JP4669611B2 - 化合物 - Google Patents

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Publication number
JP4669611B2
JP4669611B2 JP2000571053A JP2000571053A JP4669611B2 JP 4669611 B2 JP4669611 B2 JP 4669611B2 JP 2000571053 A JP2000571053 A JP 2000571053A JP 2000571053 A JP2000571053 A JP 2000571053A JP 4669611 B2 JP4669611 B2 JP 4669611B2
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compound
formula
mmol
substituents
group
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JP2000571053A
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Japanese (ja)
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JP2002525284A (ja
JP2002525284A5 (enExample
Inventor
サーストン，デイビツド・エドウイン
ハワード，フイリツプ・ウイルソン
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スパイロジエン・リミテツド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2000571053A 1998-08-27 1999-08-27 化合物 Expired - Lifetime JP4669611B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9818731.3 1998-08-27
GBGB9818731.3A GB9818731D0 (en) 1998-08-27 1998-08-27 Compounds
PCT/GB1999/002837 WO2000012507A2 (en) 1998-08-27 1999-08-27 Pyrrolobenzodiazepines

Publications (3)

Publication Number Publication Date
JP2002525284A JP2002525284A (ja) 2002-08-13
JP2002525284A5 JP2002525284A5 (enExample) 2011-01-13
JP4669611B2 true JP4669611B2 (ja) 2011-04-13

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ID=10837953

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000571053A Expired - Lifetime JP4669611B2 (ja) 1998-08-27 1999-08-27 化合物

Country Status (12)

Country Link
US (2) US6562806B1 (enExample)
EP (1) EP1109811B1 (enExample)
JP (1) JP4669611B2 (enExample)
AT (1) ATE246687T1 (enExample)
CA (1) CA2341968C (enExample)
DE (1) DE69910227T2 (enExample)
DK (1) DK1109811T3 (enExample)
ES (1) ES2205872T3 (enExample)
GB (1) GB9818731D0 (enExample)
NZ (1) NZ510492A (enExample)
PT (1) PT1109811E (enExample)
WO (1) WO2000012507A2 (enExample)

Families Citing this family (145)

* Cited by examiner, † Cited by third party
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FR2844273B1 (fr) 2002-09-05 2008-04-04 Aventis Pharma Sa Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens.
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PT1109811E (pt) 2003-12-31
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ATE246687T1 (de) 2003-08-15
US6562806B1 (en) 2003-05-13
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CA2341968C (en) 2009-04-07
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