NO316273B1 - Substituerte 6,6-hetero-bicykliske derivater og farmasöytiske preparater inneholdende dem - Google Patents

Substituerte 6,6-hetero-bicykliske derivater og farmasöytiske preparater inneholdende dem Download PDF

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Publication number
NO316273B1
NO316273B1 NO19990892A NO990892A NO316273B1 NO 316273 B1 NO316273 B1 NO 316273B1 NO 19990892 A NO19990892 A NO 19990892A NO 990892 A NO990892 A NO 990892A NO 316273 B1 NO316273 B1 NO 316273B1
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NO
Norway
Prior art keywords
alkyl
compound according
methyl
ethylpropoxy
substituents
Prior art date
Application number
NO19990892A
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English (en)
Norwegian (no)
Other versions
NO990892D0 (no
NO990892L (no
Inventor
Yuhpyng Liang Chen
Original Assignee
Pfizer
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Publication date
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Publication of NO990892D0 publication Critical patent/NO990892D0/no
Publication of NO990892L publication Critical patent/NO990892L/no
Publication of NO316273B1 publication Critical patent/NO316273B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/233—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P5/42—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of mineralocorticosteroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Psychiatry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Nutrition Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
NO19990892A 1996-08-27 1999-02-25 Substituerte 6,6-hetero-bicykliske derivater og farmasöytiske preparater inneholdende dem NO316273B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2465996P 1996-08-27 1996-08-27
PCT/IB1997/000904 WO1998008846A1 (en) 1996-08-27 1997-07-21 Substituted 6,6-hetero-bicyclic derivatives

Publications (3)

Publication Number Publication Date
NO990892D0 NO990892D0 (no) 1999-02-25
NO990892L NO990892L (no) 1999-02-25
NO316273B1 true NO316273B1 (no) 2004-01-05

Family

ID=21821740

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19990892A NO316273B1 (no) 1996-08-27 1999-02-25 Substituerte 6,6-hetero-bicykliske derivater og farmasöytiske preparater inneholdende dem

Country Status (40)

Country Link
EP (1) EP0925298B1 (cs)
JP (1) JP2000502722A (cs)
KR (1) KR100457759B1 (cs)
CN (2) CN1191236C (cs)
AP (1) AP1164A (cs)
AR (2) AR009321A1 (cs)
AT (1) ATE264327T1 (cs)
AU (1) AU726771C (cs)
BG (1) BG64316B1 (cs)
BR (1) BR9711262A (cs)
CA (1) CA2263913C (cs)
CO (1) CO4930259A1 (cs)
CZ (1) CZ67799A3 (cs)
DE (1) DE69728676T2 (cs)
DK (1) DK0925298T3 (cs)
DZ (1) DZ2299A1 (cs)
EA (1) EA002607B1 (cs)
ES (1) ES2216157T3 (cs)
GT (1) GT199700093A (cs)
HR (1) HRP970452A2 (cs)
ID (1) ID18189A (cs)
IL (1) IL128049A (cs)
IS (1) IS4970A (cs)
MY (1) MY132671A (cs)
NO (1) NO316273B1 (cs)
NZ (1) NZ333728A (cs)
OA (1) OA10980A (cs)
PA (1) PA8435001A1 (cs)
PE (1) PE108698A1 (cs)
PL (1) PL331988A1 (cs)
PT (1) PT925298E (cs)
SI (1) SI0925298T1 (cs)
SK (1) SK22599A3 (cs)
TN (1) TNSN97144A1 (cs)
TR (1) TR199900408T2 (cs)
TW (1) TW477787B (cs)
UA (1) UA66345C2 (cs)
WO (1) WO1998008846A1 (cs)
YU (1) YU35697A (cs)
ZA (1) ZA977652B (cs)

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ATE232863T1 (de) 1996-08-06 2003-03-15 Pfizer Substituierte pyrido- oder pyrimidogruppen enthaltende 6,6- oder 6,7-bicyclische derivate
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