JP2017503867A5 - - Google Patents

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JP2017503867A5
JP2017503867A5 JP2016566857A JP2016566857A JP2017503867A5 JP 2017503867 A5 JP2017503867 A5 JP 2017503867A5 JP 2016566857 A JP2016566857 A JP 2016566857A JP 2016566857 A JP2016566857 A JP 2016566857A JP 2017503867 A5 JP2017503867 A5 JP 2017503867A5
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fluoro
ethenopyrazolo
methyl
tetrahydro
alkyl
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JP2017503867A (ja
JP6490713B2 (ja
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JP2016566857A 2014-01-24 2015-01-23 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物 Active JP6490713B2 (ja)

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Application Number Priority Date Filing Date Title
US201461931506P 2014-01-24 2014-01-24
US61/931,506 2014-01-24
US201462049326P 2014-09-11 2014-09-11
US62/049,326 2014-09-11
US201562106301P 2015-01-22 2015-01-22
US62/106,301 2015-01-22
PCT/US2015/012597 WO2015112806A2 (en) 2014-01-24 2015-01-23 Diaryl macrocycles as modulators of protein kinases

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JP2019034652A Division JP2019104748A (ja) 2014-01-24 2019-02-27 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物

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JP2017503867A JP2017503867A (ja) 2017-02-02
JP2017503867A5 true JP2017503867A5 (enExample) 2018-03-08
JP6490713B2 JP6490713B2 (ja) 2019-03-27

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JP2016566857A Active JP6490713B2 (ja) 2014-01-24 2015-01-23 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2019034652A Withdrawn JP2019104748A (ja) 2014-01-24 2019-02-27 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2021001588A Pending JP2021063121A (ja) 2014-01-24 2021-01-07 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2022110613A Active JP7356546B2 (ja) 2014-01-24 2022-07-08 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2023158350A Ceased JP2023179539A (ja) 2014-01-24 2023-09-22 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物

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JP2019034652A Withdrawn JP2019104748A (ja) 2014-01-24 2019-02-27 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2021001588A Pending JP2021063121A (ja) 2014-01-24 2021-01-07 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2022110613A Active JP7356546B2 (ja) 2014-01-24 2022-07-08 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物
JP2023158350A Ceased JP2023179539A (ja) 2014-01-24 2023-09-22 タンパク質キナーゼのモジュレータとしてのジアリール大環状化合物

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US (7) US9714258B2 (enExample)
EP (6) EP3636650A1 (enExample)
JP (5) JP6490713B2 (enExample)
KR (1) KR102402179B1 (enExample)
CN (3) CN106170289B (enExample)
AP (1) AP2016009383A0 (enExample)
AU (2) AU2015209239C1 (enExample)
CA (1) CA2936079C (enExample)
CL (1) CL2016001876A1 (enExample)
CY (3) CY1121850T1 (enExample)
DK (3) DK3572416T3 (enExample)
EA (2) EA031863B1 (enExample)
ES (3) ES2976459T3 (enExample)
FI (2) FI3636649T3 (enExample)
FR (1) FR25C1013I2 (enExample)
HR (3) HRP20221518T1 (enExample)
HU (4) HUE060554T2 (enExample)
IL (2) IL246860B (enExample)
LT (4) LT3097107T (enExample)
MX (2) MX2016009588A (enExample)
MY (1) MY193524A (enExample)
NL (1) NL301322I2 (enExample)
NO (1) NO2025015I1 (enExample)
NZ (2) NZ722375A (enExample)
PE (1) PE20160931A1 (enExample)
PH (1) PH12016501463A1 (enExample)
PL (3) PL3636649T3 (enExample)
PT (3) PT3097107T (enExample)
RS (3) RS59059B1 (enExample)
SG (2) SG10202000191YA (enExample)
SI (3) SI3636649T1 (enExample)
SM (3) SMT201900388T1 (enExample)
UA (1) UA121206C2 (enExample)
WO (1) WO2015112806A2 (enExample)
ZA (2) ZA201604654B (enExample)

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