NO20051527L - 3-(sulfonamidoetyl) -indol-derivater for anvendelse som glukocorticoid-mimetica ved behandling av inflammatoriske, allergiske og proliferative sykdommer. - Google Patents

3-(sulfonamidoetyl) -indol-derivater for anvendelse som glukocorticoid-mimetica ved behandling av inflammatoriske, allergiske og proliferative sykdommer.

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Publication number
NO20051527L
NO20051527L NO20051527A NO20051527A NO20051527L NO 20051527 L NO20051527 L NO 20051527L NO 20051527 A NO20051527 A NO 20051527A NO 20051527 A NO20051527 A NO 20051527A NO 20051527 L NO20051527 L NO 20051527L
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NO
Norway
Prior art keywords
allergic
inflammatory
sulfonamidoethyl
treatment
proliferative diseases
Prior art date
Application number
NO20051527A
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English (en)
Other versions
NO20051527D0 (no
Inventor
Daniel Richard Marshall
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of NO20051527D0 publication Critical patent/NO20051527D0/no
Publication of NO20051527L publication Critical patent/NO20051527L/no

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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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  • Chemical & Material Sciences (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
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Abstract

Forbindelser med formel (I) hvor R\ R\ R^ R^ R\ R', R', R*, R', R'°, X og Y er som definert heri eller en tautomer, prodmg, solvat eller salt derav; farmasøytiske preparater inneholdende slike forbindelser og metoder for å modulere glukokortikoidreseptorfunksjonen og metoder for behandling av sykdomtilstander eller tilstander mediert av glukokortikoidreseptorfunksjonen eller karakterisert ved infiammatoriske, allergiske eller prohferative prosesser hos en pasient ved anvendelse av disse forbindelser.
NO20051527A 2002-08-29 2005-03-22 3-(sulfonamidoetyl) -indol-derivater for anvendelse som glukocorticoid-mimetica ved behandling av inflammatoriske, allergiske og proliferative sykdommer. NO20051527L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40743802P 2002-08-29 2002-08-29
PCT/US2003/025062 WO2004019935A1 (en) 2002-08-29 2003-08-12 -3 (sulfonamidoethyl) -indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases

Publications (2)

Publication Number Publication Date
NO20051527D0 NO20051527D0 (no) 2005-03-22
NO20051527L true NO20051527L (no) 2005-03-22

Family

ID=31978485

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20051527A NO20051527L (no) 2002-08-29 2005-03-22 3-(sulfonamidoetyl) -indol-derivater for anvendelse som glukocorticoid-mimetica ved behandling av inflammatoriske, allergiske og proliferative sykdommer.

Country Status (23)

Country Link
US (1) US20040097574A1 (no)
EP (1) EP1539141B1 (no)
JP (1) JP4619786B2 (no)
KR (1) KR20050036982A (no)
CN (1) CN1678306A (no)
AT (1) ATE473740T1 (no)
AU (1) AU2003255259A1 (no)
BR (1) BR0313923A (no)
CA (1) CA2496580A1 (no)
CO (1) CO5550451A2 (no)
DE (1) DE60333371D1 (no)
EA (1) EA011095B1 (no)
EC (1) ECSP055611A (no)
ES (1) ES2349164T3 (no)
HR (1) HRP20050185A2 (no)
MX (1) MXPA05002297A (no)
NO (1) NO20051527L (no)
NZ (1) NZ538932A (no)
PL (1) PL375513A1 (no)
RS (1) RS20050174A (no)
UA (1) UA82675C2 (no)
WO (1) WO2004019935A1 (no)
ZA (1) ZA200500153B (no)

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EA011095B1 (ru) 2008-12-30
ATE473740T1 (de) 2010-07-15
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AU2003255259A1 (en) 2004-03-19
US20040097574A1 (en) 2004-05-20
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CN1678306A (zh) 2005-10-05
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