - Bisykliske heterosykliske forbindelser som FGFR-inhibitorer, farmasøytisk sammensetning og terapeutisk anvendelse - Google Patents

Bisykliske heterosykliske forbindelser som FGFR-inhibitorer, farmasøytisk sammensetning og terapeutisk anvendelse Download PDF

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Publication number
NO343370B1
NO343370B1 NO20092657A NO20092657A NO343370B1 NO 343370 B1 NO343370 B1 NO 343370B1 NO 20092657 A NO20092657 A NO 20092657A NO 20092657 A NO20092657 A NO 20092657A NO 343370 B1 NO343370 B1 NO 343370B1
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Norway
Prior art keywords
phenyl
alkyl
pyridin
groups
ethyl
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Application number
NO20092657A
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English (en)
Norwegian (no)
Other versions
NO20092657L (no
Inventor
Valerio Berdini
Gordon Saxty
Michael Alistair O'brien
Maria Grazia Carr
Adrian Liam Gill
Miles Stuart Congreve
Gilbert Ebai Besong
Owen Callaghan
Charlotte Mary Griffiths-Jones
Andrew Madin
Christopher William Murray
Rajdeep Kaur Nijjar
Andrew Pike
Richard David Taylor
Emma Vickerstaffe
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Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0625826A external-priority patent/GB0625826D0/en
Priority claimed from GB0720000A external-priority patent/GB0720000D0/en
Application filed by Astex Therapeutics Ltd filed Critical Astex Therapeutics Ltd
Publication of NO20092657L publication Critical patent/NO20092657L/no
Publication of NO343370B1 publication Critical patent/NO343370B1/no

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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NO20092657A 2006-12-22 2009-07-13 Bisykliske heterosykliske forbindelser som FGFR-inhibitorer, farmasøytisk sammensetning og terapeutisk anvendelse NO343370B1 (no)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US87154306P 2006-12-22 2006-12-22
GB0625826A GB0625826D0 (en) 2006-12-22 2006-12-22 New compounds
US97958707P 2007-10-12 2007-10-12
GB0720000A GB0720000D0 (en) 2007-10-12 2007-10-12 New compounds
US98103907P 2007-10-18 2007-10-18
PCT/GB2007/004934 WO2008078091A1 (en) 2006-12-22 2007-12-21 Bicyclic heterocyclic compounds as fgfr inhibitors

Publications (2)

Publication Number Publication Date
NO20092657L NO20092657L (no) 2009-09-17
NO343370B1 true NO343370B1 (no) 2019-02-11

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NO20092657A NO343370B1 (no) 2006-12-22 2009-07-13 Bisykliske heterosykliske forbindelser som FGFR-inhibitorer, farmasøytisk sammensetning og terapeutisk anvendelse

Country Status (11)

Country Link
US (1) US8895745B2 (index.php)
EP (1) EP2114941B1 (index.php)
JP (1) JP5442448B2 (index.php)
CN (1) CN101679408B (index.php)
AR (1) AR064491A1 (index.php)
AU (1) AU2007337886C1 (index.php)
CA (1) CA2672172C (index.php)
HR (1) HRP20150642T1 (index.php)
MX (1) MX2009006706A (index.php)
NO (1) NO343370B1 (index.php)
WO (1) WO2008078091A1 (index.php)

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