NO20065864L - Femleddete heterosykler anvendelige som serinproteaseinhibitorer - Google Patents
Femleddete heterosykler anvendelige som serinproteaseinhibitorerInfo
- Publication number
- NO20065864L NO20065864L NO20065864A NO20065864A NO20065864L NO 20065864 L NO20065864 L NO 20065864L NO 20065864 A NO20065864 A NO 20065864A NO 20065864 A NO20065864 A NO 20065864A NO 20065864 L NO20065864 L NO 20065864L
- Authority
- NO
- Norway
- Prior art keywords
- factor
- formula
- compounds
- serine protease
- protease inhibitors
- Prior art date
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- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A61P9/06—Antiarrhythmics
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
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PCT/US2005/021212 WO2005123050A2 (en) | 2004-06-15 | 2005-06-14 | Five-membered heterocycles useful as serine protease inhibitors |
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NO20065864A NO20065864L (no) | 2004-06-15 | 2006-12-15 | Femleddete heterosykler anvendelige som serinproteaseinhibitorer |
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EP (1) | EP1773786B1 (ru) |
JP (1) | JP4791460B2 (ru) |
KR (1) | KR20070024601A (ru) |
AU (1) | AU2005254102A1 (ru) |
BR (1) | BRPI0512084A (ru) |
CA (1) | CA2570472A1 (ru) |
ES (1) | ES2628279T3 (ru) |
IL (1) | IL179844A0 (ru) |
MX (1) | MXPA06014642A (ru) |
NO (1) | NO20065864L (ru) |
RU (1) | RU2007101073A (ru) |
WO (1) | WO2005123050A2 (ru) |
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- 2005-06-14 MX MXPA06014642A patent/MXPA06014642A/es active IP Right Grant
- 2005-06-14 KR KR1020067026365A patent/KR20070024601A/ko not_active Application Discontinuation
- 2005-06-14 WO PCT/US2005/021212 patent/WO2005123050A2/en active Application Filing
- 2005-06-14 ES ES05773261.2T patent/ES2628279T3/es active Active
- 2005-06-14 BR BRPI0512084-5A patent/BRPI0512084A/pt not_active IP Right Cessation
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2006
- 2006-12-05 IL IL179844A patent/IL179844A0/en unknown
- 2006-12-15 NO NO20065864A patent/NO20065864L/no not_active Application Discontinuation
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2008
- 2008-09-12 US US12/209,235 patent/US8101778B2/en active Active
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- 2011-12-15 US US13/326,809 patent/US8716492B2/en active Active
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Also Published As
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IL179844A0 (en) | 2007-07-04 |
RU2007101073A (ru) | 2008-07-20 |
US20120088758A1 (en) | 2012-04-12 |
JP2008502700A (ja) | 2008-01-31 |
KR20070024601A (ko) | 2007-03-02 |
EP1773786A2 (en) | 2007-04-18 |
US7453002B2 (en) | 2008-11-18 |
US8716492B2 (en) | 2014-05-06 |
CA2570472A1 (en) | 2005-12-29 |
BRPI0512084A (pt) | 2008-02-06 |
US9079860B2 (en) | 2015-07-14 |
US10112936B2 (en) | 2018-10-30 |
WO2005123050A3 (en) | 2007-01-04 |
MXPA06014642A (es) | 2007-02-12 |
US8101778B2 (en) | 2012-01-24 |
US20050282805A1 (en) | 2005-12-22 |
US20170166560A1 (en) | 2017-06-15 |
AU2005254102A1 (en) | 2005-12-29 |
US20090036438A1 (en) | 2009-02-05 |
JP4791460B2 (ja) | 2011-10-12 |
US20140206706A1 (en) | 2014-07-24 |
US20150259297A1 (en) | 2015-09-17 |
EP1773786B1 (en) | 2017-04-26 |
ES2628279T3 (es) | 2017-08-02 |
US9617224B2 (en) | 2017-04-11 |
WO2005123050A2 (en) | 2005-12-29 |
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