NO20023014D0 - Fremgangsmåte for fremstilling av 4-(heteroarylmetyl)-halogen- 1(2H)-ftalaziononer - Google Patents

Fremgangsmåte for fremstilling av 4-(heteroarylmetyl)-halogen- 1(2H)-ftalaziononer

Info

Publication number
NO20023014D0
NO20023014D0 NO20023014A NO20023014A NO20023014D0 NO 20023014 D0 NO20023014 D0 NO 20023014D0 NO 20023014 A NO20023014 A NO 20023014A NO 20023014 A NO20023014 A NO 20023014A NO 20023014 D0 NO20023014 D0 NO 20023014D0
Authority
NO
Norway
Prior art keywords
phthalazionones
heteroarylmethyl
halo
preparation
reaction
Prior art date
Application number
NO20023014A
Other languages
English (en)
Other versions
NO20023014L (no
NO321357B1 (no
Inventor
Orlin Petrov
Tamas Heiner
Harribert Neh
Martin Krueger
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO20023014D0 publication Critical patent/NO20023014D0/no
Publication of NO20023014L publication Critical patent/NO20023014L/no
Publication of NO321357B1 publication Critical patent/NO321357B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
NO20023014A 1999-12-23 2002-06-21 Fremgangsmate for fremstilling av 4-(heteroarylmetyl)-halogen-1(2H)-ftalazinoner NO321357B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19963607A DE19963607B4 (de) 1999-12-23 1999-12-23 Verfahren zur Herstellung von 4-(Heteroaryl-methyl) halogen-1(2H)-phthalazinonen
PCT/EP2000/013027 WO2001047912A1 (de) 1999-12-23 2000-12-20 Verfahren zur herstellung von 4-(heteroaryl-methyl)-halogen-1(2h)-phthalazinonen

Publications (3)

Publication Number Publication Date
NO20023014D0 true NO20023014D0 (no) 2002-06-21
NO20023014L NO20023014L (no) 2002-06-21
NO321357B1 NO321357B1 (no) 2006-05-02

Family

ID=7934888

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20023014A NO321357B1 (no) 1999-12-23 2002-06-21 Fremgangsmate for fremstilling av 4-(heteroarylmetyl)-halogen-1(2H)-ftalazinoner

Country Status (32)

Country Link
US (1) US6891041B2 (no)
EP (1) EP1242405B1 (no)
JP (1) JP2003529555A (no)
KR (1) KR100654265B1 (no)
CN (1) CN1221545C (no)
AT (1) ATE273972T1 (no)
AU (1) AU772981B2 (no)
BG (1) BG65387B1 (no)
BR (1) BR0016634A (no)
CA (1) CA2395407C (no)
CZ (1) CZ20022146A3 (no)
DE (2) DE19963607B4 (no)
DK (1) DK1242405T3 (no)
EE (1) EE04940B1 (no)
ES (1) ES2223626T3 (no)
HK (1) HK1055296A1 (no)
HR (1) HRP20020605B1 (no)
HU (1) HUP0300992A3 (no)
IL (2) IL150017A0 (no)
MX (1) MXPA02006224A (no)
NO (1) NO321357B1 (no)
NZ (1) NZ519285A (no)
PL (1) PL200714B1 (no)
PT (1) PT1242405E (no)
RO (1) RO121211B1 (no)
RS (1) RS50458B (no)
RU (1) RU2250900C2 (no)
SI (1) SI1242405T1 (no)
SK (1) SK285522B6 (no)
UA (1) UA72021C2 (no)
WO (1) WO2001047912A1 (no)
ZA (1) ZA200205853B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1296984B1 (it) * 1997-12-19 1999-08-03 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
US7151102B2 (en) * 2000-10-30 2006-12-19 Kudos Pharmaceuticals Limited Phthalazinone derivatives
GB0419072D0 (en) * 2004-08-26 2004-09-29 Kudos Pharm Ltd Phthalazinone derivatives
TWI404716B (zh) * 2006-10-17 2013-08-11 Kudos Pharm Ltd 酞嗪酮(phthalazinone)衍生物
MX2010004028A (es) * 2007-10-17 2010-04-30 Kudos Pharm Ltd 4-[3-(4-ciclopropancarbonil-piperacin-1-carbonil)-4-fluoro-bencil ]-2h-ftalacin-1-ona.
EP2346495B2 (en) 2008-10-07 2023-05-24 Kudos Pharmaceuticals Limited Pharmaceutical formulation 514
US8937178B2 (en) 2013-03-13 2015-01-20 Flatley Discovery Lab Phthalazinone compounds and methods for the treatment of cystic fibrosis
WO2016146303A1 (en) * 2015-03-19 2016-09-22 Clariant International Ltd Biodegradable sugar-amide-surfactants for enhanced oil recovery

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE567431A (no) * 1957-05-07
GB1293565A (en) * 1969-05-03 1972-10-18 Aspro Nicholas Ltd Aminophthalazines and pharmaceutical compositions thereof
IE47592B1 (en) * 1977-12-29 1984-05-02 Ici Ltd Enzyme inhibitory phthalazin-4-ylacetic acid derivatives, pharmaceutical compositions thereof,and process for their manufacture
EP0634404A1 (en) * 1993-07-13 1995-01-18 Rhone Poulenc Agriculture Ltd. Phtalazin derivatives and their use as pesticides
JP3919835B2 (ja) * 1994-08-09 2007-05-30 エーザイ・アール・アンド・ディー・マネジメント株式会社 縮合ピリダジン系化合物
DE69533057T2 (de) * 1994-08-09 2005-06-16 Eisai Co., Ltd. Kondensierte pyridazinverbindungen
ATE236134T1 (de) * 1996-12-18 2003-04-15 Neurogen Corp Isoquinolinamin und phtalazinamin derivate, die reagieren mit crf rezeptoren
CO4950519A1 (es) * 1997-02-13 2000-09-01 Novartis Ag Ftalazinas, preparaciones farmaceuticas que las comprenden y proceso para su preparacion
IT1296984B1 (it) * 1997-12-19 1999-08-03 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
ITMI981670A1 (it) * 1998-07-21 2000-01-21 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
ITMI981671A1 (it) * 1998-07-21 2000-01-21 Zambon Spa Derivati ftalazinici inibitori della fosfodisterasi 4
ITMI20000261A1 (it) * 2000-02-16 2001-08-16 Zambon Group Processo per la preparazione di piridiniliden-ftalidi

Also Published As

Publication number Publication date
BG106843A (en) 2003-02-28
DE19963607B4 (de) 2005-12-15
IL150017A0 (en) 2002-12-01
EP1242405B1 (de) 2004-08-18
CN1221545C (zh) 2005-10-05
PT1242405E (pt) 2004-11-30
SK285522B6 (sk) 2007-03-01
US20040192695A1 (en) 2004-09-30
NO20023014L (no) 2002-06-21
RU2250900C2 (ru) 2005-04-27
NO321357B1 (no) 2006-05-02
CN1413203A (zh) 2003-04-23
KR20020062363A (ko) 2002-07-25
NZ519285A (en) 2004-12-24
SK8922002A3 (en) 2002-11-06
PL200714B1 (pl) 2009-01-30
UA72021C2 (en) 2005-01-17
YU47302A (sh) 2005-06-10
SI1242405T1 (en) 2005-02-28
HRP20020605B1 (en) 2007-06-30
BR0016634A (pt) 2002-10-15
PL355525A1 (en) 2004-05-04
HUP0300992A2 (hu) 2003-08-28
CZ20022146A3 (cs) 2002-09-11
ATE273972T1 (de) 2004-09-15
US6891041B2 (en) 2005-05-10
RS50458B (sr) 2010-03-02
DK1242405T3 (da) 2004-11-01
HRP20020605A2 (en) 2004-12-31
RO121211B1 (ro) 2007-01-30
CA2395407C (en) 2009-04-28
MXPA02006224A (es) 2002-12-05
DE19963607A1 (de) 2001-07-12
BG65387B1 (bg) 2008-05-30
IL150017A (en) 2006-12-31
ES2223626T3 (es) 2005-03-01
AU772981B2 (en) 2004-05-13
EP1242405A1 (de) 2002-09-25
CA2395407A1 (en) 2001-07-05
DE50007520D1 (de) 2004-09-23
AU2012201A (en) 2001-07-09
HK1055296A1 (en) 2004-01-02
HUP0300992A3 (en) 2005-11-28
ZA200205853B (en) 2004-02-18
EE200200307A (et) 2003-06-16
JP2003529555A (ja) 2003-10-07
WO2001047912A1 (de) 2001-07-05
RU2002119559A (ru) 2004-01-10
KR100654265B1 (ko) 2006-12-07
EE04940B1 (et) 2007-12-17

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