KR100908166B1 - 5ｈｔ2ｃ 수용체 조절제 - Google Patents

5ｈｔ2ｃ 수용체 조절제 Download PDF

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Publication number
KR100908166B1
KR100908166B1 KR1020087000551A KR20087000551A KR100908166B1 KR 100908166 B1 KR100908166 B1 KR 100908166B1 KR 1020087000551 A KR1020087000551 A KR 1020087000551A KR 20087000551 A KR20087000551 A KR 20087000551A KR 100908166 B1 KR100908166 B1 KR 100908166B1
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Prior art keywords
tetrahydro
benzazine
methyl
delete delete
methoxy
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Expired - Lifetime
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Korean (ko)
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KR20080009340A (ko
Inventor
브라이언 스미스
제프리 스미스
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아레나 파마슈티칼스, 인크.
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29255581&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR100908166(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 아레나 파마슈티칼스, 인크. filed Critical 아레나 파마슈티칼스, 인크.
Publication of KR20080009340A publication Critical patent/KR20080009340A/ko
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Publication of KR100908166B1 publication Critical patent/KR100908166B1/ko
Assigned to 에-자이가부시기가이샤 reassignment 에-자이가부시기가이샤 권리의 전부이전등록 Assignors: 아레나 파마슈티칼스, 인크.
Assigned to 에자이 알앤드디 매니지먼트 가부시키가이샤 reassignment 에자이 알앤드디 매니지먼트 가부시키가이샤 권리의 전부이전등록 Assignors: 에-자이가부시기가이샤
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    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Addiction (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
KR1020087000551A 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제 Expired - Lifetime KR100908166B1 (ko)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US37205802P 2002-04-12 2002-04-12
US60/372,058 2002-04-12
US40549502P 2002-08-23 2002-08-23
US60/405,495 2002-08-23
US43460702P 2002-12-18 2002-12-18
US60/434,607 2002-12-18
US10/410,991 US6953787B2 (en) 2002-04-12 2003-04-10 5HT2C receptor modulators
US10/410,991 2003-04-10
PCT/US2003/011076 WO2003086306A2 (en) 2002-04-12 2003-04-11 5ht2c receptor modulators

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020047016198A Division KR100812925B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020097000060A Division KR100908167B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제

Publications (2)

Publication Number Publication Date
KR20080009340A KR20080009340A (ko) 2008-01-28
KR100908166B1 true KR100908166B1 (ko) 2009-07-16

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ID=29255581

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Application Number Title Priority Date Filing Date
KR1020087000551A Expired - Lifetime KR100908166B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제
KR1020097000060A Expired - Lifetime KR100908167B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제
KR1020047016198A Expired - Lifetime KR100812925B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제

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KR1020097000060A Expired - Lifetime KR100908167B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제
KR1020047016198A Expired - Lifetime KR100812925B1 (ko) 2002-04-12 2003-04-11 5ｈｔ2ｃ 수용체 조절제

Country Status (28)

Country Link
US (11) US6953787B2 (https=)
EP (4) EP2363394A1 (https=)
JP (5) JP4155926B2 (https=)
KR (3) KR100908166B1 (https=)
CN (5) CN100486967C (https=)
AT (1) ATE294781T1 (https=)
AU (1) AU2003221866B2 (https=)
BR (2) BRPI0309303B8 (https=)
CA (1) CA2481723C (https=)
CR (2) CR7503A (https=)
DE (1) DE60300610T2 (https=)
DK (1) DK1411881T3 (https=)
ES (2) ES2670568T3 (https=)
GE (1) GEP20074197B (https=)
IL (1) IL164162A0 (https=)
IS (1) IS2134B (https=)
MX (1) MXPA04009965A (https=)
MY (1) MY141476A (https=)
NO (1) NO323528B1 (https=)
NZ (1) NZ535381A (https=)
PL (4) PL231405B1 (https=)
PT (1) PT1411881E (https=)
RU (1) RU2317982C2 (https=)
SI (1) SI1411881T1 (https=)
TW (1) TWI252105B (https=)
UA (1) UA77788C2 (https=)
WO (1) WO2003086306A2 (https=)
ZA (1) ZA200408506B (https=)

Families Citing this family (85)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8478824B2 (en) * 2002-02-05 2013-07-02 Portauthority Technologies Inc. Apparatus and method for controlling unauthorized dissemination of electronic mail
SE0200968D0 (sv) * 2002-03-26 2002-03-26 Lars Baltzer Novel polypeptide scaffolds and use thereof
US6953787B2 (en) * 2002-04-12 2005-10-11 Arena Pharmaceuticals, Inc. 5HT2C receptor modulators
US7595311B2 (en) 2002-05-24 2009-09-29 Exelixis, Inc. Azepinoindole derivatives as pharmaceutical agents
TWI329111B (en) 2002-05-24 2010-08-21 X Ceptor Therapeutics Inc Azepinoindole and pyridoindole derivatives as pharmaceutical agents
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