JPS5892610A - 経口用放出調整複合単位製剤 - Google Patents
経口用放出調整複合単位製剤Info
- Publication number
- JPS5892610A JPS5892610A JP56194342A JP19434281A JPS5892610A JP S5892610 A JPS5892610 A JP S5892610A JP 56194342 A JP56194342 A JP 56194342A JP 19434281 A JP19434281 A JP 19434281A JP S5892610 A JPS5892610 A JP S5892610A
- Authority
- JP
- Japan
- Prior art keywords
- active substance
- core
- coating
- formulation according
- formulation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK5164/81 | 1981-11-20 | ||
| DK516481A DK150008C (da) | 1981-11-20 | 1981-11-20 | Fremgangsmaade til fremstilling af et farmaceutisk oralt polydepotpraeparat |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5892610A true JPS5892610A (ja) | 1983-06-02 |
| JPH0478611B2 JPH0478611B2 (cg-RX-API-DMAC7.html) | 1992-12-11 |
Family
ID=8140030
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP56194342A Granted JPS5892610A (ja) | 1981-11-20 | 1981-12-01 | 経口用放出調整複合単位製剤 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4606909A (cg-RX-API-DMAC7.html) |
| EP (1) | EP0080341B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JPS5892610A (cg-RX-API-DMAC7.html) |
| AT (1) | ATE30380T1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU563725B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA1198370A (cg-RX-API-DMAC7.html) |
| DE (2) | DE3277520D1 (cg-RX-API-DMAC7.html) |
| DK (1) | DK150008C (cg-RX-API-DMAC7.html) |
| FI (1) | FI79943C (cg-RX-API-DMAC7.html) |
| NO (1) | NO823891L (cg-RX-API-DMAC7.html) |
| NZ (1) | NZ202565A (cg-RX-API-DMAC7.html) |
| ZA (1) | ZA828433B (cg-RX-API-DMAC7.html) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61143316A (ja) * | 1984-12-17 | 1986-07-01 | Chugai Pharmaceut Co Ltd | 安定な錠剤の製造法 |
| JPS6248618A (ja) * | 1985-08-27 | 1987-03-03 | Zeria Shinyaku Kogyo Kk | 徐放性製剤およびその製造法 |
| JP2010270128A (ja) * | 1998-11-02 | 2010-12-02 | Elan Pharma Internatl Ltd | 多粒子改質放出組成物 |
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| JPS4962618A (cg-RX-API-DMAC7.html) * | 1972-08-30 | 1974-06-18 | ||
| US4173626A (en) * | 1978-12-11 | 1979-11-06 | Merck & Co., Inc. | Sustained release indomethacin |
| JPS5587717A (en) * | 1978-12-05 | 1980-07-02 | Haessle Ab | Cardiotonic glycoside containing medicine |
| JPS55100314A (en) * | 1979-01-25 | 1980-07-31 | Adria Lab Inc | Continuously releasing drug composition |
| US4291016A (en) * | 1976-07-27 | 1981-09-22 | Sandoz Ltd. | Enteric coated mixture of 4-(2-hydroxy-3-isopropylamino-propoxy) indole and sodium lauryl sulphate |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3081233A (en) * | 1960-08-08 | 1963-03-12 | Upjohn Co | Enteric-coated pilules |
| FR1503582A (fr) * | 1966-07-18 | 1967-12-01 | Sedaph Soc D Applic Pharma Sa | Procédé de préparation d'une nouvelle forme solide de médicament |
| FR2059978A1 (en) * | 1969-08-20 | 1971-06-11 | Sogeras | Enteric coating of sensitive medicaments inp |
| DE2031871C3 (de) * | 1970-06-27 | 1974-06-27 | Roehm Gmbh, 6100 Darmstadt | Überzugsmasse für Arzneiformen |
| FR2116256A1 (en) * | 1970-12-02 | 1972-07-13 | Sobio Lab | Enteric - coated l-dopa - for treatment of parkinsonism with reduced gastrointestinal side-effects |
| GB1468172A (en) * | 1973-03-28 | 1977-03-23 | Benzon As Alfred | Oral drug preparations |
| DE2336218C3 (de) * | 1973-07-17 | 1985-11-14 | Byk Gulden Lomberg Chemische Fabrik Gmbh, 7750 Konstanz | Orale Arzneiform |
| GB1576376A (en) * | 1977-03-30 | 1980-10-08 | Benzon As Alfred | Multiple-unit drug dose |
| IT1115596B (it) * | 1978-03-13 | 1986-02-03 | Bayer Italia Spa | Metodo per la preparazione di microgranuli gastoresistenti ed enterosolubili di sostanze farmaceutiche,in particolare di sostanze proteiche e microgranuli preparati con detto metodo |
| SE7813246L (sv) * | 1978-12-22 | 1980-06-23 | Haessle Ab | Fast farmaceutisk beredning innehallande kroppar med flera ytskikt |
| SE8003805L (sv) * | 1980-05-21 | 1981-11-22 | Haessle Ab | En farmaceutisk beredning med forbettrade utlosningsegenskap |
-
1981
- 1981-11-20 DK DK516481A patent/DK150008C/da not_active IP Right Cessation
- 1981-12-01 JP JP56194342A patent/JPS5892610A/ja active Granted
-
1982
- 1982-11-16 ZA ZA828433A patent/ZA828433B/xx unknown
- 1982-11-19 NZ NZ202565A patent/NZ202565A/en unknown
- 1982-11-19 AT AT82306170T patent/ATE30380T1/de active
- 1982-11-19 DE DE8282306170T patent/DE3277520D1/de not_active Expired
- 1982-11-19 DE DE198282306170T patent/DE80341T1/de active Pending
- 1982-11-19 NO NO823891A patent/NO823891L/no unknown
- 1982-11-19 AU AU90722/82A patent/AU563725B2/en not_active Ceased
- 1982-11-19 EP EP82306170A patent/EP0080341B1/en not_active Expired
- 1982-11-19 FI FI823975A patent/FI79943C/fi not_active IP Right Cessation
- 1982-11-22 CA CA000416035A patent/CA1198370A/en not_active Expired
-
1984
- 1984-06-20 US US06/622,393 patent/US4606909A/en not_active Expired - Fee Related
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4962618A (cg-RX-API-DMAC7.html) * | 1972-08-30 | 1974-06-18 | ||
| US4291016A (en) * | 1976-07-27 | 1981-09-22 | Sandoz Ltd. | Enteric coated mixture of 4-(2-hydroxy-3-isopropylamino-propoxy) indole and sodium lauryl sulphate |
| JPS5587717A (en) * | 1978-12-05 | 1980-07-02 | Haessle Ab | Cardiotonic glycoside containing medicine |
| US4173626A (en) * | 1978-12-11 | 1979-11-06 | Merck & Co., Inc. | Sustained release indomethacin |
| JPS55100314A (en) * | 1979-01-25 | 1980-07-31 | Adria Lab Inc | Continuously releasing drug composition |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61143316A (ja) * | 1984-12-17 | 1986-07-01 | Chugai Pharmaceut Co Ltd | 安定な錠剤の製造法 |
| JPS6248618A (ja) * | 1985-08-27 | 1987-03-03 | Zeria Shinyaku Kogyo Kk | 徐放性製剤およびその製造法 |
| JP2010270128A (ja) * | 1998-11-02 | 2010-12-02 | Elan Pharma Internatl Ltd | 多粒子改質放出組成物 |
| JP4827915B2 (ja) * | 2005-03-07 | 2011-11-30 | アルファ ワッセルマン ソシエタ ペル アチオニ | リファキシミンを含む胃抵抗性薬剤組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| FI823975A0 (fi) | 1982-11-19 |
| DK150008B (da) | 1986-11-17 |
| DK516481A (da) | 1983-05-21 |
| EP0080341A3 (en) | 1983-09-14 |
| ATE30380T1 (de) | 1987-11-15 |
| DE3277520D1 (en) | 1987-12-03 |
| DE80341T1 (de) | 1983-10-27 |
| FI79943C (fi) | 1990-04-10 |
| CA1198370A (en) | 1985-12-24 |
| JPH0478611B2 (cg-RX-API-DMAC7.html) | 1992-12-11 |
| ZA828433B (en) | 1983-08-31 |
| FI823975L (fi) | 1983-05-21 |
| AU9072282A (en) | 1983-05-26 |
| NO823891L (no) | 1983-05-24 |
| US4606909A (en) | 1986-08-19 |
| EP0080341B1 (en) | 1987-10-28 |
| DK150008C (da) | 1987-05-25 |
| EP0080341A2 (en) | 1983-06-01 |
| NZ202565A (en) | 1987-03-06 |
| AU563725B2 (en) | 1987-07-23 |
| FI79943B (fi) | 1989-12-29 |
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