NO328580B1 - 4-(2-butylamino)-2,7-dimetyl-8-(2-metyl-6-metoksypyrid-3-yl)pyrazolo-[1,5-A]-1,3,5-triazin, et farmasoytisk akseptabelt promedikament derav, farmasoytisk preparat, anvendelse av forbindelsen samt fremstilt gjenstand omfattende denne - Google Patents
4-(2-butylamino)-2,7-dimetyl-8-(2-metyl-6-metoksypyrid-3-yl)pyrazolo-[1,5-A]-1,3,5-triazin, et farmasoytisk akseptabelt promedikament derav, farmasoytisk preparat, anvendelse av forbindelsen samt fremstilt gjenstand omfattende denne Download PDFInfo
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- NO328580B1 NO328580B1 NO20034023A NO20034023A NO328580B1 NO 328580 B1 NO328580 B1 NO 328580B1 NO 20034023 A NO20034023 A NO 20034023A NO 20034023 A NO20034023 A NO 20034023A NO 328580 B1 NO328580 B1 NO 328580B1
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- compound
- prodrug
- pharmaceutically acceptable
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27540301P | 2001-03-13 | 2001-03-13 | |
| PCT/US2002/006837 WO2002072202A1 (fr) | 2001-03-13 | 2002-03-06 | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, ses enantiomeres et sels pharmaceutiquement acceptables en tant que ligands du recepteur de la corticoliberine |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20034023L NO20034023L (no) | 2003-09-11 |
| NO20034023D0 NO20034023D0 (no) | 2003-09-11 |
| NO328580B1 true NO328580B1 (no) | 2010-03-22 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| NO20034023A NO328580B1 (no) | 2001-03-13 | 2003-09-11 | 4-(2-butylamino)-2,7-dimetyl-8-(2-metyl-6-metoksypyrid-3-yl)pyrazolo-[1,5-A]-1,3,5-triazin, et farmasoytisk akseptabelt promedikament derav, farmasoytisk preparat, anvendelse av forbindelsen samt fremstilt gjenstand omfattende denne |
Country Status (36)
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| EP (1) | EP1368094B1 (fr) |
| JP (1) | JP4549630B2 (fr) |
| KR (1) | KR100875595B1 (fr) |
| CN (1) | CN100427093C (fr) |
| AR (1) | AR032986A1 (fr) |
| AT (1) | ATE355102T1 (fr) |
| AU (1) | AU2002245605B2 (fr) |
| BG (1) | BG66331B1 (fr) |
| BR (1) | BR0208357A (fr) |
| CA (1) | CA2440553C (fr) |
| CY (1) | CY1106607T1 (fr) |
| CZ (1) | CZ20032481A3 (fr) |
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| ES (1) | ES2282401T3 (fr) |
| GE (1) | GEP20053608B (fr) |
| HK (1) | HK1057182A1 (fr) |
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| HU (1) | HU229317B1 (fr) |
| IL (2) | IL157615A0 (fr) |
| IS (1) | IS2839B (fr) |
| MX (1) | MXPA03008185A (fr) |
| MY (1) | MY146935A (fr) |
| NO (1) | NO328580B1 (fr) |
| NZ (1) | NZ528207A (fr) |
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| US7094782B1 (en) * | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
| HU229317B1 (en) * | 2001-03-13 | 2013-10-28 | Bristol Myers Squibb Pharma Co | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine derivatives, and enantiomers of the same az cortikotropine releasing factor (cfr) ligands |
| FR2842809A1 (fr) * | 2002-07-26 | 2004-01-30 | Greenpharma Sas | NOUVELLES PYRAZOLO[1,5-a]-1,3,5-TRIAZINES SUBSTITUEES ET LEURS ANALOGUES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, UTILISATION A TITRE DE MEDICAMENT ET PROCEDES POUR LEUR PREPARATION |
| AR041470A1 (es) * | 2002-10-17 | 2005-05-18 | Upjohn Co | Compuestos de pirrolo (1,2 - b) piridazina y sus usos |
| US7329658B2 (en) | 2003-02-06 | 2008-02-12 | Pfizer Inc | Cannabinoid receptor ligands and uses thereof |
| US7176210B2 (en) * | 2003-02-10 | 2007-02-13 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
| US7041671B2 (en) | 2003-04-02 | 2006-05-09 | Pfizer Inc | Pyrrolo[1,2-b]pyridazine compounds and their uses |
| US7056920B2 (en) | 2003-04-04 | 2006-06-06 | Pfizer Inc | Pyrrolo[1,2-B]pyridazine compounds and their uses |
| US7034023B2 (en) * | 2003-04-04 | 2006-04-25 | Pfizer Inc | Pyrrolo[1,2-B]pyridazine compounds and their uses |
| BRPI0409444A (pt) * | 2003-04-15 | 2006-04-18 | Pharmacia & Upjohn Co Llc | compostos de pirrolo[1,2-b]piridazina e suas utilizações |
| US7153961B2 (en) | 2003-11-25 | 2006-12-26 | Bristol-Myers Squibb Pharma Co. | Salt and crystalline form thereof of a corticotropin releasing factor receptor antagonist |
| US7208596B2 (en) * | 2003-11-25 | 2007-04-24 | Bristol-Myers Squibb Pharma Company | Processes for the preparation of pyrazolo[1,5-a]-1,3,5-triazines and intermediates thereof |
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| PT1049699E (pt) * | 1998-01-28 | 2004-08-31 | Bristol Myers Squibb Pharma Co | Pirazolotriazinas como antagonistas de flc |
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