RS50863B - 4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin - Google Patents

4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin

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Publication number
RS50863B
RS50863B YUP-715/03A YUP71503A RS50863B RS 50863 B RS50863 B RS 50863B YU P71503 A YUP71503 A YU P71503A RS 50863 B RS50863 B RS 50863B
Authority
RS
Serbia
Prior art keywords
methoxypyrid
pyrazolo
butylamino
triazine
dimethyl
Prior art date
Application number
YUP-715/03A
Other languages
English (en)
Inventor
Paul Gilligan
Original Assignee
Bristol-Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company
Publication of YU71503A publication Critical patent/YU71503A/sh
Publication of RS50863B publication Critical patent/RS50863B/sr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Abstract

4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il)pirazolo[1,5-a]-1,3,5-triazin, u kome je amino funkcionalna grupa vezana za grupu koja se, kada se primenjuje sisarima, otcepljuje kako bi se obrazovala aminska funkcionalna grupa ili njegova farmaceutski prihvatljiva so.Prijava sadrži još 9 patentnih zahteva.
YUP-715/03A 2001-03-13 2002-03-06 4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin RS50863B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US27540301P 2001-03-13 2001-03-13

Publications (2)

Publication Number Publication Date
YU71503A YU71503A (sh) 2006-05-25
RS50863B true RS50863B (sr) 2010-08-31

Family

ID=23052141

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-715/03A RS50863B (sr) 2001-03-13 2002-03-06 4-(2-butilamino)-2,7-dimetil-8-(2-metil-6-metoksipirid-3-il) pirazolo/1,5a/-1,3,5-triazin,njegovi enantiomeri i farmaceutski prihvatljive soli kao ligandi receptora za faktor koji oslobađa kortikotropin

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US (4) US20030125330A1 (sr)
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JP (1) JP4549630B2 (sr)
KR (1) KR100875595B1 (sr)
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AR (1) AR032986A1 (sr)
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NO (1) NO328580B1 (sr)
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PL (1) PL208278B1 (sr)
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RS (1) RS50863B (sr)
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UA (1) UA74634C2 (sr)
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AR032986A1 (es) 2003-12-03
WO2002072202A1 (en) 2002-09-19
US20030125330A1 (en) 2003-07-03
DK1368094T3 (da) 2007-07-02
SK11572003A3 (sk) 2004-02-03
US20080139567A1 (en) 2008-06-12
BG108189A (bg) 2004-09-30
EP1368094A1 (en) 2003-12-10
MY146935A (en) 2012-10-15
ES2282401T3 (es) 2007-10-16
CA2440553C (en) 2010-06-08
ATE355102T1 (de) 2006-03-15
EP1368094A4 (en) 2004-03-31
HRP20030822A2 (en) 2004-04-30
BG66331B1 (bg) 2013-06-28
CA2440553A1 (en) 2002-09-19
NO20034023L (no) 2003-09-11
HRP20030822B1 (en) 2008-01-31
CZ20032481A3 (cs) 2007-12-27
JP4549630B2 (ja) 2010-09-22
NZ528207A (en) 2006-02-24
KR20030080086A (ko) 2003-10-10
PL208278B1 (pl) 2011-04-29
HK1057182A1 (en) 2004-03-19
US20070054913A1 (en) 2007-03-08
US7358252B2 (en) 2008-04-15
RU2003130093A (ru) 2005-03-20
RU2292347C2 (ru) 2007-01-27
DE60218434T2 (de) 2007-11-08
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PL368644A1 (en) 2005-04-04
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MXPA03008185A (es) 2004-01-29
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