JP2019511466A5 - - Google Patents

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JP2019511466A5
JP2019511466A5 JP2018542231A JP2018542231A JP2019511466A5 JP 2019511466 A5 JP2019511466 A5 JP 2019511466A5 JP 2018542231 A JP2018542231 A JP 2018542231A JP 2018542231 A JP2018542231 A JP 2018542231A JP 2019511466 A5 JP2019511466 A5 JP 2019511466A5
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JP6883045B2 (ja
JP2019511466A (ja
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Priority claimed from PCT/US2017/017408 external-priority patent/WO2017139603A1/en
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JP2018542231A 2016-02-12 2017-02-10 オレキシン受容体調節因子としてのハロ置換ピペリジン Active JP6883045B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201662294940P 2016-02-12 2016-02-12
US62/294,940 2016-02-12
US201662336102P 2016-05-13 2016-05-13
US62/336,102 2016-05-13
PCT/US2017/017408 WO2017139603A1 (en) 2016-02-12 2017-02-10 Halo-substituted piperidines as orexin receptor modulators

Publications (3)

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JP2019511466A JP2019511466A (ja) 2019-04-25
JP2019511466A5 true JP2019511466A5 (enExample) 2020-03-19
JP6883045B2 JP6883045B2 (ja) 2021-06-02

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JP2018542231A Active JP6883045B2 (ja) 2016-02-12 2017-02-10 オレキシン受容体調節因子としてのハロ置換ピペリジン

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US (4) US10894789B2 (enExample)
EP (1) EP3414241B1 (enExample)
JP (1) JP6883045B2 (enExample)
KR (1) KR102738491B1 (enExample)
CN (1) CN109219606B (enExample)
AU (1) AU2017217931B2 (enExample)
BR (1) BR112018016446B1 (enExample)
CA (1) CA3013927C (enExample)
CL (1) CL2018002121A1 (enExample)
CO (1) CO2018009290A2 (enExample)
CR (1) CR20180429A (enExample)
CY (1) CY1125461T1 (enExample)
DK (1) DK3414241T3 (enExample)
DO (1) DOP2018000179A (enExample)
EA (1) EA036542B9 (enExample)
ES (1) ES2923790T3 (enExample)
HR (1) HRP20220906T1 (enExample)
HU (1) HUE059280T2 (enExample)
IL (1) IL260788B (enExample)
LT (1) LT3414241T (enExample)
MX (1) MX2018009656A (enExample)
MY (1) MY195239A (enExample)
PH (1) PH12018501708A1 (enExample)
PL (1) PL3414241T3 (enExample)
PT (1) PT3414241T (enExample)
RS (1) RS63471B1 (enExample)
SG (1) SG11201806368VA (enExample)
SI (1) SI3414241T1 (enExample)
SM (1) SMT202200323T1 (enExample)
SV (1) SV2018005731A (enExample)
TN (1) TN2018000280A1 (enExample)
TW (1) TWI710557B (enExample)
WO (1) WO2017139603A1 (enExample)
ZA (1) ZA201805839B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3414241T3 (pl) 2016-02-12 2022-10-03 Astrazeneca Ab Piperydyny podstawione halo jako modulatory receptora oreksyny
AU2018326734B2 (en) 2017-09-01 2023-08-17 Chronos Therapeutics Limited Substituted 2-azabicyclo(3.1.1)heptane and 2-azabicyclo(3.2.1)octane derivatives as orexin receptor antagonists
JP6874217B2 (ja) * 2017-09-28 2021-05-19 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規なｎ−（２，２−ジフルオロエチル）−ｎ−［（ピリミジニルアミノ）プロパニル］アリールカルボキサミド
US20210169883A1 (en) * 2018-07-27 2021-06-10 Icahn School Of Medicine At Mount Sinai Method of treating aggression with orexin receptor antagonists
WO2021085550A1 (ja) 2019-11-01 2021-05-06 ユニマテック株式会社 含フッ素ピリミジン化合物およびその製造方法
GB202311281D0 (en) 2023-07-21 2023-09-06 Bial Portela & Ca Sa Orexin receptor antagonists
GB202311280D0 (en) 2023-07-21 2023-09-06 Bial Portela & Ca Sa Orexin receptor antagonists

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