RS50863B - 4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin - Google Patents

4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin

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Publication number
RS50863B
RS50863B YUP-715/03A YUP71503A RS50863B RS 50863 B RS50863 B RS 50863B YU P71503 A YUP71503 A YU P71503A RS 50863 B RS50863 B RS 50863B
Authority
RS
Serbia
Prior art keywords
methoxypyrid
pyrazolo
butylamino
triazine
dimethyl
Prior art date
Application number
YUP-715/03A
Other languages
English (en)
Inventor
Paul Gilligan
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Publication of YU71503A publication Critical patent/YU71503A/sh
Publication of RS50863B publication Critical patent/RS50863B/sr

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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Abstract

4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il)pirazolo[1,5-a]-1,3,5-triazin, u kome je amino funkcionalna grupa vezana za grupu koja se, kada se primenjuje sisarima, otcepljuje kako bi se obrazovala aminska funkcionalna grupa ili njegova farmaceutski prihvatljiva so.Prijava sadrži još 9 patentnih zahteva.
YUP-715/03A 2001-03-13 2002-03-06 4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin RS50863B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US27540301P 2001-03-13 2001-03-13

Publications (2)

Publication Number Publication Date
YU71503A YU71503A (sh) 2006-05-25
RS50863B true RS50863B (sr) 2010-08-31

Family

ID=23052141

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-715/03A RS50863B (sr) 2001-03-13 2002-03-06 4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin

Country Status (36)

Country Link
US (4) US20030125330A1 (sr)
EP (1) EP1368094B1 (sr)
JP (1) JP4549630B2 (sr)
KR (1) KR100875595B1 (sr)
CN (1) CN100427093C (sr)
AR (1) AR032986A1 (sr)
AT (1) ATE355102T1 (sr)
AU (1) AU2002245605B2 (sr)
BG (1) BG66331B1 (sr)
BR (1) BR0208357A (sr)
CA (1) CA2440553C (sr)
CY (1) CY1106607T1 (sr)
CZ (1) CZ20032481A3 (sr)
DE (1) DE60218434T2 (sr)
DK (1) DK1368094T3 (sr)
EE (1) EE05433B1 (sr)
ES (1) ES2282401T3 (sr)
GE (1) GEP20053608B (sr)
HK (1) HK1057182A1 (sr)
HR (1) HRP20030822B1 (sr)
HU (1) HU229317B1 (sr)
IL (2) IL157615A0 (sr)
IS (1) IS2839B (sr)
MX (1) MXPA03008185A (sr)
MY (1) MY146935A (sr)
NO (1) NO328580B1 (sr)
NZ (1) NZ528207A (sr)
PL (1) PL208278B1 (sr)
PT (1) PT1368094E (sr)
RS (1) RS50863B (sr)
RU (1) RU2292347C2 (sr)
SK (1) SK287603B6 (sr)
TW (1) TWI257388B (sr)
UA (1) UA74634C2 (sr)
WO (1) WO2002072202A1 (sr)
ZA (1) ZA200306995B (sr)

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WO2002072202A1 (en) * 2001-03-13 2002-09-19 Bristol-Myers Squibb Pharma Company 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands

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