NO309474B1 - 4-Aminotetrahydrobenzisoksazol eller -isotiazolforbindelser - Google Patents

4-Aminotetrahydrobenzisoksazol eller -isotiazolforbindelser Download PDF

Info

Publication number
NO309474B1
NO309474B1 NO973948A NO973948A NO309474B1 NO 309474 B1 NO309474 B1 NO 309474B1 NO 973948 A NO973948 A NO 973948A NO 973948 A NO973948 A NO 973948A NO 309474 B1 NO309474 B1 NO 309474B1
Authority
NO
Norway
Prior art keywords
group
tetrahydro
hydrogen
phenyl
benzisoxazole
Prior art date
Application number
NO973948A
Other languages
English (en)
Norwegian (no)
Other versions
NO973948D0 (no
NO973948L (no
Inventor
Erik Falch
Povl Krogsgaard-Larsen
Jens Kristian Perregaard
Bente Froelund
Arne Schousboe
Lenz Sibylle Moltzen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of NO973948D0 publication Critical patent/NO973948D0/no
Publication of NO973948L publication Critical patent/NO973948L/no
Publication of NO309474B1 publication Critical patent/NO309474B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nozzles (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
NO973948A 1995-02-28 1997-08-27 4-Aminotetrahydrobenzisoksazol eller -isotiazolforbindelser NO309474B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK20795 1995-02-28
PCT/DK1996/000084 WO1996026929A1 (en) 1995-02-28 1996-02-28 4-aminotetrahydrobenzisoxazole or -isothiazole compounds

Publications (3)

Publication Number Publication Date
NO973948D0 NO973948D0 (no) 1997-08-27
NO973948L NO973948L (no) 1997-08-27
NO309474B1 true NO309474B1 (no) 2001-02-05

Family

ID=8090951

Family Applications (1)

Application Number Title Priority Date Filing Date
NO973948A NO309474B1 (no) 1995-02-28 1997-08-27 4-Aminotetrahydrobenzisoksazol eller -isotiazolforbindelser

Country Status (30)

Country Link
US (2) US5998613A (pl)
EP (1) EP0812318B1 (pl)
JP (1) JPH11501016A (pl)
KR (1) KR100242675B1 (pl)
CN (1) CN1087290C (pl)
AT (1) ATE317391T1 (pl)
AU (1) AU697610B2 (pl)
BG (1) BG63258B1 (pl)
BR (1) BR9607443A (pl)
CA (1) CA2213127A1 (pl)
CZ (1) CZ290837B6 (pl)
DE (1) DE69635798T2 (pl)
DK (1) DK0812318T3 (pl)
EA (1) EA000380B1 (pl)
EE (1) EE03483B1 (pl)
ES (1) ES2253748T3 (pl)
FI (1) FI973519A7 (pl)
HU (1) HUP9800631A3 (pl)
IL (1) IL117295A (pl)
IS (1) IS2352B (pl)
NO (1) NO309474B1 (pl)
NZ (1) NZ301653A (pl)
PL (1) PL187404B1 (pl)
RO (1) RO119545B1 (pl)
SI (1) SI0812318T1 (pl)
SK (1) SK281879B6 (pl)
TR (1) TR199700873T1 (pl)
UA (1) UA43396C2 (pl)
WO (1) WO1996026929A1 (pl)
ZA (1) ZA961591B (pl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100491282B1 (ko) 1996-07-24 2005-05-24 워너-램버트 캄파니 엘엘씨 통증 치료용 이소부틸가바 및 그의 유도체
GB9622370D0 (en) 1996-10-28 1997-01-08 Merck Sharp & Dohme Therapeutic agents
US20030185754A1 (en) * 2001-01-16 2003-10-02 Genset, S.A. Treatment of CNS disorders using D-amino acid oxidase and D-aspartate oxidase antagonists
US20030166554A1 (en) * 2001-01-16 2003-09-04 Genset, S.A. Treatment of CNS disorders using D-amino acid oxidase and D-aspartate oxidase antagonists
US7417040B2 (en) * 2004-03-01 2008-08-26 Bristol-Myers Squibb Company Fused tricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3
US7378426B2 (en) * 2004-03-01 2008-05-27 Bristol-Myers Squibb Company Fused heterotricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3
BRPI1011729A2 (pt) * 2009-05-05 2016-03-15 Hoffmann La Roche derivados de isoxazol-tiazol como um receptor inverso gaba a agonista para uso no tratamento de distúrbios cognitivos
US8686009B2 (en) 2009-06-25 2014-04-01 Alkermes Pharma Ireland Limited Prodrugs of NH-acidic compounds
CN105758807B (zh) * 2016-02-22 2019-01-29 山东出入境检验检疫局检验检疫技术中心 一种鉴别废润滑油的方法
WO2019173230A1 (en) 2018-03-05 2019-09-12 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2602643C2 (de) * 1976-01-24 1984-12-20 Bayer Ag, 5090 Leverkusen 1,2-Benzisothiazolinone-3, Verfahren zu ihrer Herstellung sowie Arzneimittel
US4411901A (en) * 1981-12-23 1983-10-25 Mead Johnson & Company Benzisothiazole and benzisoxazole piperazine derivatives
US4452799A (en) * 1981-12-23 1984-06-05 Mead Johnson & Company Benzisothiazole and benzisoxazole piperazine derivatives
US4514414A (en) * 1982-10-25 1985-04-30 Smithkline Beckman Corporation N-Substituted pyrrolidineacetic acids and their esters
US4804663A (en) 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
DK288385D0 (da) * 1985-06-26 1985-06-26 Novo Industri As Aminosyrederivater
US5321037A (en) * 1986-12-26 1994-06-14 Sankyo Company, Limited Isoxazole derivatives for use as cerebro-active drugs and central muscle relaxants
ZA879631B (en) * 1986-12-26 1989-08-30 Sankyo Co Centrally-acting muscle relaxants
US5225412A (en) * 1991-04-29 1993-07-06 Hoechst-Roussel Pharmaceuticals Incorporated Benzoisothiazole-and benzisoxazole-3-carboxamides
US5143923B1 (en) * 1991-04-29 1993-11-02 Hoechst-Roussel Pharmaceuticals Incorporated Benzoisothiazole-and benzisoxazole-3-carboxamides

Also Published As

Publication number Publication date
CZ271197A3 (cs) 1998-03-18
WO1996026929A1 (en) 1996-09-06
MX9706280A (es) 1998-06-30
SK281879B6 (sk) 2001-08-06
AU697610B2 (en) 1998-10-15
EP0812318B1 (en) 2006-02-08
FI973519L (fi) 1997-08-27
RO119545B1 (ro) 2004-12-30
PL187404B1 (pl) 2004-07-30
EA199700199A1 (ru) 1998-02-26
DK0812318T3 (da) 2006-06-06
HK1008527A1 (en) 1999-07-30
KR100242675B1 (ko) 2000-03-02
ES2253748T3 (es) 2006-06-01
EE03483B1 (et) 2001-08-15
AU4713196A (en) 1996-09-18
BG63258B1 (bg) 2001-07-31
ATE317391T1 (de) 2006-02-15
BR9607443A (pt) 1998-05-26
SI0812318T1 (sl) 2006-06-30
ZA961591B (en) 1996-08-28
TR199700873T1 (xx) 1998-01-21
NZ301653A (en) 1998-12-23
HUP9800631A3 (en) 1998-12-28
CN1176638A (zh) 1998-03-18
SK115197A3 (en) 1998-02-04
IL117295A0 (en) 1996-06-18
IS2352B (is) 2008-04-15
FI973519A0 (fi) 1997-08-27
EA000380B1 (ru) 1999-06-24
US5998613A (en) 1999-12-07
DE69635798T2 (de) 2006-08-17
IS4542A (is) 1997-08-13
NO973948D0 (no) 1997-08-27
KR19980702546A (ko) 1998-07-15
CZ290837B6 (cs) 2002-10-16
EP0812318A1 (en) 1997-12-17
NO973948L (no) 1997-08-27
UA43396C2 (uk) 2001-12-17
CA2213127A1 (en) 1996-09-06
IL117295A (en) 1999-11-30
CN1087290C (zh) 2002-07-10
HUP9800631A2 (hu) 1998-08-28
PL321956A1 (en) 1998-01-05
US6174909B1 (en) 2001-01-16
BG101894A (bg) 1998-05-29
FI973519A7 (fi) 1997-08-27
EE9700197A (et) 1998-02-16
DE69635798D1 (de) 2006-04-20
JPH11501016A (ja) 1999-01-26

Similar Documents

Publication Publication Date Title
JPH09509155A (ja) プロテアーゼインヒビター
DK2646443T3 (en) CAT-II inhibitors
NO800222L (no) Engangsbleie.
CN106414439B (zh) 作为食欲素受体拮抗剂的哌啶衍生物
NO309474B1 (no) 4-Aminotetrahydrobenzisoksazol eller -isotiazolforbindelser
NO314581B1 (no) Opplösning av aminer
CN116368138B (zh) 氧杂螺环取代的吡咯并吡唑衍生物及其中间体和制备方法
CA2521300A1 (en) Beta-carbolines useful for treating inflammatory disease
EP1735311B1 (en) Beta-carbolines useful for treating inflammatory disease
NO320332B1 (no) Fremgangsmate ved fremstilling av 2-azadihydroksybicyklo [2.2.2]-heptanforbindelser samt L-tartarsyresalter av forbindelsene
DK159679B (da) Analogifremgangsmaade til fremstilling af hydroxyderivater af 1-(p-methoxybenzoyl)-2-pyrrolidon samt beskyttede hydroxyderivater af 1-(p-methoxybenzoyl)-2-pyrrolidon til anvendelse ved fremgangsmaaden
NO762085L (pl)
MXPA97006280A (en) Compounds 4-aminotetrahidrobenzisoxasol oisotia
CA2509225C (en) Indol derivatives and their use as 5-ht ligands
JP2004502694A (ja) チエノピロリジノン
US6649761B2 (en) Process for preparing piperazinepentaneamide HIV protease inhibitors
HU211128A9 (en) Substituted isoxazole and isothiazole derivatives
WO1997005134A1 (fr) Composes heterocycliques pour le traitement de l'ischemie myocardique
CN118930552A (zh) 异苯并呋喃-1(3h)-酮类化合物及其制备方法、药物组合物和用途
CS212736B2 (en) Method of preparing 3h-pyrido-/3,2-e/-1,4-diazepines
JP2641879B2 (ja) 光学活性を有するヒダントイン誘導体の製法
CS268187B2 (en) Method of new tetrahydrobenzothiazolo-quinolines production
NO330342B1 (no) Ny fremgangsmate for fremstilling av imidazolylforbindelser
NZ626745A (en) Cyclic amide derivatives as inhibitors of 11 - beta - hydroxysteroid dehydrogenase and uses thereof
NO842221L (no) Fremgangsmaate til fremstilling av trisubstituerte oksazolidinoner