KR850000969B1 - 안드로스탄 카보티오에이트의 제조방법 - Google Patents

안드로스탄 카보티오에이트의 제조방법 Download PDF

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Publication number
KR850000969B1
KR850000969B1 KR1019810000442A KR810000442A KR850000969B1 KR 850000969 B1 KR850000969 B1 KR 850000969B1 KR 1019810000442 A KR1019810000442 A KR 1019810000442A KR 810000442 A KR810000442 A KR 810000442A KR 850000969 B1 KR850000969 B1 KR 850000969B1
Authority
KR
South Korea
Prior art keywords
hydroxy
diene
methyl
solution
ethyl acetate
Prior art date
Application number
KR1019810000442A
Other languages
English (en)
Korean (ko)
Other versions
KR830005262A (ko
Inventor
헨리 필립스 고든
맥도날드 베인 브리안
윌리암슨 크리스토퍼
필립 스티플스 이안
브루스 레잉 스투워트
Original Assignee
글락소 그룹 리미티드
배리 안소니뉴샘
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 글락소 그룹 리미티드, 배리 안소니뉴샘 filed Critical 글락소 그룹 리미티드
Publication of KR830005262A publication Critical patent/KR830005262A/ko
Application granted granted Critical
Publication of KR850000969B1 publication Critical patent/KR850000969B1/ko

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/0026—Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • C07J71/0015—Oxiranes at position 9(11)
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1019810000442A 1980-02-15 1981-02-13 안드로스탄 카보티오에이트의 제조방법 KR850000969B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8005174 1980-02-15
GB8005174 1980-02-15
GB8013339 1980-04-23
GB8013339 1980-04-23

Publications (2)

Publication Number Publication Date
KR830005262A KR830005262A (ko) 1983-08-03
KR850000969B1 true KR850000969B1 (ko) 1985-07-02

Family

ID=26274505

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019810000442A KR850000969B1 (ko) 1980-02-15 1981-02-13 안드로스탄 카보티오에이트의 제조방법

Country Status (23)

Country Link
KR (1) KR850000969B1 (es)
AT (1) AT395427B (es)
AU (1) AU544517B2 (es)
BG (1) BG60700B2 (es)
CH (2) CH651307A5 (es)
CZ (1) CZ281275B6 (es)
DE (2) DE3153379C2 (es)
DK (1) DK147022C (es)
ES (5) ES8207194A1 (es)
FI (1) FI70904C (es)
FR (2) FR2477156A1 (es)
HK (1) HK58385A (es)
IE (1) IE51394B1 (es)
IT (1) IT1170717B (es)
KE (1) KE3526A (es)
MX (1) MX9202717A (es)
MY (1) MY8500757A (es)
NL (2) NL191792C (es)
NZ (1) NZ196260A (es)
PT (1) PT72502B (es)
SE (1) SE452468B (es)
SG (1) SG36885G (es)
SK (1) SK403491A3 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA817929B (en) * 1980-12-22 1982-10-27 Upjohn Co 5alpha-and 5beta-androstane-17beta-carboxylates

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1436549A (en) * 1972-06-15 1976-05-19 Glaxo Lab Ltd 17beta-mercaptocarbonyl-3alpha-hydroxy-steroids and their esters
GB1438940A (en) * 1972-07-19 1976-06-09 Glaxo Lab Ltd 17beta-haloalkoxycarbonyl-17alpha-oxysteroids
GB1514476A (en) * 1974-08-30 1978-06-14 Glaxo Lab Ltd Alkyl and haloalkyl androst-4-ene and androsta-1,4-diene-17beta-carboxylates
US4188385A (en) * 1978-04-05 1980-02-12 Syntex (U.S.A.) Inc. Thioetianic acid derivatives
GB1580517A (en) * 1978-04-06 1980-12-03 Fowler I Crutches

Also Published As

Publication number Publication date
CZ403491A3 (en) 1994-03-16
ES524985A0 (es) 1985-01-01
SK278140B6 (en) 1996-02-07
FR2485542A1 (fr) 1981-12-31
KE3526A (en) 1985-06-07
NL8100707A (nl) 1981-09-16
ES8502447A1 (es) 1985-01-01
ES532055A0 (es) 1985-10-16
SE8101010L (sv) 1981-08-16
ES8600936A1 (es) 1985-10-16
FI810444L (fi) 1981-08-16
NL191792B (nl) 1996-04-01
NL960029I1 (nl) 1997-02-03
MX9202717A (es) 1992-06-30
ES518161A0 (es) 1984-01-16
FR2477156A1 (fr) 1981-09-04
DE3105307A1 (de) 1981-12-10
ATA67481A (de) 1992-05-15
DK147022C (da) 1984-08-27
PT72502A (en) 1981-03-01
NL960029I2 (nl) 1997-04-01
IT1170717B (it) 1987-06-03
AU6729881A (en) 1981-08-20
NZ196260A (en) 1983-11-30
PT72502B (en) 1982-02-05
KR830005262A (ko) 1983-08-03
FI70904C (fi) 1986-10-27
BG60700B2 (bg) 1995-12-29
CH644615A5 (de) 1984-08-15
IE810282L (en) 1981-08-15
FI70904B (fi) 1986-07-18
ES499394A0 (es) 1982-09-01
ES8305379A1 (es) 1983-04-01
ES8402317A1 (es) 1984-01-16
IT8147792A0 (it) 1981-02-13
FR2485542B1 (es) 1983-06-10
MY8500757A (en) 1985-12-31
SE452468B (sv) 1987-11-30
DE3153379C2 (es) 1992-11-19
AU544517B2 (en) 1985-06-06
CZ281275B6 (cs) 1996-08-14
NL191792C (nl) 1996-08-02
SG36885G (en) 1985-11-15
DK62381A (da) 1981-08-16
SK403491A3 (en) 1996-02-07
FR2477156B1 (es) 1984-11-16
AT395427B (de) 1992-12-28
ES8207194A1 (es) 1982-09-01
CH651307A5 (de) 1985-09-13
ES509539A0 (es) 1983-04-01
HK58385A (en) 1985-08-16
DE3105307C2 (es) 1988-09-29
DK147022B (da) 1984-03-19
IE51394B1 (en) 1986-12-24

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