JP6437452B2 - Ｐｉｍキナーゼ阻害剤として有用な二環式芳香族カルボキサミド化合物 - Google Patents

Ｐｉｍキナーゼ阻害剤として有用な二環式芳香族カルボキサミド化合物 Download PDF

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JP6437452B2
JP6437452B2 JP2015552897A JP2015552897A JP6437452B2 JP 6437452 B2 JP6437452 B2 JP 6437452B2 JP 2015552897 A JP2015552897 A JP 2015552897A JP 2015552897 A JP2015552897 A JP 2015552897A JP 6437452 B2 JP6437452 B2 JP 6437452B2
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amino
alkyl
carboxamide
pharmaceutically acceptable
pyridin
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JP2016505021A (ja
JP2016505021A5 (OSRAM
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ユン−ロン・リ
デイビッド・エム・バーンズ
フォン・ハオ
チュ−ビアオ・シュエ
ワン・アンライ
ジュン・パン
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Incyte Holdings Corp
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Organic Chemistry (AREA)
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
  • Pulmonology (AREA)
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  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Transplantation (AREA)
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  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2015552897A 2013-01-14 2014-01-14 Ｐｉｍキナーゼ阻害剤として有用な二環式芳香族カルボキサミド化合物 Active JP6437452B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361752249P 2013-01-14 2013-01-14
US61/752,249 2013-01-14
US201361791275P 2013-03-15 2013-03-15
US61/791,275 2013-03-15
PCT/US2014/011487 WO2014110574A1 (en) 2013-01-14 2014-01-14 Bicyclic aromatic carboxamide compounds useful as pim kinase inhibitors

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JP2016505021A JP2016505021A (ja) 2016-02-18
JP2016505021A5 JP2016505021A5 (OSRAM) 2017-02-02
JP6437452B2 true JP6437452B2 (ja) 2018-12-12

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US (2) US9278950B2 (OSRAM)
EP (1) EP2943485B1 (OSRAM)
JP (1) JP6437452B2 (OSRAM)
CA (1) CA2897200C (OSRAM)
ES (1) ES2649156T3 (OSRAM)
WO (1) WO2014110574A1 (OSRAM)

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CA2897200A1 (en) 2014-07-17
US20140200216A1 (en) 2014-07-17
HK1216316A1 (en) 2016-11-11
JP2016505021A (ja) 2016-02-18
US20160137626A1 (en) 2016-05-19
US9676750B2 (en) 2017-06-13
EP2943485B1 (en) 2017-09-20
ES2649156T3 (es) 2018-01-10
EP2943485A1 (en) 2015-11-18

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