JP2021528451A5 - - Google Patents

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Publication number
JP2021528451A5
JP2021528451A5 JP2020572372A JP2020572372A JP2021528451A5 JP 2021528451 A5 JP2021528451 A5 JP 2021528451A5 JP 2020572372 A JP2020572372 A JP 2020572372A JP 2020572372 A JP2020572372 A JP 2020572372A JP 2021528451 A5 JP2021528451 A5 JP 2021528451A5
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Japan
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alkylene
alkyl
halo
independently selected
membered
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JP2020572372A
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English (en)
Japanese (ja)
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JP7214086B2 (ja
JP2021528451A (ja
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Priority claimed from PCT/EP2019/067351 external-priority patent/WO2020002611A1/en
Publication of JP2021528451A publication Critical patent/JP2021528451A/ja
Publication of JP2021528451A5 publication Critical patent/JP2021528451A5/ja
Application granted granted Critical
Publication of JP7214086B2 publication Critical patent/JP7214086B2/ja
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JP2020572372A 2018-06-28 2019-06-28 二環式コア部分を有する新規lxrモジュレーター Active JP7214086B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18180450.1 2018-06-28
EP18180450 2018-06-28
PCT/EP2019/067351 WO2020002611A1 (en) 2018-06-28 2019-06-28 Novel lxr modulators with bicyclic core moiety

Publications (3)

Publication Number Publication Date
JP2021528451A JP2021528451A (ja) 2021-10-21
JP2021528451A5 true JP2021528451A5 (enExample) 2022-06-16
JP7214086B2 JP7214086B2 (ja) 2023-01-30

Family

ID=62947921

Family Applications (1)

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JP2020572372A Active JP7214086B2 (ja) 2018-06-28 2019-06-28 二環式コア部分を有する新規lxrモジュレーター

Country Status (27)

Country Link
US (3) US11618747B2 (enExample)
EP (1) EP3814331B9 (enExample)
JP (1) JP7214086B2 (enExample)
KR (1) KR102678581B1 (enExample)
CN (1) CN112689630A (enExample)
AR (1) AR117599A1 (enExample)
AU (1) AU2019293727B2 (enExample)
BR (1) BR112020026405A2 (enExample)
CA (1) CA3104956C (enExample)
CL (1) CL2020003300A1 (enExample)
DK (1) DK3814331T3 (enExample)
EA (1) EA202092821A1 (enExample)
ES (1) ES2956045T3 (enExample)
FI (1) FI3814331T3 (enExample)
HU (1) HUE063538T2 (enExample)
IL (2) IL310623A (enExample)
LT (1) LT3814331T (enExample)
MX (1) MX2020014258A (enExample)
PH (1) PH12020552269A1 (enExample)
PL (1) PL3814331T3 (enExample)
PT (1) PT3814331T (enExample)
PY (1) PY1950412A (enExample)
SI (1) SI3814331T1 (enExample)
SM (1) SMT202300334T1 (enExample)
TW (1) TWI748194B (enExample)
UY (1) UY38283A (enExample)
WO (1) WO2020002611A1 (enExample)

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CN118791407A (zh) 2018-05-22 2024-10-18 奥索生物公司 亚磺酰基氨基苯甲酰胺以及磺酰基氨基苯甲酰胺衍生物
TWI748194B (zh) 2018-06-28 2021-12-01 德商菲尼克斯 Fxr有限責任公司 含有雙環核心部分之新穎lxr調節劑
US20230159502A1 (en) * 2020-04-03 2023-05-25 Vertex Pharmaceuticals Incorporated Indole derivatives as alpha-1-antitrypsin modulators for treating alpha-1-antitrypsin deficiency (aatd)
WO2021203014A1 (en) 2020-04-03 2021-10-07 Vertex Pharmaceuticals Incorporated Pyrano[4,3-b]l ndole derivatives as alpha-1 -antitrypsin modulators for treating alpha-1 -antitrypsin deficiency (aatd)
EP4126863A1 (en) 2020-04-03 2023-02-08 Vertex Pharmaceuticals Incorporated 1 h-pyrazolo[4,3-g]isoquinoline and 1 h-pyrazolo[4,3-g]quinoline derivatives as alpha-1 -antitrypsin modulators for treating alpha-1 -antitrypsin deficiency (aatd)
WO2024097897A1 (en) * 2022-11-03 2024-05-10 Orsobio, Inc. Lxr modulators with bicyclic core moiety for treating dyslipidemias

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TWI748194B (zh) 2018-06-28 2021-12-01 德商菲尼克斯 Fxr有限責任公司 含有雙環核心部分之新穎lxr調節劑
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