NO20083057L - Sulfonyl substituerte 1H-indoler som ligander til 5-hydroksytryptamin reseptorer - Google Patents
Sulfonyl substituerte 1H-indoler som ligander til 5-hydroksytryptamin reseptorerInfo
- Publication number
- NO20083057L NO20083057L NO20083057A NO20083057A NO20083057L NO 20083057 L NO20083057 L NO 20083057L NO 20083057 A NO20083057 A NO 20083057A NO 20083057 A NO20083057 A NO 20083057A NO 20083057 L NO20083057 L NO 20083057L
- Authority
- NO
- Norway
- Prior art keywords
- indoles
- ligands
- sulfonyl substituted
- hydroxytryptamine
- receptors
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Pulmonology (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Nutrition Science (AREA)
- Psychology (AREA)
- Vascular Medicine (AREA)
- Rheumatology (AREA)
- Child & Adolescent Psychology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Toxicology (AREA)
- Immunology (AREA)
- Gynecology & Obstetrics (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US75883306P | 2006-01-13 | 2006-01-13 | |
PCT/US2007/060454 WO2007084841A2 (en) | 2006-01-13 | 2007-01-12 | Sulfonyl substituted 1h-indoles as ligands for the 5-hydroxytryptamine receptors |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20083057L true NO20083057L (no) | 2008-10-03 |
Family
ID=38179679
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20083057A NO20083057L (no) | 2006-01-13 | 2008-07-09 | Sulfonyl substituerte 1H-indoler som ligander til 5-hydroksytryptamin reseptorer |
Country Status (16)
Country | Link |
---|---|
US (1) | US7645752B2 (es) |
EP (1) | EP1973876A2 (es) |
JP (1) | JP2009523734A (es) |
KR (1) | KR20080114688A (es) |
CN (1) | CN101370775A (es) |
AU (1) | AU2007206016A1 (es) |
BR (1) | BRPI0706523A2 (es) |
CA (1) | CA2636007A1 (es) |
CR (1) | CR10138A (es) |
EC (1) | ECSP088620A (es) |
IL (1) | IL192695A0 (es) |
MX (1) | MX2008009022A (es) |
NO (1) | NO20083057L (es) |
RU (1) | RU2008127501A (es) |
WO (1) | WO2007084841A2 (es) |
ZA (1) | ZA200806071B (es) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
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CA2721910A1 (en) * | 2008-04-23 | 2009-10-29 | Merck Sharp & Dohme Corp. | Cyclobutyl sulfones as notch sparing gamma secretase inhibitors |
US8598119B2 (en) | 2008-05-27 | 2013-12-03 | Intra-Cellular Therapies, Inc. | Methods and compositions for sleep disorders and other disorders |
ES2646834T3 (es) | 2010-08-20 | 2017-12-18 | Amira Pharmaceuticals, Inc. | Inhibidores de autotaxina y usos de los mismos |
WO2012166415A1 (en) | 2011-05-27 | 2012-12-06 | Amira Pharmaceuticals, Inc. | Heterocyclic autotaxin inhibitors and uses thereof |
EP2968320B1 (en) | 2013-03-15 | 2020-11-11 | Intra-Cellular Therapies, Inc. | Organic compounds |
KR20230058736A (ko) | 2013-12-03 | 2023-05-03 | 인트라-셀룰라 써래피스, 인코퍼레이티드. | 신규한 방법 |
EP3125893B1 (en) | 2014-04-04 | 2023-09-20 | Intra-Cellular Therapies, Inc. | Deuterated heterocycle fused gamma-carbolines as antagonists of 5-ht2a receptors |
WO2016004882A1 (en) | 2014-07-08 | 2016-01-14 | Sunshine Lake Pharma Co., Ltd. | Aromatic heterocyclic derivatives and pharmaceutical applications thereof |
PT3407888T (pt) | 2016-01-26 | 2021-03-19 | Intra Cellular Therapies Inc | Compostos de piridopirroloquinoxalina, suas composições e utilizações |
IL297676B2 (en) | 2016-03-25 | 2023-12-01 | Intra Cellular Therapies Inc | A controlled or delayed release pharmaceutical preparation containing a deuterated compound |
US10654854B2 (en) | 2016-03-28 | 2020-05-19 | Intra-Cellular Therapies, Inc. | Salts and crystals of ITI-007 |
EP3436083A4 (en) | 2016-03-28 | 2019-11-27 | Intra-Cellular Therapies, Inc. | NEW COMPOSITIONS AND METHODS |
JP6997718B2 (ja) | 2016-03-28 | 2022-01-18 | イントラ-セルラー・セラピーズ・インコーポレイテッド | 新規共結晶 |
WO2018071233A1 (en) | 2016-10-12 | 2018-04-19 | Intra-Cellular Therapies, Inc. | Amorphous solid dispersions |
US10961245B2 (en) | 2016-12-29 | 2021-03-30 | Intra-Cellular Therapies, Inc. | Substituted heterocycle fused gamma-carbolines for treatment of central nervous system disorders |
US10906906B2 (en) | 2016-12-29 | 2021-02-02 | Intra-Cellular Therapies, Inc. | Organic compounds |
IL304026A (en) | 2017-03-24 | 2023-08-01 | Intra Cellular Therapies Inc | New preparations and methods |
US11517557B2 (en) * | 2017-07-13 | 2022-12-06 | Tonix Pharmaceuticals Holding Corp. | Analogs of cyclobenzaprine and amitriptyline |
CN111093664B (zh) | 2017-07-26 | 2023-06-02 | 细胞内治疗公司 | 有机化合物 |
IL272249B2 (en) | 2017-07-26 | 2023-11-01 | Intra Cellular Therapies Inc | organic compounds |
CA3094204A1 (en) | 2018-03-16 | 2019-09-19 | Intra-Cellular Therapies, Inc. | Novel methods |
BR112021003838A2 (pt) | 2018-08-31 | 2021-05-18 | Intra-Cellular Therapies, Inc. | métodos novos |
BR112021003655A2 (pt) | 2018-08-31 | 2021-05-18 | Intra-Cellular Therapies, Inc. | métodos novos |
BR112021006488A2 (pt) | 2018-10-05 | 2021-07-06 | Annapurna Bio Inc | compostos e composições para o tratamento de condições associadas com atividade do receptor apj |
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-
2007
- 2007-01-12 CA CA002636007A patent/CA2636007A1/en not_active Abandoned
- 2007-01-12 AU AU2007206016A patent/AU2007206016A1/en not_active Abandoned
- 2007-01-12 WO PCT/US2007/060454 patent/WO2007084841A2/en active Application Filing
- 2007-01-12 JP JP2008550530A patent/JP2009523734A/ja not_active Withdrawn
- 2007-01-12 CN CNA2007800023497A patent/CN101370775A/zh not_active Withdrawn
- 2007-01-12 US US11/622,649 patent/US7645752B2/en not_active Expired - Fee Related
- 2007-01-12 MX MX2008009022A patent/MX2008009022A/es not_active Application Discontinuation
- 2007-01-12 BR BRPI0706523-0A patent/BRPI0706523A2/pt not_active Application Discontinuation
- 2007-01-12 KR KR1020087019566A patent/KR20080114688A/ko not_active Application Discontinuation
- 2007-01-12 RU RU2008127501/04A patent/RU2008127501A/ru not_active Application Discontinuation
- 2007-01-12 EP EP07710091A patent/EP1973876A2/en not_active Withdrawn
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2008
- 2008-07-08 IL IL192695A patent/IL192695A0/en unknown
- 2008-07-09 NO NO20083057A patent/NO20083057L/no not_active Application Discontinuation
- 2008-07-11 EC EC2008008620A patent/ECSP088620A/es unknown
- 2008-07-11 ZA ZA200806071A patent/ZA200806071B/xx unknown
- 2008-07-11 CR CR10138A patent/CR10138A/es not_active Application Discontinuation
Also Published As
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US7645752B2 (en) | 2010-01-12 |
ECSP088620A (es) | 2008-08-29 |
IL192695A0 (en) | 2009-02-11 |
CN101370775A (zh) | 2009-02-18 |
US20070203120A1 (en) | 2007-08-30 |
BRPI0706523A2 (pt) | 2011-01-04 |
JP2009523734A (ja) | 2009-06-25 |
AU2007206016A1 (en) | 2007-07-26 |
RU2008127501A (ru) | 2010-02-20 |
CA2636007A1 (en) | 2007-07-26 |
EP1973876A2 (en) | 2008-10-01 |
WO2007084841A2 (en) | 2007-07-26 |
KR20080114688A (ko) | 2008-12-31 |
ZA200806071B (en) | 2009-04-29 |
MX2008009022A (es) | 2008-09-24 |
CR10138A (es) | 2008-10-03 |
WO2007084841A3 (en) | 2007-09-13 |
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