ZA200806071B - Sulfonyl substituted 1H-indoles as ligands for the 5-hydroxytryptamine receptors - Google Patents

Sulfonyl substituted 1H-indoles as ligands for the 5-hydroxytryptamine receptors

Info

Publication number
ZA200806071B
ZA200806071B ZA200806071A ZA200806071A ZA200806071B ZA 200806071 B ZA200806071 B ZA 200806071B ZA 200806071 A ZA200806071 A ZA 200806071A ZA 200806071 A ZA200806071 A ZA 200806071A ZA 200806071 B ZA200806071 B ZA 200806071B
Authority
ZA
South Africa
Prior art keywords
indoles
ligands
sulfonyl substituted
hydroxytryptamine receptors
hydroxytryptamine
Prior art date
Application number
ZA200806071A
Other languages
English (en)
Inventor
Robert E Mcdevitt
Li Yanfang
Albert J Robichaud
Gavin D Heffernan
Richard D Coghlan
Ronald C Bernotas
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of ZA200806071B publication Critical patent/ZA200806071B/xx

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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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ZA200806071A 2006-01-13 2008-07-11 Sulfonyl substituted 1H-indoles as ligands for the 5-hydroxytryptamine receptors ZA200806071B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75883306P 2006-01-13 2006-01-13

Publications (1)

Publication Number Publication Date
ZA200806071B true ZA200806071B (en) 2009-04-29

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ZA200806071A ZA200806071B (en) 2006-01-13 2008-07-11 Sulfonyl substituted 1H-indoles as ligands for the 5-hydroxytryptamine receptors

Country Status (16)

Country Link
US (1) US7645752B2 (xx)
EP (1) EP1973876A2 (xx)
JP (1) JP2009523734A (xx)
KR (1) KR20080114688A (xx)
CN (1) CN101370775A (xx)
AU (1) AU2007206016A1 (xx)
BR (1) BRPI0706523A2 (xx)
CA (1) CA2636007A1 (xx)
CR (1) CR10138A (xx)
EC (1) ECSP088620A (xx)
IL (1) IL192695A0 (xx)
MX (1) MX2008009022A (xx)
NO (1) NO20083057L (xx)
RU (1) RU2008127501A (xx)
WO (1) WO2007084841A2 (xx)
ZA (1) ZA200806071B (xx)

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US20070203120A1 (en) 2007-08-30
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US7645752B2 (en) 2010-01-12
CN101370775A (zh) 2009-02-18
BRPI0706523A2 (pt) 2011-01-04
EP1973876A2 (en) 2008-10-01
JP2009523734A (ja) 2009-06-25
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AU2007206016A1 (en) 2007-07-26
IL192695A0 (en) 2009-02-11

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