NO20073926L - Pyrazolforbindelser som modulerer aktivitet av CDK-, GSK- og aurorakinaser - Google Patents
Pyrazolforbindelser som modulerer aktivitet av CDK-, GSK- og aurorakinaserInfo
- Publication number
- NO20073926L NO20073926L NO20073926A NO20073926A NO20073926L NO 20073926 L NO20073926 L NO 20073926L NO 20073926 A NO20073926 A NO 20073926A NO 20073926 A NO20073926 A NO 20073926A NO 20073926 L NO20073926 L NO 20073926L
- Authority
- NO
- Norway
- Prior art keywords
- gsk
- cdk
- aurorakinases
- compounds
- pyrazole compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64059704P | 2004-12-30 | 2004-12-30 | |
| US64047504P | 2004-12-30 | 2004-12-30 | |
| GB0428552A GB0428552D0 (en) | 2004-12-30 | 2004-12-30 | Pharmaceutical compounds |
| GB0428554A GB0428554D0 (en) | 2004-12-30 | 2004-12-30 | Pharmaceutical compounds |
| PCT/GB2005/005097 WO2006070195A1 (en) | 2004-12-30 | 2005-12-30 | Pyrazole compounds that modulate the activity of cdk, gsk and aurora kinases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20073926L true NO20073926L (no) | 2007-10-01 |
Family
ID=39495737
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20073926A NO20073926L (no) | 2004-12-30 | 2007-07-26 | Pyrazolforbindelser som modulerer aktivitet av CDK-, GSK- og aurorakinaser |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US8110573B2 (de) |
| EP (2) | EP2395000A1 (de) |
| JP (1) | JP5507049B2 (de) |
| KR (1) | KR101334511B1 (de) |
| AU (1) | AU2005321091B2 (de) |
| BR (1) | BRPI0519759A2 (de) |
| CA (1) | CA2593993C (de) |
| IL (1) | IL183751A0 (de) |
| MX (1) | MX2007008008A (de) |
| NO (1) | NO20073926L (de) |
| NZ (1) | NZ555982A (de) |
| RU (1) | RU2416610C2 (de) |
| TW (1) | TWI427077B (de) |
| WO (1) | WO2006070195A1 (de) |
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| JP5507049B2 (ja) | 2004-12-30 | 2014-05-28 | アステックス、セラピューティックス、リミテッド | 医薬品 |
| KR101411167B1 (ko) | 2005-04-13 | 2014-06-23 | 아스텍스 테라퓨틱스 리미티드 | 하이드록시벤즈아미드 유도체 및 ｈｓｐ90 억제제로서의이의 용도 |
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2005
- 2005-12-30 JP JP2007548898A patent/JP5507049B2/ja not_active Expired - Fee Related
- 2005-12-30 BR BRPI0519759-7A patent/BRPI0519759A2/pt not_active IP Right Cessation
- 2005-12-30 US US11/813,031 patent/US8110573B2/en not_active Expired - Fee Related
- 2005-12-30 EP EP11180160A patent/EP2395000A1/de not_active Withdrawn
- 2005-12-30 KR KR1020077017527A patent/KR101334511B1/ko not_active IP Right Cessation
- 2005-12-30 TW TW094147642A patent/TWI427077B/zh not_active IP Right Cessation
- 2005-12-30 MX MX2007008008A patent/MX2007008008A/es active IP Right Grant
- 2005-12-30 EP EP05823721A patent/EP1833819A1/de not_active Withdrawn
- 2005-12-30 NZ NZ555982A patent/NZ555982A/en not_active IP Right Cessation
- 2005-12-30 AU AU2005321091A patent/AU2005321091B2/en not_active Ceased
- 2005-12-30 WO PCT/GB2005/005097 patent/WO2006070195A1/en active Application Filing
- 2005-12-30 RU RU2007128959/04A patent/RU2416610C2/ru not_active IP Right Cessation
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Also Published As
| Publication number | Publication date |
|---|---|
| TWI427077B (zh) | 2014-02-21 |
| AU2005321091B2 (en) | 2012-04-12 |
| MX2007008008A (es) | 2007-11-12 |
| IL183751A0 (en) | 2007-09-20 |
| US20080132495A1 (en) | 2008-06-05 |
| TW200635918A (en) | 2006-10-16 |
| KR101334511B1 (ko) | 2013-11-29 |
| RU2007128959A (ru) | 2009-02-10 |
| US20120190673A1 (en) | 2012-07-26 |
| NZ555982A (en) | 2011-01-28 |
| AU2005321091A1 (en) | 2006-07-06 |
| BRPI0519759A2 (pt) | 2009-03-10 |
| KR20070094639A (ko) | 2007-09-20 |
| EP1833819A1 (de) | 2007-09-19 |
| JP5507049B2 (ja) | 2014-05-28 |
| CA2593993C (en) | 2014-07-29 |
| JP2008526722A (ja) | 2008-07-24 |
| US8110573B2 (en) | 2012-02-07 |
| WO2006070195A8 (en) | 2006-08-24 |
| CA2593993A1 (en) | 2006-07-06 |
| EP2395000A1 (de) | 2011-12-14 |
| RU2416610C2 (ru) | 2011-04-20 |
| US8778936B2 (en) | 2014-07-15 |
| WO2006070195A1 (en) | 2006-07-06 |
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