KR100748386B1 - 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체 - Google Patents

단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체 Download PDF

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KR100748386B1
KR100748386B1 KR1020037005805A KR20037005805A KR100748386B1 KR 100748386 B1 KR100748386 B1 KR 100748386B1 KR 1020037005805 A KR1020037005805 A KR 1020037005805A KR 20037005805 A KR20037005805 A KR 20037005805A KR 100748386 B1 KR100748386 B1 KR 100748386B1
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formula
compound
alkyl
solution
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KR20030042036A (ko
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라이너 알베르트
니겔 그라함 쿠크
실바인 코텐스
클라우스 에르하르트
장-삐에르 에베노우
리차드 세드라니
마트 페터 본
유르겐 바그너
게르하르트 젠크
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노파르티스 아게
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  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
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  • Communicable Diseases (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
KR1020037005805A 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체 Expired - Fee Related KR100748386B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US24640000P 2000-11-07 2000-11-07
US60/246,400 2000-11-07
US28370501P 2001-04-13 2001-04-13
US60/283,705 2001-04-13
PCT/EP2001/012785 WO2002038561A1 (en) 2000-11-07 2001-11-05 Indolylmaleimide derivatives as protein kinase c inhibitors

Related Child Applications (1)

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KR1020067017472A Division KR100916613B1 (ko) 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체

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Publication Number Publication Date
KR20030042036A KR20030042036A (ko) 2003-05-27
KR100748386B1 true KR100748386B1 (ko) 2007-08-10

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KR1020037005805A Expired - Fee Related KR100748386B1 (ko) 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체
KR1020067017472A Expired - Fee Related KR100916613B1 (ko) 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체
KR1020087002849A Ceased KR20080014934A (ko) 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체

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KR1020067017472A Expired - Fee Related KR100916613B1 (ko) 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체
KR1020087002849A Ceased KR20080014934A (ko) 2000-11-07 2001-11-05 단백질 키나제 ｃ 억제제로서의 인돌릴말레이미드 유도체

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EP (2) EP1337527B1 (enExample)
JP (1) JP4234426B2 (enExample)
KR (3) KR100748386B1 (enExample)
CN (1) CN1253449C (enExample)
AR (1) AR035211A1 (enExample)
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PE20040079A1 (es) 2002-04-03 2004-04-19 Novartis Ag Derivados de indolilmaleimida
JP2005531607A (ja) * 2002-06-05 2005-10-20 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ キナーゼ阻害剤として置換ピロリン
EP1513830A1 (en) 2002-06-05 2005-03-16 Janssen Pharmaceutica N.V. Bisindolyl-maleimid derivatives as kinase inhibitors
GB0303319D0 (en) * 2003-02-13 2003-03-19 Novartis Ag Organic compounds
US8598146B2 (en) 2003-09-16 2013-12-03 Garvan Institute Of Medical Research Methods for identifying modulators of protein kinase C-epsilon (PKCε) and method of treatment of aberrant glucose metabolism associated therewith
WO2005039549A1 (en) * 2003-10-27 2005-05-06 Novartis Ag Indolyl-pyrroledione derivatives for the treatment of neurological and vascular disorders related to beta-amyloid generation and/or aggregation
CA2545340A1 (en) * 2003-11-10 2005-05-26 Synta Pharmaceuticals, Corp. Fused heterocyclic compounds
GB0401089D0 (en) * 2004-01-19 2004-02-18 Novartis Ag Organic compounds
ATE391127T1 (de) 2004-01-19 2008-04-15 Novartis Pharma Gmbh Indolylmaleimidderivate
BRPI0509754A (pt) * 2004-04-08 2007-10-16 Novartis Ag inibidores de proteìna quinase c para o tratamento de doenças auto-imunes e de rejeição a transplante
GB0410713D0 (en) * 2004-05-13 2004-06-16 Novartis Ag Organic compounds
WO2006061212A1 (en) 2004-12-08 2006-06-15 Johannes Gutenberg-Universität Mainz 3-(indolyl)-4-arylmaleimide derivatives and their use as angiogenesis inhibitors
GB0504203D0 (en) * 2005-03-01 2005-04-06 Novartis Ag Organic compounds
GB0507918D0 (en) 2005-04-19 2005-05-25 Novartis Ag Organic compounds
WO2006117212A2 (en) 2005-05-04 2006-11-09 Develogen Aktiengesellschaft Use of gsk-3 inhibitors for preventing and treating pancreatic autoimmune disorders
GB0511060D0 (en) 2005-05-31 2005-07-06 Novartis Ag Organic compounds
DE602006019732D1 (de) 2005-07-11 2011-03-03 Novartis Ag Indolylmaleimidderivate
BRPI0617830B8 (pt) 2005-10-26 2021-05-25 Novartis Ag uso de um anticorpo de ligação il-1beta e composições farmacêuticas compreendendo o mesmo
NZ568182A (en) 2005-11-21 2010-08-27 Novartis Ag Neuroendocrine tumor treatment using MTOR inhibitors
GB0601744D0 (en) 2006-01-27 2006-03-08 Novartis Ag Organic compounds
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