MX377534B - Compuestos para usarse en el tratamiento de hiperinsulinemia. - Google Patents

Compuestos para usarse en el tratamiento de hiperinsulinemia.

Info

Publication number
MX377534B
MX377534B MX2016011160A MX2016011160A MX377534B MX 377534 B MX377534 B MX 377534B MX 2016011160 A MX2016011160 A MX 2016011160A MX 2016011160 A MX2016011160 A MX 2016011160A MX 377534 B MX377534 B MX 377534B
Authority
MX
Mexico
Prior art keywords
treatment
compounds
hyperinsulinemia
hyperinsulinaemia
relates
Prior art date
Application number
MX2016011160A
Other languages
English (en)
Spanish (es)
Other versions
MX2016011160A (es
Inventor
Michael Kagey
Steven B Landau
Original Assignee
Tensha Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tensha Therapeutics Inc filed Critical Tensha Therapeutics Inc
Publication of MX2016011160A publication Critical patent/MX2016011160A/es
Publication of MX377534B publication Critical patent/MX377534B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2016011160A 2014-02-28 2015-02-27 Compuestos para usarse en el tratamiento de hiperinsulinemia. MX377534B (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201461946682P 2014-02-28 2014-02-28
US201462019777P 2014-07-01 2014-07-01
US201462054620P 2014-09-24 2014-09-24
PCT/US2015/018118 WO2015131113A1 (en) 2014-02-28 2015-02-27 Treatment of conditions associated with hyperinsulinaemia

Publications (2)

Publication Number Publication Date
MX2016011160A MX2016011160A (es) 2017-04-27
MX377534B true MX377534B (es) 2025-03-10

Family

ID=52693055

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016011160A MX377534B (es) 2014-02-28 2015-02-27 Compuestos para usarse en el tratamiento de hiperinsulinemia.

Country Status (12)

Country Link
US (1) US10925881B2 (https=)
EP (1) EP3110424A1 (https=)
JP (2) JP2017506666A (https=)
KR (1) KR20160130778A (https=)
CN (1) CN106456653A (https=)
AU (1) AU2015222805B2 (https=)
CA (1) CA2940472A1 (https=)
IL (1) IL247354B (https=)
MX (1) MX377534B (https=)
RU (1) RU2722179C2 (https=)
SG (1) SG11201607108XA (https=)
WO (1) WO2015131113A1 (https=)

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CA2929652A1 (en) 2013-11-08 2015-05-14 Dana-Farber Cancer Institute, Inc. Combination therapy for cancer using bromodomain and extra-terminal (bet) protein inhibitors
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SG11201607108XA (en) 2014-02-28 2016-09-29 Tensha Therapeutics Inc Treatment of conditions associated with hyperinsulinaemia
BR112017008714A2 (pt) 2014-10-27 2017-12-19 Tensha Therapeutics Inc inibidores de bromodomínio
CA2989313A1 (en) 2015-06-26 2016-12-29 Tensha Therapeutics, Inc. Treatment of nut midline carcinoma
RU2018112953A (ru) * 2015-09-11 2019-10-14 Дана-Фарбер Кэнсер Инститьют, Инк. Ацетамидтиенотриазолодиазепины и пути их применения
HK1256417A1 (zh) 2015-09-11 2019-09-20 达纳-法伯癌症研究所股份有限公司 氰基噻吩并三唑并二氮杂环庚三烯及其用途
MX2018006499A (es) 2015-11-25 2018-08-01 Dana Farber Cancer Inst Inc Inhibidores de bromodominio bivalentes y usos de los mismos.
KR20190092429A (ko) * 2016-12-16 2019-08-07 에프. 호프만-라 로슈 아게 다이아제핀 유도체의 제조 방법
CN111094263A (zh) * 2017-09-14 2020-05-01 豪夫迈·罗氏有限公司 可用于制造药物的新化合物
MX2020013608A (es) 2018-06-13 2021-03-09 Worg Pharmaceuticals Hangzhou Co Ltd Preparacion de derivados de triazepina condensados y su uso como inhibidores de bet.
CN111253871A (zh) * 2020-03-13 2020-06-09 东莞市永益诚电子有限公司 一种钢化膜及其制备方法

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JP2017506666A (ja) 2017-03-09
KR20160130778A (ko) 2016-11-14
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RU2016138027A (ru) 2018-04-03
IL247354B (en) 2020-06-30
US10925881B2 (en) 2021-02-23
RU2722179C2 (ru) 2020-05-28
CA2940472A1 (en) 2015-09-03
WO2015131113A1 (en) 2015-09-03
CN106456653A (zh) 2017-02-22
MX2016011160A (es) 2017-04-27
AU2015222805A1 (en) 2016-09-15
AU2015222805B2 (en) 2020-05-21
SG11201607108XA (en) 2016-09-29
US20170209461A1 (en) 2017-07-27

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