HRP20030822B1 - 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands - Google Patents

4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands

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Publication number
HRP20030822B1
HRP20030822B1 HR20030822A HRP20030822A HRP20030822B1 HR P20030822 B1 HRP20030822 B1 HR P20030822B1 HR 20030822 A HR20030822 A HR 20030822A HR P20030822 A HRP20030822 A HR P20030822A HR P20030822 B1 HRP20030822 B1 HR P20030822B1
Authority
HR
Croatia
Prior art keywords
pyrazolo
pharmaceutically acceptable
methoxypyrid
butylamino
triazine
Prior art date
Application number
HR20030822A
Other languages
English (en)
Croatian (hr)
Inventor
J. Gilligan Paul
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Publication of HRP20030822A2 publication Critical patent/HRP20030822A2/xx
Publication of HRP20030822B1 publication Critical patent/HRP20030822B1/xx

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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HR20030822A 2001-03-13 2003-10-10 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands HRP20030822B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27540301P 2001-03-13 2001-03-13
PCT/US2002/006837 WO2002072202A1 (fr) 2001-03-13 2002-03-06 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, ses enantiomeres et sels pharmaceutiquement acceptables en tant que ligands du recepteur de la corticoliberine

Publications (2)

Publication Number Publication Date
HRP20030822A2 HRP20030822A2 (en) 2004-04-30
HRP20030822B1 true HRP20030822B1 (en) 2008-01-31

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HR20030822A HRP20030822B1 (en) 2001-03-13 2003-10-10 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl)pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands

Country Status (36)

Country Link
US (4) US20030125330A1 (fr)
EP (1) EP1368094B1 (fr)
JP (1) JP4549630B2 (fr)
KR (1) KR100875595B1 (fr)
CN (1) CN100427093C (fr)
AR (1) AR032986A1 (fr)
AT (1) ATE355102T1 (fr)
AU (1) AU2002245605B2 (fr)
BG (1) BG66331B1 (fr)
BR (1) BR0208357A (fr)
CA (1) CA2440553C (fr)
CY (1) CY1106607T1 (fr)
CZ (1) CZ20032481A3 (fr)
DE (1) DE60218434T2 (fr)
DK (1) DK1368094T3 (fr)
EE (1) EE05433B1 (fr)
ES (1) ES2282401T3 (fr)
GE (1) GEP20053608B (fr)
HK (1) HK1057182A1 (fr)
HR (1) HRP20030822B1 (fr)
HU (1) HU229317B1 (fr)
IL (2) IL157615A0 (fr)
IS (1) IS2839B (fr)
MX (1) MXPA03008185A (fr)
MY (1) MY146935A (fr)
NO (1) NO328580B1 (fr)
NZ (1) NZ528207A (fr)
PL (1) PL208278B1 (fr)
PT (1) PT1368094E (fr)
RS (1) RS50863B (fr)
RU (1) RU2292347C2 (fr)
SK (1) SK287603B6 (fr)
TW (1) TWI257388B (fr)
UA (1) UA74634C2 (fr)
WO (1) WO2002072202A1 (fr)
ZA (1) ZA200306995B (fr)

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BRPI0409444A (pt) * 2003-04-15 2006-04-18 Pharmacia & Upjohn Co Llc compostos de pirrolo[1,2-b]piridazina e suas utilizações
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WO2008036579A1 (fr) * 2006-09-20 2008-03-27 Eli Lilly And Company Thiazole pyrazolopyrimidines convenant comme antagonistes du récepteur du crf1
JP2015516979A (ja) * 2012-04-23 2015-06-18 ホルスボールマッシュマイヤー ニューロケミー ゲーエムベーハーＨｏｌｓｂｏｅｒｍａｓｃｈｍｅｙｅｒ Ｎｅｕｒｏｃｈｅｍｉｅ Ｇｍｂｈ Ｃｒｈ過剰活性を有する患者の治療に用いるためのｃｒｈｒ１アンタゴニスト
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CA2891122C (fr) 2012-11-14 2021-07-20 The Johns Hopkins University Methodes et compositions pour le traitement de la schizophrenie
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KR102079844B1 (ko) * 2016-09-20 2020-02-20 가톨릭대학교 산학협력단 담석 용해제를 포함하는 담낭 질환 치료용 약학 조성물
BR112020002967A2 (pt) 2017-08-14 2020-08-11 Spruce Biosciences, Inc. antagonistas de receptor de fator de liberação de corticotropina
KR20240023691A (ko) 2020-08-12 2024-02-22 스프루스 바이오사이언시스 인코포레이티드 다낭성 난소 증후군을 치료하기 위한 방법 및 조성물
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