JP4621939B2 - ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法 - Google Patents

５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法 Download PDF

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Publication number
JP4621939B2
JP4621939B2 JP2004102963A JP2004102963A JP4621939B2 JP 4621939 B2 JP4621939 B2 JP 4621939B2 JP 2004102963 A JP2004102963 A JP 2004102963A JP 2004102963 A JP2004102963 A JP 2004102963A JP 4621939 B2 JP4621939 B2 JP 4621939B2
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group
hydroxy
mmol
branched
linear
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Expired - Lifetime
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JP2004102963A
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English (en)
Japanese (ja)
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JP2005289824A (ja
Inventor
幸生 内田
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Ihara Chemical Industry Co Ltd
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Ihara Chemical Industry Co Ltd
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Application filed by Ihara Chemical Industry Co Ltd filed Critical Ihara Chemical Industry Co Ltd
Priority to JP2004102963A priority Critical patent/JP4621939B2/ja
Priority to CA2560936A priority patent/CA2560936C/en
Priority to AU2005228017A priority patent/AU2005228017B2/en
Priority to EP05728918.3A priority patent/EP1767528B1/en
Priority to TW094110223A priority patent/TWI357899B/zh
Priority to ES05728918.3T priority patent/ES2508765T3/es
Priority to BRPI0509353A priority patent/BRPI0509353B1/pt
Priority to KR1020067019480A priority patent/KR101205731B1/ko
Priority to PL05728918T priority patent/PL1767528T3/pl
Priority to RU2006138241/04A priority patent/RU2386619C2/ru
Priority to NZ550143A priority patent/NZ550143A/en
Priority to PCT/JP2005/006806 priority patent/WO2005095352A1/ja
Priority to MXPA06011130 priority patent/MX280092B/es
Priority to CN2005800106359A priority patent/CN1938278B/zh
Priority to US10/594,710 priority patent/US7488831B2/en
Priority to UAA200611331A priority patent/UA83910C2/ru
Publication of JP2005289824A publication Critical patent/JP2005289824A/ja
Priority to CR8640A priority patent/CR8640A/es
Priority to IL178233A priority patent/IL178233A/en
Priority to IN5581DE2006 priority patent/IN2006DE05581A/en
Publication of JP4621939B2 publication Critical patent/JP4621939B2/ja
Application granted granted Critical
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28—Two oxygen or sulfur atoms
    • C07D231/30—Two oxygen or sulfur atoms attached in positions 3 and 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2004102963A 2004-03-31 2004-03-31 ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法 Expired - Lifetime JP4621939B2 (ja)

Priority Applications (19)

Application Number Priority Date Filing Date Title
JP2004102963A JP4621939B2 (ja) 2004-03-31 2004-03-31 ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法
NZ550143A NZ550143A (en) 2004-03-31 2005-03-31 Process for producing 5-hydroxy-4-thiomethylpyrazole compound
MXPA06011130 MX280092B (es) 2004-03-31 2005-03-31 Proceso para producir un compuesto de 5 - hidroxi - 4 - tiometilpirazol.
EP05728918.3A EP1767528B1 (en) 2004-03-31 2005-03-31 Process for producing 5-hydroxy-4-thiomethylpyrazole compound
TW094110223A TWI357899B (en) 2004-03-31 2005-03-31 Process for producing 5-hydroxy-4-thiomethylpyrazo
ES05728918.3T ES2508765T3 (es) 2004-03-31 2005-03-31 Procedimiento para producir un compuesto de 5-hidroxi-4-tiometilpirazol
BRPI0509353A BRPI0509353B1 (pt) 2004-03-31 2005-03-31 processo para a produção de um composto de 5-hidróxi-4-tiometilpirazol
KR1020067019480A KR101205731B1 (ko) 2004-03-31 2005-03-31 5-히드록시-4-티오메틸피라졸 화합물의 제조 방법
PL05728918T PL1767528T3 (pl) 2004-03-31 2005-03-31 Sposób wytwarzania związku 5-hydroksy-4-tiometylopirazolowego
RU2006138241/04A RU2386619C2 (ru) 2004-03-31 2005-03-31 Способ получения 5-гидрокси-4-тиометилпиразольного соединения
CA2560936A CA2560936C (en) 2004-03-31 2005-03-31 Process for producing 5-hydroxy-4-thiomethylpyrazole compound
PCT/JP2005/006806 WO2005095352A1 (ja) 2004-03-31 2005-03-31 ５－ヒドロキシ－４－チオメチルピラゾール化合物の製造方法
AU2005228017A AU2005228017B2 (en) 2004-03-31 2005-03-31 Process for producing 5-hydroxy-4-thiomethylpyrazole compound
CN2005800106359A CN1938278B (zh) 2004-03-31 2005-03-31 5-羟基-4-硫甲基吡唑化合物的制备方法
US10/594,710 US7488831B2 (en) 2004-03-31 2005-03-31 Process for producing 5-hydroxy-4-thiomethylpyrazole compound
UAA200611331A UA83910C2 (ru) 2004-03-31 2005-03-31 Способ получения 5-гидрокси-4-тиометилпиразольного соединения
CR8640A CR8640A (es) 2004-03-31 2006-09-20 Proceso para producir un compuesto de 5-hidroxi-4-tiometilpirazol
IL178233A IL178233A (en) 2004-03-31 2006-09-21 Process for making 5-hydroxy-4-thiomethylpyrazole
IN5581DE2006 IN2006DE05581A (https=) 2004-03-31 2006-09-25

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2004102963A JP4621939B2 (ja) 2004-03-31 2004-03-31 ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法

Publications (2)

Publication Number Publication Date
JP2005289824A JP2005289824A (ja) 2005-10-20
JP4621939B2 true JP4621939B2 (ja) 2011-02-02

Family

ID=35063690

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004102963A Expired - Lifetime JP4621939B2 (ja) 2004-03-31 2004-03-31 ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法

Country Status (19)

Country Link
US (1) US7488831B2 (https=)
EP (1) EP1767528B1 (https=)
JP (1) JP4621939B2 (https=)
KR (1) KR101205731B1 (https=)
CN (1) CN1938278B (https=)
AU (1) AU2005228017B2 (https=)
BR (1) BRPI0509353B1 (https=)
CA (1) CA2560936C (https=)
CR (1) CR8640A (https=)
ES (1) ES2508765T3 (https=)
IL (1) IL178233A (https=)
IN (1) IN2006DE05581A (https=)
MX (1) MX280092B (https=)
NZ (1) NZ550143A (https=)
PL (1) PL1767528T3 (https=)
RU (1) RU2386619C2 (https=)
TW (1) TWI357899B (https=)
UA (1) UA83910C2 (https=)
WO (1) WO2005095352A1 (https=)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006037945A1 (en) 2004-10-05 2006-04-13 Syngenta Limited Isoxazoline derivatives and their use as herbicides
US7714142B2 (en) * 2004-12-20 2010-05-11 Ihara Chemical Industry Co., Ltd. Process for production of (4,5-dihydroisoxazol-3-Y) thio-carboxamidine salts
JP2007031342A (ja) * 2005-07-27 2007-02-08 Ihara Chem Ind Co Ltd ５−ヒドロキシ−１−アルキルピラゾール誘導体の製造方法
NZ570495A (en) 2006-02-14 2011-10-28 Ihara Chemical Ind Co Process for production of 5-alkoxy-4-hydroxymethylpyrazole compound
EP2167464B1 (en) * 2007-05-25 2014-12-03 AbbVie Deutschland GmbH & Co KG Heterocyclic compounds as positive modulators of metabotropic glutamate receptor 2 (mglu2 receptor)
GB0916267D0 (en) 2009-09-16 2009-10-28 Syngenta Ltd Herbicidal compounds
CN102666502B (zh) 2009-11-26 2015-01-07 巴斯夫欧洲公司 生产5,5-二取代的4,5-二氢异噁唑-3-硫基甲脒盐的方法
CA2781409A1 (en) 2009-11-26 2011-06-03 Basf Se Method for producing 5,5-disubstituted 2-isoxazolines
EP2571854B1 (en) * 2010-05-20 2014-11-05 Bayer Intellectual Property GmbH Method for manufacturing 1-alkyl-3-difluormethyl-5-hydroxypyrazoles
CN103843198B (zh) 2011-07-29 2016-05-04 萨斯喀彻温大学 聚合物基谐振器天线
CN103387541B (zh) * 2012-05-10 2016-02-10 中国中化股份有限公司 一种取代吡唑醚类化合物的制备方法
JP6400247B1 (ja) * 2015-11-16 2018-10-03 ロンザ・リミテッド １−メチル−３−（トリフルオロメチル）−１ｈ−ピラゾール−５−オールの調製方法
TW201835036A (zh) 2017-02-27 2018-10-01 瑞士商隆薩有限公司 製備1-甲基-3-(三氟甲基)-1h-吡唑-5-醇的方法
JP6664036B2 (ja) * 2017-12-27 2020-03-13 クミアイ化学工業株式会社 チオカルボキサミジン塩化合物の製造方法
WO2019230831A1 (ja) * 2018-05-31 2019-12-05 クミアイ化学工業株式会社 含フッ素ピラゾール誘導体の製造方法及びその中間体
AR119524A1 (es) 2019-07-30 2021-12-22 Adama Agan Ltd Proceso e intermediarios para la preparación de piroxasulfona
EP4053125B1 (en) 2019-10-31 2024-12-04 Kumiai Chemical Industry Co., Ltd. Process for the production of a pyroxasulfone herbicide
WO2021176456A1 (en) 2020-03-05 2021-09-10 Adama Agan Ltd. Process and intermediates for the preparation of pyroxasulfone
CN111574511A (zh) * 2020-06-28 2020-08-25 安徽久易农业股份有限公司 一种砜吡草唑的合成方法及其应用
EP4177252A3 (en) 2020-07-10 2023-08-09 Adama Agan Ltd. Process and intermediates for the preparation of pyroxasulfone, fenoxasulfone and various sulfone analogs of 5,5-dimethyl-4h-1,2-oxazole
CN112110912B (zh) * 2020-07-31 2022-07-05 绍兴贝斯美化工股份有限公司 一种合成硫醚类中间体的方法
WO2023074828A1 (ja) 2021-10-29 2023-05-04 クミアイ化学工業株式会社 ジスルフィド化合物、ポリスルフィド化合物及びその用途
AR127776A1 (es) 2021-11-28 2024-02-28 Adama Agan Ltd Composiciones de concentrado en suspensión de alta carga
CN114716428B (zh) * 2022-05-06 2024-02-06 山东潍坊润丰化工股份有限公司 制备砜吡草唑中间体的方法
CN115850178B (zh) * 2022-12-28 2025-04-04 宁夏格瑞精细化工有限公司 一种1-甲基-3-(三氟甲基)-1h-吡唑-5-醇的制备方法
CN117417333B (zh) * 2023-10-07 2026-02-17 安徽久易农业股份有限公司 一种砜吡草唑的合成工艺
CN120590326B (zh) * 2025-06-05 2025-12-23 济南万兴达化工有限公司 一种1-甲基-3-（三氟甲基）-1h-吡唑-5-醇的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
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US4918085A (en) * 1989-03-02 1990-04-17 Rhone-Poulenc Ag Company Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles, compositions and use
CO5221057A1 (es) * 2000-03-02 2002-11-28 Aventis Cropscience Sa Componentes y composiciones plagicidas
JP4465133B2 (ja) * 2001-02-08 2010-05-19 クミアイ化学工業株式会社 イソオキサゾリン誘導体及びこれを有効成分とする除草剤
EP1405853B1 (en) * 2001-06-21 2010-11-03 Kumiai Chemical Industry Co., Ltd. Isoxazoline derivatives and herbicides
AU2003252447B2 (en) * 2002-08-01 2008-06-05 Kumiai Chemical Industry Co., Ltd. Pyrazole derivatives and process for the production thereof
UA78071C2 (en) * 2002-08-07 2007-02-15 Kumiai Chemical Industry Co Herbicidal composition

Also Published As

Publication number Publication date
RU2006138241A (ru) 2008-05-10
CA2560936A1 (en) 2005-10-13
IN2006DE05581A (https=) 2007-08-31
EP1767528B1 (en) 2014-09-17
KR101205731B1 (ko) 2012-11-28
TW200536832A (en) 2005-11-16
KR20070003964A (ko) 2007-01-05
MX280092B (es) 2010-10-18
MXPA06011130A (es) 2007-01-25
NZ550143A (en) 2010-04-30
AU2005228017B2 (en) 2010-09-30
WO2005095352A1 (ja) 2005-10-13
BRPI0509353A8 (pt) 2017-09-19
CR8640A (es) 2007-08-28
BRPI0509353B1 (pt) 2019-01-02
US20070185334A1 (en) 2007-08-09
BRPI0509353A (pt) 2007-09-11
RU2386619C2 (ru) 2010-04-20
IL178233A (en) 2014-02-27
IL178233A0 (en) 2006-12-31
CN1938278B (zh) 2012-12-12
PL1767528T3 (pl) 2015-03-31
ES2508765T3 (es) 2014-10-16
CA2560936C (en) 2013-01-08
TWI357899B (en) 2012-02-11
CN1938278A (zh) 2007-03-28
JP2005289824A (ja) 2005-10-20
EP1767528A4 (en) 2010-04-21
AU2005228017A1 (en) 2005-10-13
EP1767528A1 (en) 2007-03-28
UA83910C2 (ru) 2008-08-26
US7488831B2 (en) 2009-02-10

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