JP4828407B2 - 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法 - Google Patents

3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法 Download PDF

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JP4828407B2
JP4828407B2 JP2006503737A JP2006503737A JP4828407B2 JP 4828407 B2 JP4828407 B2 JP 4828407B2 JP 2006503737 A JP2006503737 A JP 2006503737A JP 2006503737 A JP2006503737 A JP 2006503737A JP 4828407 B2 JP4828407 B2 JP 4828407B2
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pyridinyl
azabicyclo
methyl
oct
compounds
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JP2006518746A (ja
JP2006518746A5 (enExample
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マズロブ,アナトリー・エイ
クルチツク,ヨーゼフ
マイオ,ラン
シーマンズ,アンジエラ・エス
フイリツプス,テレサ・ヤングピーター
シユミツト,ジエフリー・ダニエル
ミラー,クレイグ・ハリスン
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ターガセプト,インコーポレイテッド
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0455Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems

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JP2006503737A 2003-02-21 2004-02-20 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法 Expired - Fee Related JP4828407B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/372,642 US6953855B2 (en) 1998-12-11 2003-02-21 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof
US10/372,642 2003-02-21
PCT/US2004/005044 WO2004076449A2 (en) 2003-02-21 2004-02-20 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2011021779A Division JP5211183B2 (ja) 2003-02-21 2011-02-03 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法
JP2011021778A Division JP5291728B2 (ja) 2003-02-21 2011-02-03 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法

Publications (3)

Publication Number Publication Date
JP2006518746A JP2006518746A (ja) 2006-08-17
JP2006518746A5 JP2006518746A5 (enExample) 2007-04-12
JP4828407B2 true JP4828407B2 (ja) 2011-11-30

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JP2006503737A Expired - Fee Related JP4828407B2 (ja) 2003-02-21 2004-02-20 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法
JP2011021778A Expired - Fee Related JP5291728B2 (ja) 2003-02-21 2011-02-03 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法
JP2011021779A Expired - Fee Related JP5211183B2 (ja) 2003-02-21 2011-02-03 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法

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Application Number Title Priority Date Filing Date
JP2011021778A Expired - Fee Related JP5291728B2 (ja) 2003-02-21 2011-02-03 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法
JP2011021779A Expired - Fee Related JP5211183B2 (ja) 2003-02-21 2011-02-03 3−置換−2(アリールアルキル)−1−アザビシクロアルカンおよびこれらの使用方法

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US (11) US6953855B2 (enExample)
EP (1) EP1594869B9 (enExample)
JP (3) JP4828407B2 (enExample)
KR (3) KR101098490B1 (enExample)
CN (2) CN101220026A (enExample)
AT (1) ATE381563T1 (enExample)
AU (1) AU2004215386B2 (enExample)
BR (1) BRPI0407708A (enExample)
CA (1) CA2514135C (enExample)
CY (1) CY1107175T1 (enExample)
DE (1) DE602004010787T2 (enExample)
DK (1) DK1594869T3 (enExample)
EA (1) EA011033B1 (enExample)
ES (1) ES2300749T3 (enExample)
IL (3) IL169797A (enExample)
MX (1) MXPA05008926A (enExample)
NO (3) NO332757B1 (enExample)
NZ (3) NZ565177A (enExample)
PL (3) PL395717A1 (enExample)
PT (1) PT1594869E (enExample)
WO (1) WO2004076449A2 (enExample)
ZA (1) ZA200506515B (enExample)

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EP1697378B1 (en) * 2003-12-22 2007-11-21 Memory Pharmaceuticals Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, and 1,2-benzisothiazoles, and preparation and uses thereof
SE0400708D0 (sv) * 2004-03-22 2004-03-22 Aprea Ab New compounds and use thereof
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US7488737B2 (en) * 2004-04-22 2009-02-10 Memory Pharmaceutical Corporation Indoles, 1H-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof
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