KR101063585B1 - 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체 - Google Patents

피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체 Download PDF

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KR101063585B1
KR101063585B1 KR1020097011570A KR20097011570A KR101063585B1 KR 101063585 B1 KR101063585 B1 KR 101063585B1 KR 1020097011570 A KR1020097011570 A KR 1020097011570A KR 20097011570 A KR20097011570 A KR 20097011570A KR 101063585 B1 KR101063585 B1 KR 101063585B1
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leu
gly
ser
ala
val
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KR20090078841A (ko
Inventor
다까히로 이시이
다까시 수가네
준 마에다
후미에 나라자끼
아끼오 가께후다
겐따로 사또
다쯔히사 다까하시
다까또시 가나야마
치까시 사이또
조따로 스즈끼
치사또 가나이
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아스텔라스세이야쿠 가부시키가이샤
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Publication of KR20090078841A publication Critical patent/KR20090078841A/ko
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Assigned to 아우토반 쎄라퓨틱스, 인크. reassignment 아우토반 쎄라퓨틱스, 인크. 권리의 전부이전등록 Assignors: 아스텔라스세이야쿠 가부시키가이샤
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    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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  • Otolaryngology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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KR1020097011570A 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체 Expired - Fee Related KR101063585B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2005040197 2005-02-17
JPJP-P-2005-040197 2005-02-17
JPJP-P-2005-303065 2005-10-18
JP2005303065 2005-10-18
PCT/JP2006/302698 WO2006088075A1 (ja) 2005-02-17 2006-02-16 ピリジル 非芳香族含窒素ヘテロ環－１－カルボン酸エステル誘導体

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KR1020077020924A Division KR101063663B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르유도체

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KR20090078841A KR20090078841A (ko) 2009-07-20
KR101063585B1 true KR101063585B1 (ko) 2011-09-07

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KR1020097011570A Expired - Fee Related KR101063585B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체
KR1020097011569A Expired - Fee Related KR101065979B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르 유도체
KR1020077020924A Expired - Fee Related KR101063663B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르유도체

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KR1020077020924A Expired - Fee Related KR101063663B1 (ko) 2005-02-17 2006-02-16 피리딜 비방향족 질소 함유 헤테로환-1-카르복실산에스테르유도체

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US (3) US7919495B2 (enExample)
EP (2) EP1849773B1 (enExample)
JP (1) JP4702361B2 (enExample)
KR (3) KR101063585B1 (enExample)
CN (1) CN101160287B (enExample)
AU (3) AU2006215080B2 (enExample)
BR (1) BRPI0608205B8 (enExample)
CA (1) CA2598294C (enExample)
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DK (2) DK2607362T3 (enExample)
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PT (2) PT1849773E (enExample)
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SI (2) SI1849773T1 (enExample)
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JPWO2008023720A1 (ja) * 2006-08-23 2010-01-14 アステラス製薬株式会社 ウレア化合物又はその塩
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