JP4901727B2 - コートされた錠剤処方および方法 - Google Patents

コートされた錠剤処方および方法 Download PDF

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Publication number
JP4901727B2
JP4901727B2 JP2007515382A JP2007515382A JP4901727B2 JP 4901727 B2 JP4901727 B2 JP 4901727B2 JP 2007515382 A JP2007515382 A JP 2007515382A JP 2007515382 A JP2007515382 A JP 2007515382A JP 4901727 B2 JP4901727 B2 JP 4901727B2
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JP
Japan
Prior art keywords
coating layer
coating
tablet
coated
polymer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
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JP2007515382A
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English (en)
Japanese (ja)
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JP2008501025A (ja
JP2008501025A5 (OSRAM
Inventor
ディブヤカント・デサイ
ビン・ブイ・リ
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of JP2008501025A publication Critical patent/JP2008501025A/ja
Publication of JP2008501025A5 publication Critical patent/JP2008501025A5/ja
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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2007515382A 2004-05-28 2005-05-26 コートされた錠剤処方および方法 Expired - Lifetime JP4901727B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US57531904P 2004-05-28 2004-05-28
US60/575,319 2004-05-28
PCT/US2005/018692 WO2005117841A1 (en) 2004-05-28 2005-05-26 Coated tablet formulation and method

Publications (3)

Publication Number Publication Date
JP2008501025A JP2008501025A (ja) 2008-01-17
JP2008501025A5 JP2008501025A5 (OSRAM) 2008-07-03
JP4901727B2 true JP4901727B2 (ja) 2012-03-21

Family

ID=34971747

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007515382A Expired - Lifetime JP4901727B2 (ja) 2004-05-28 2005-05-26 コートされた錠剤処方および方法

Country Status (33)

Country Link
US (4) US7951400B2 (OSRAM)
EP (3) EP2298288B2 (OSRAM)
JP (1) JP4901727B2 (OSRAM)
KR (2) KR20120064141A (OSRAM)
CN (2) CN1988891B (OSRAM)
AR (2) AR049062A1 (OSRAM)
AU (1) AU2005249467B2 (OSRAM)
BR (1) BRPI0510419B8 (OSRAM)
CA (1) CA2568391C (OSRAM)
CY (2) CY1117813T1 (OSRAM)
DK (2) DK1753406T4 (OSRAM)
ES (3) ES2754573T3 (OSRAM)
GE (1) GEP20094639B (OSRAM)
HR (2) HRP20160880T4 (OSRAM)
HU (2) HUE029039T2 (OSRAM)
IL (2) IL179454A (OSRAM)
LT (1) LT2298288T (OSRAM)
ME (2) ME02643B (OSRAM)
MX (1) MXPA06013711A (OSRAM)
MY (1) MY147639A (OSRAM)
NO (1) NO343907B1 (OSRAM)
NZ (1) NZ551591A (OSRAM)
PE (1) PE20060425A1 (OSRAM)
PH (1) PH12013500450A1 (OSRAM)
PL (2) PL2298288T5 (OSRAM)
PT (2) PT2298288T (OSRAM)
RS (2) RS54929B2 (OSRAM)
RU (1) RU2372894C2 (OSRAM)
SI (3) SI1753406T1 (OSRAM)
TW (2) TWI354569B (OSRAM)
UA (1) UA88168C2 (OSRAM)
WO (1) WO2005117841A1 (OSRAM)
ZA (1) ZA200609541B (OSRAM)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2022135147A (ja) * 2021-03-04 2022-09-15 日医工株式会社 サキサグリプチン含有錠剤
US11786472B2 (en) 2020-06-23 2023-10-17 Sawai Pharmaceutical Co., Ltd. Preparation containing saxagliptin and method for producing the same

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