NO306948B1 - Piperidin- og piperazinderivater, farmasoeytiske preparater som inneholder slike forbindelser, samt anvendelse av forbindelsene til fremstilling av legemidler - Google Patents

Piperidin- og piperazinderivater, farmasoeytiske preparater som inneholder slike forbindelser, samt anvendelse av forbindelsene til fremstilling av legemidler

Info

Publication number
NO306948B1
NO306948B1 NO943616A NO943616A NO306948B1 NO 306948 B1 NO306948 B1 NO 306948B1 NO 943616 A NO943616 A NO 943616A NO 943616 A NO943616 A NO 943616A NO 306948 B1 NO306948 B1 NO 306948B1
Authority
NO
Norway
Prior art keywords
compounds
piperidine
piperazine derivatives
manufacture
pharmaceutical preparations
Prior art date
Application number
NO943616A
Other languages
English (en)
Other versions
NO943616L (no
NO943616D0 (no
Inventor
Henning Boettcher
Christoph Seyfried
Gerd Bartoszyk
Hartmut Greiner
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of NO943616D0 publication Critical patent/NO943616D0/no
Publication of NO943616L publication Critical patent/NO943616L/no
Publication of NO306948B1 publication Critical patent/NO306948B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
NO943616A 1993-09-30 1994-09-29 Piperidin- og piperazinderivater, farmasoeytiske preparater som inneholder slike forbindelser, samt anvendelse av forbindelsene til fremstilling av legemidler NO306948B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4333254A DE4333254A1 (de) 1993-09-30 1993-09-30 Piperidine und Piperazine

Publications (3)

Publication Number Publication Date
NO943616D0 NO943616D0 (no) 1994-09-29
NO943616L NO943616L (no) 1995-03-31
NO306948B1 true NO306948B1 (no) 2000-01-17

Family

ID=6499013

Family Applications (1)

Application Number Title Priority Date Filing Date
NO943616A NO306948B1 (no) 1993-09-30 1994-09-29 Piperidin- og piperazinderivater, farmasoeytiske preparater som inneholder slike forbindelser, samt anvendelse av forbindelsene til fremstilling av legemidler

Country Status (21)

Country Link
US (1) US5532241A (no)
EP (1) EP0648767B1 (no)
JP (2) JP4065034B2 (no)
KR (1) KR100341190B1 (no)
CN (1) CN1056610C (no)
AT (1) ATE153663T1 (no)
AU (1) AU679774B2 (no)
CA (1) CA2133152C (no)
CZ (1) CZ293558B6 (no)
DE (2) DE4333254A1 (no)
DK (1) DK0648767T3 (no)
ES (1) ES2105454T3 (no)
GR (1) GR3024551T3 (no)
HU (1) HU218918B (no)
NO (1) NO306948B1 (no)
PL (1) PL178137B1 (no)
RU (1) RU2132848C1 (no)
SK (1) SK281793B6 (no)
TW (1) TW313569B (no)
UA (1) UA34449C2 (no)
ZA (1) ZA947622B (no)

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US6656950B2 (en) * 2001-04-25 2003-12-02 Wyeth Antidepressant azaheterocyclylmethyl derivatives of 1,4-dioxino[2,3-b]pyridine
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JP4897221B2 (ja) * 2002-12-20 2012-03-14 チバ ホールディング インコーポレーテッド アミン類の合成及びその合成のための中間体
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DE10315285A1 (de) 2003-04-04 2004-10-14 Merck Patent Gmbh Chromenonindole
DE10326939A1 (de) * 2003-06-16 2005-01-05 Merck Patent Gmbh Indol-Derivate
DE10326940A1 (de) * 2003-06-16 2005-01-05 Merck Patent Gmbh Indol-Derivate
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CN102949364A (zh) * 2011-08-30 2013-03-06 天津药物研究院 一种含有效成分盐酸维拉佐酮的缓释片
US9505744B2 (en) 2011-11-23 2016-11-29 Assia Chemical Industries Ltd. Solid state forms of vilazodone and vilazodone hydrochloride
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ITMI20120531A1 (it) 2012-04-02 2013-10-03 Erregierre Spa Procedimento per la preparazione di vilazodone cloridrato
US9969721B2 (en) 2012-04-12 2018-05-15 Alembic Pharmaceuticals Limited Process for the preparation of vilazodone hydrochloride and its amorphous form
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CN102659660B (zh) * 2012-05-11 2014-07-02 杭州和泽医药科技有限公司 3-(4-氯丁基)-1h-吲哚-5-氰基的制备方法及其应用
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TR201702104A2 (tr) 2017-02-13 2018-08-27 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Vi̇lazodon hi̇droklorür farmasöti̇k bi̇leşi̇mleri̇
TR201702103A2 (tr) 2017-02-13 2018-08-27 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Vilazodon hi̇droklorürün tablet formlari
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Also Published As

Publication number Publication date
KR100341190B1 (ko) 2002-11-13
EP0648767B1 (de) 1997-05-28
US5532241A (en) 1996-07-02
CZ293558B6 (cs) 2004-06-16
UA34449C2 (uk) 2001-03-15
HU9402806D0 (en) 1995-01-30
AU7424494A (en) 1995-04-13
RU2132848C1 (ru) 1999-07-10
NO943616L (no) 1995-03-31
KR950008510A (ko) 1995-04-17
JPH07149762A (ja) 1995-06-13
GR3024551T3 (en) 1997-12-31
TW313569B (no) 1997-08-21
JP4065034B2 (ja) 2008-03-19
HU218918B (hu) 2000-12-28
HUT71833A (en) 1996-02-28
ES2105454T3 (es) 1997-10-16
EP0648767A1 (de) 1995-04-19
CZ237094A3 (en) 1995-04-12
AU679774B2 (en) 1997-07-10
PL305216A1 (en) 1995-04-03
NO943616D0 (no) 1994-09-29
SK281793B6 (sk) 2001-08-06
JP4700017B2 (ja) 2011-06-15
ZA947622B (en) 1995-05-16
DE59402902D1 (de) 1997-07-03
PL178137B1 (pl) 2000-03-31
DE4333254A1 (de) 1995-04-06
JP2007119502A (ja) 2007-05-17
CA2133152A1 (en) 1995-03-31
DK0648767T3 (da) 1997-12-22
CA2133152C (en) 2005-08-30
RU94035660A (ru) 1996-07-20
CN1056610C (zh) 2000-09-20
ATE153663T1 (de) 1997-06-15
SK118494A3 (en) 1995-05-10
CN1106811A (zh) 1995-08-16

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