KR101098490B1 - 3­치환­2（아릴알킬）­1­아자바이시클로알칸 및 그 사용방법 - Google Patents

3­치환­2（아릴알킬）­1­아자바이시클로알칸 및 그 사용방법 Download PDF

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KR101098490B1
KR101098490B1 KR1020107026476A KR20107026476A KR101098490B1 KR 101098490 B1 KR101098490 B1 KR 101098490B1 KR 1020107026476 A KR1020107026476 A KR 1020107026476A KR 20107026476 A KR20107026476 A KR 20107026476A KR 101098490 B1 KR101098490 B1 KR 101098490B1
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pyridinyl
azabicyclo
methyl
oct
compounds
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KR20100130239A (ko
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안나톨리 에이. 마주로프
조제프 크루시크
란 미아오
안젤라 에스. 시먼스
테레사 영피터 필립스
제프리 다니엘 슈미트
크레이그 해리슨 밀러
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타가셉트 인코포레이티드
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
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    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0455—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07D487/08—Bridged systems

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  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
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  • Proteomics, Peptides & Aminoacids (AREA)
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KR1020107026476A 2003-02-21 2004-02-20 3­치환­2（아릴알킬）­1­아자바이시클로알칸 및 그 사용방법 Expired - Fee Related KR101098490B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/372,642 2003-02-21
US10/372,642 US6953855B2 (en) 1998-12-11 2003-02-21 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof

Related Parent Applications (1)

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KR1020057015424A Division KR101098481B1 (ko) 2003-02-21 2004-02-20 3-치환-2(아릴알킬)-1-아자바이시클로알칸 및 그 사용방법

Publications (2)

Publication Number Publication Date
KR20100130239A KR20100130239A (ko) 2010-12-10
KR101098490B1 true KR101098490B1 (ko) 2011-12-26

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KR1020107026476A Expired - Fee Related KR101098490B1 (ko) 2003-02-21 2004-02-20 3­치환­2（아릴알킬）­1­아자바이시클로알칸 및 그 사용방법
KR1020057015424A Expired - Fee Related KR101098481B1 (ko) 2003-02-21 2004-02-20 3-치환-2(아릴알킬)-1-아자바이시클로알칸 및 그 사용방법
KR1020107026477A Expired - Fee Related KR101098480B1 (ko) 2003-02-21 2004-02-20 3­치환­2（아릴알킬）­1­아자바이시클로알칸 및 그 사용방법

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KR1020057015424A Expired - Fee Related KR101098481B1 (ko) 2003-02-21 2004-02-20 3-치환-2(아릴알킬)-1-아자바이시클로알칸 및 그 사용방법
KR1020107026477A Expired - Fee Related KR101098480B1 (ko) 2003-02-21 2004-02-20 3­치환­2（아릴알킬）­1­아자바이시클로알칸 및 그 사용방법

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US (11) US6953855B2 (enExample)
EP (1) EP1594869B9 (enExample)
JP (3) JP4828407B2 (enExample)
KR (3) KR101098490B1 (enExample)
CN (2) CN101220026A (enExample)
AT (1) ATE381563T1 (enExample)
AU (1) AU2004215386B2 (enExample)
BR (1) BRPI0407708A (enExample)
CA (1) CA2514135C (enExample)
CY (1) CY1107175T1 (enExample)
DE (1) DE602004010787T2 (enExample)
DK (1) DK1594869T3 (enExample)
EA (1) EA011033B1 (enExample)
ES (1) ES2300749T3 (enExample)
IL (3) IL169797A (enExample)
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NZ (3) NZ565178A (enExample)
PL (3) PL395717A1 (enExample)
PT (1) PT1594869E (enExample)
WO (1) WO2004076449A2 (enExample)
ZA (1) ZA200506515B (enExample)

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DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
GB0220581D0 (en) 2002-09-04 2002-10-09 Novartis Ag Organic Compound
AU2003276919B2 (en) 2002-09-25 2013-05-16 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof
US7750022B2 (en) 2003-08-13 2010-07-06 Neurosearch A/S Quinuclidine derivatives and their pharmaceutical use
PL1697378T3 (pl) 2003-12-22 2008-04-30 Memory Pharm Corp Indole, 1h-indazole, 1,2-benzoizoksazole i 1,2-benzoizotiazole oraz ich wytwarzanie i zastosowania
SE0400708D0 (sv) * 2004-03-22 2004-03-22 Aprea Ab New compounds and use thereof
US20050234095A1 (en) 2004-03-25 2005-10-20 Wenge Xie Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
WO2006001894A1 (en) * 2004-04-22 2006-01-05 Memory Pharmaceutical Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof
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PE20060437A1 (es) 2004-06-18 2006-06-08 Novartis Ag COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR
GB0415746D0 (en) 2004-07-14 2004-08-18 Novartis Ag Organic compounds
JP2008525464A (ja) * 2004-12-22 2008-07-17 メモリー・ファーマシューティカルズ・コーポレイション α−７ニコチン性受容体リガンド並びにその製造及び使用
WO2007001225A1 (en) * 2005-06-29 2007-01-04 Astrazeneca Thiophene-2-carboxamide derivatives as alpha 7 nicotinic receptor modulators.
US20070082939A1 (en) * 2005-07-26 2007-04-12 Lippa Arnold S Methods and compositions for the treatment of neuropathies and related disorders
ATE482959T1 (de) 2005-08-22 2010-10-15 Targacept Inc Heteroarylsubstituierte diazatricycloalkane, verfahren zu deren herstellung und deren anwendung
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CA2623558A1 (en) * 2005-09-27 2007-04-05 Myriad Genetics, Inc. Pyrrole derivatives as therapeutic compounds
GB0521508D0 (en) 2005-10-21 2005-11-30 Novartis Ag Organic compounds
GB0525673D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
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