JP2017222697A5 - - Google Patents
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- Publication number
- JP2017222697A5 JP2017222697A5 JP2017142601A JP2017142601A JP2017222697A5 JP 2017222697 A5 JP2017222697 A5 JP 2017222697A5 JP 2017142601 A JP2017142601 A JP 2017142601A JP 2017142601 A JP2017142601 A JP 2017142601A JP 2017222697 A5 JP2017222697 A5 JP 2017222697A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- buten
- fluorophenyl
- bromo
- bis
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims 5
- -1 3- (2-bromo-4-fluorophenyl) -4,4-bis (methylthio) -3-buten-2-one Chemical compound 0.000 claims 3
- 150000001204 N-oxides Chemical class 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15704609P | 2009-03-03 | 2009-03-03 | |
| US61/157,046 | 2009-03-03 | ||
| US30405310P | 2010-02-12 | 2010-02-12 | |
| US61/304,053 | 2010-02-12 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011553063A Division JP6285090B2 (ja) | 2009-03-03 | 2010-03-03 | 殺菌・殺カビ性ピラゾール |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017222697A JP2017222697A (ja) | 2017-12-21 |
| JP2017222697A5 true JP2017222697A5 (https=) | 2018-02-08 |
| JP6641326B2 JP6641326B2 (ja) | 2020-02-05 |
Family
ID=42139982
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011553063A Active JP6285090B2 (ja) | 2009-03-03 | 2010-03-03 | 殺菌・殺カビ性ピラゾール |
| JP2015102333A Withdrawn JP2015172062A (ja) | 2009-03-03 | 2015-05-20 | 殺菌・殺カビ性ピラゾール |
| JP2016252244A Withdrawn JP2017081965A (ja) | 2009-03-03 | 2016-12-27 | 殺菌・殺カビ性ピラゾール |
| JP2017142601A Active JP6641326B2 (ja) | 2009-03-03 | 2017-07-24 | 殺菌・殺カビ性ピラゾール |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011553063A Active JP6285090B2 (ja) | 2009-03-03 | 2010-03-03 | 殺菌・殺カビ性ピラゾール |
| JP2015102333A Withdrawn JP2015172062A (ja) | 2009-03-03 | 2015-05-20 | 殺菌・殺カビ性ピラゾール |
| JP2016252244A Withdrawn JP2017081965A (ja) | 2009-03-03 | 2016-12-27 | 殺菌・殺カビ性ピラゾール |
Country Status (30)
| Country | Link |
|---|---|
| US (5) | US9062005B2 (https=) |
| EP (2) | EP2403834B1 (https=) |
| JP (4) | JP6285090B2 (https=) |
| KR (1) | KR101752925B1 (https=) |
| CN (2) | CN102421756A (https=) |
| AR (1) | AR075713A1 (https=) |
| AU (1) | AU2010221440B2 (https=) |
| BR (1) | BRPI1005812B8 (https=) |
| CA (1) | CA2750862C (https=) |
| CO (1) | CO6361933A2 (https=) |
| DK (1) | DK2403834T3 (https=) |
| ES (1) | ES2562178T3 (https=) |
| GE (1) | GEP20156211B (https=) |
| HR (1) | HRP20160111T1 (https=) |
| HU (1) | HUE026926T2 (https=) |
| IL (1) | IL214184A (https=) |
| ME (1) | ME02349B (https=) |
| MX (1) | MX2011008900A (https=) |
| MY (1) | MY159364A (https=) |
| NZ (1) | NZ594181A (https=) |
| PE (2) | PE20130039A1 (https=) |
| PL (1) | PL2403834T3 (https=) |
| PT (1) | PT2403834E (https=) |
| RS (1) | RS54531B1 (https=) |
| RU (1) | RU2577247C2 (https=) |
| SI (1) | SI2403834T1 (https=) |
| TW (1) | TWI548344B (https=) |
| UA (1) | UA124518C2 (https=) |
| WO (1) | WO2010101973A1 (https=) |
| ZA (1) | ZA201105391B (https=) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR075713A1 (es) * | 2009-03-03 | 2011-04-20 | Du Pont | Pirazoles fungicidas |
| TW201245155A (en) | 2010-09-01 | 2012-11-16 | Du Pont | Fungicidal pyrazoles |
| TWI504350B (zh) * | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
| TWI568721B (zh) | 2012-02-01 | 2017-02-01 | 杜邦股份有限公司 | 殺真菌之吡唑混合物 |
| WO2013126283A1 (en) | 2012-02-20 | 2013-08-29 | E. I. Du Pont De Nemours And Company | Fungicidal pyrazoles |
| EP2864293B1 (en) * | 2012-06-22 | 2016-04-27 | E. I. du Pont de Nemours and Company | Fungicidal 4-methylanilino pyrazoles |
| EP3010908A1 (en) | 2013-02-20 | 2016-04-27 | E. I. du Pont de Nemours and Company | Fungicidal pyrazoles |
| US20140235689A1 (en) * | 2013-02-20 | 2014-08-21 | E I Du Pont De Nemours And Company | Fungicidal pyrazoles |
| US20140288074A1 (en) * | 2013-03-22 | 2014-09-25 | E I Du Pont De Nemours And Company | Fungicidal pyrazoles |
| TWI652012B (zh) * | 2013-05-20 | 2019-03-01 | 杜邦股份有限公司 | 殺真菌吡唑的固態形式 |
| WO2015026646A1 (en) | 2013-08-20 | 2015-02-26 | E. I. Du Pont De Nemours And Company | Fungicidal pyrazoles |
| TWI652014B (zh) * | 2013-09-13 | 2019-03-01 | 美商艾佛艾姆希公司 | 雜環取代之雙環唑殺蟲劑 |
| CN106458925A (zh) | 2014-05-06 | 2017-02-22 | 杜邦公司 | 杀真菌吡唑类 |
| JP2017522334A (ja) | 2014-07-24 | 2017-08-10 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 殺真菌性ピラゾール誘導体 |
| WO2016026830A1 (en) * | 2014-08-21 | 2016-02-25 | Bayer Cropscience Aktiengesellschaft | Novel fungicidal pyrazole derivatives |
| CA2978066A1 (en) | 2015-03-19 | 2016-09-22 | E I Du Pont De Nemours And Company | Fungicidal pyrazoles |
| ES2911341T3 (es) * | 2015-04-29 | 2022-05-18 | The State Of Israel Ministry Of Agriculture & Rural Development Agricultural Res Organization Aro Vo | Composiciones antifitopatogénicas |
| CA2988493A1 (en) * | 2015-06-01 | 2016-12-08 | Ishihara Sangyo Kaisha, Ltd. | Fungicide composition and plant disease control method |
| US11214565B2 (en) | 2015-11-20 | 2022-01-04 | Denali Therapeutics Inc. | Compound, compositions, and methods |
| US11028080B2 (en) | 2016-03-11 | 2021-06-08 | Denali Therapeutics Inc. | Substituted pyrimidines as LRKK2 inhibitors |
| MD3472153T2 (ro) | 2016-06-16 | 2022-03-31 | Denali Therapeutics Inc | Pirimidin-2-ilamino-1H-pirazoli în calitate de inhibitori L RRK2 pentru utilizare în tratamentul tulburărilor neurodegenerative |
| WO2018052838A1 (en) | 2016-09-16 | 2018-03-22 | E. I. Du Pont De Nemours And Company | Fungicidal pyrazoles |
| CN107286097B (zh) * | 2017-07-13 | 2019-06-25 | 青岛清原化合物有限公司 | 双唑草酮c晶型及其制备方法和用途 |
| DK3904350T3 (da) | 2018-04-12 | 2023-11-13 | Bayer Ag | N-(cyclopropylmethyl)-5-(methylsulfonyl)-n-{1-[1-(pyrimidin-2-yl)-1h-1,2,4-triazol-5-yl]ethyl}benzamidderivater og de tilsvarende pyridincarboxamidderivater som pesticider |
| TWI819078B (zh) * | 2018-09-06 | 2023-10-21 | 美商富曼西公司 | 殺真菌之經硝苯胺基取代之吡唑 |
| AU2019337618A1 (en) * | 2018-09-14 | 2021-04-01 | Fmc Corporation | Fungicidal halomethyl ketones and hydrates |
| TWI912287B (zh) | 2020-03-11 | 2026-01-21 | 美商富曼西公司 | 殺真菌劑混合物 |
| CN113549053B (zh) * | 2020-04-23 | 2022-09-13 | 沈阳中化农药化工研发有限公司 | 一种吡唑喹（唑）啉醚类化合物及其应用 |
| US20240324596A1 (en) * | 2023-03-28 | 2024-10-03 | Fmc Corporation | Substituted tolyl fungicides |
| CN119504619B (zh) * | 2024-10-10 | 2026-02-17 | 江苏省农业科学院 | 具有抗真菌活性的化合物及其制备方法和应用 |
Family Cites Families (49)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2891855A (en) | 1954-08-16 | 1959-06-23 | Geigy Ag J R | Compositions and methods for influencing the growth of plants |
| US3235361A (en) | 1962-10-29 | 1966-02-15 | Du Pont | Method for the control of undesirable vegetation |
| US3060084A (en) | 1961-06-09 | 1962-10-23 | Du Pont | Improved homogeneous, readily dispersed, pesticidal concentrate |
| US3299566A (en) | 1964-06-01 | 1967-01-24 | Olin Mathieson | Water soluble film containing agricultural chemicals |
| US3309192A (en) | 1964-12-02 | 1967-03-14 | Du Pont | Method of controlling seedling weed grasses |
| US4144050A (en) | 1969-02-05 | 1979-03-13 | Hoechst Aktiengesellschaft | Micro granules for pesticides and process for their manufacture |
| US3920442A (en) | 1972-09-18 | 1975-11-18 | Du Pont | Water-dispersible pesticide aggregates |
| US4172714A (en) | 1976-12-20 | 1979-10-30 | E. I. Du Pont De Nemours And Company | Dry compactible, swellable herbicidal compositions and pellets produced therefrom |
| DK569478A (da) | 1977-12-23 | 1979-07-02 | Montedison Spa | Phosphor og thiophosphorsyreestere af substituerede hydroxypyrazoler samt fremgangsmaade til fremstilling deraf |
| GB2054555A (en) | 1979-07-27 | 1981-02-18 | Abbott Lab | Pyrazolyl amino imidazolines |
| GB2076801A (en) * | 1980-04-14 | 1981-12-09 | Erba Farmitalia | alpha , beta -Disubstituted Acrylamido Cephalosporins |
| GB2095558B (en) | 1981-03-30 | 1984-10-24 | Avon Packers Ltd | Formulation of agricultural chemicals |
| DE3246493A1 (de) | 1982-12-16 | 1984-06-20 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von wasserdispergierbaren granulaten |
| JPH01319478A (ja) * | 1988-06-20 | 1989-12-25 | Mitsui Toatsu Chem Inc | 免疫調節作用を有する化合物 |
| US5180587A (en) | 1988-06-28 | 1993-01-19 | E. I. Du Pont De Nemours And Company | Tablet formulations of pesticides |
| DE69033861T2 (de) | 1989-08-30 | 2002-06-06 | Kynoch Agrochemicals (Proprietary) Ltd., Sandton | Herstellung eines Dosierungsmittels |
| ES2065680T3 (es) | 1990-03-12 | 1995-02-16 | Du Pont | Granulos de plaguicida dispersables en agua o solubles en agua a partir de aglutinantes activados por calor. |
| US5189040A (en) * | 1990-05-28 | 1993-02-23 | Sumitomo Chemical Company, Limited | Pyrazole derivatives, method for producing the same and agricultural and/or horticultural fungicides containing the same as active ingredient |
| EP0480679B1 (en) | 1990-10-11 | 1996-09-18 | Sumitomo Chemical Company Limited | Pesticidal composition |
| FR2676057B1 (fr) * | 1991-05-02 | 1995-03-03 | Therapeutique Moder Lab | Derives de 1,2-dithiole-3-thione, procede de preparation de ces derives, ainsi que l'utilisation de ces derives comme intermediaires de synthese ou comme medicaments. |
| FR2682379B1 (fr) * | 1991-10-09 | 1994-02-11 | Rhone Poulenc Agrochimie | Nouveaux phenylpyrazoles fongicides. |
| WO1993019054A1 (en) * | 1992-03-26 | 1993-09-30 | Dowelanco | N-heterocyclic nitro anilines as fungicides |
| JPH0665237A (ja) * | 1992-05-07 | 1994-03-08 | Nissan Chem Ind Ltd | 置換ピラゾール誘導体および農園芸用殺菌剤 |
| SK140295A3 (en) | 1993-05-12 | 1996-09-04 | Du Pont | Condensed bicyclic pyrimidinones, fungicidal agents on their base and inhibition method of plant deseases by using them |
| JPH0816059B2 (ja) * | 1993-05-21 | 1996-02-21 | 三井東圧化学株式会社 | 免疫調節剤 |
| DE4405207A1 (de) * | 1994-02-18 | 1995-08-24 | Bayer Ag | N-Pyrazolylaniline und N-Pyrazolylaminopyridine |
| JPH08208620A (ja) * | 1995-02-03 | 1996-08-13 | Takeda Chem Ind Ltd | アミノピラゾール誘導体、その製造法および用途 |
| BR9609613A (pt) | 1995-07-05 | 1999-05-25 | Du Pont | Composto composição fungicida e método de controle de doenças de plantas |
| JPH09208620A (ja) | 1996-02-02 | 1997-08-12 | Sumitomo Bakelite Co Ltd | 硬化性エラストマー及びその製造方法 |
| ATE216999T1 (de) | 1996-03-11 | 2002-05-15 | Syngenta Participations Ag | Pyrimidin-4-on derivate als pestizidesmittel |
| AU7726898A (en) * | 1997-05-22 | 1998-12-11 | G.D. Searle & Co. | Pyrazole derivatives as p38 kinase inhibitors |
| GB9719411D0 (en) | 1997-09-12 | 1997-11-12 | Ciba Geigy Ag | New Pesticides |
| JP2000095778A (ja) * | 1998-09-28 | 2000-04-04 | Ube Ind Ltd | ピラゾール誘導体、その製造法及び農園芸用の殺菌剤 |
| DE10136065A1 (de) | 2001-07-25 | 2003-02-13 | Bayer Cropscience Ag | Pyrazolylcarboxanilide |
| TWI283164B (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| AR042067A1 (es) | 2002-11-27 | 2005-06-08 | Bayer Pharmaceuticals Corp | Derivados de anilinopirazol utiles en el tratamiento de la diabetes |
| GB0315657D0 (en) | 2003-07-03 | 2003-08-13 | Astex Technology Ltd | Pharmaceutical compounds |
| US7517998B2 (en) | 2004-06-01 | 2009-04-14 | Boehringer Ingelheim International Gmbh | Non nucleoside reverse transcriptase inhibitors |
| CA2620425A1 (en) | 2005-08-31 | 2007-03-08 | Bayer Healthcare Llc | Anilinopyrazole derivatives useful for the treatment of diabetes |
| MX2008015648A (es) | 2006-06-21 | 2009-01-09 | Du Pont | Pirazinonas como inhibidores de proliferacion celular. |
| WO2008093639A1 (ja) * | 2007-01-29 | 2008-08-07 | Takeda Pharmaceutical Company Limited | ピラゾール化合物 |
| PE20091953A1 (es) * | 2008-05-08 | 2010-01-09 | Du Pont | Azoles sustituidos como fungicidas |
| AR075713A1 (es) * | 2009-03-03 | 2011-04-20 | Du Pont | Pirazoles fungicidas |
| WO2011051958A1 (en) | 2009-10-30 | 2011-05-05 | E.I. Du Pont De Nemours And Company | Fungicidal pyrazolones |
| TW201117722A (en) | 2009-11-04 | 2011-06-01 | Du Pont | Fungicidal mixtures |
| WO2012023143A1 (en) | 2010-08-19 | 2012-02-23 | E. I. Du Pont De Nemours And Company | Fungicidal pyrazoles |
| TWI504350B (zh) | 2010-09-01 | 2015-10-21 | Du Pont | 殺真菌吡唑及其混合物 |
| TW201245155A (en) | 2010-09-01 | 2012-11-16 | Du Pont | Fungicidal pyrazoles |
| AU2011307289A1 (en) | 2010-09-29 | 2013-02-21 | E. I. Du Pont De Nemours And Company | Fungicidal imidazoles |
-
2010
- 2010-03-02 AR ARP100100624A patent/AR075713A1/es active IP Right Grant
- 2010-03-03 BR BRPI1005812A patent/BRPI1005812B8/pt active IP Right Grant
- 2010-03-03 MX MX2011008900A patent/MX2011008900A/es active IP Right Grant
- 2010-03-03 HR HRP20160111T patent/HRP20160111T1/hr unknown
- 2010-03-03 CA CA2750862A patent/CA2750862C/en active Active
- 2010-03-03 NZ NZ594181A patent/NZ594181A/xx unknown
- 2010-03-03 MY MYPI2011003394A patent/MY159364A/en unknown
- 2010-03-03 PE PE2012001543A patent/PE20130039A1/es active IP Right Grant
- 2010-03-03 JP JP2011553063A patent/JP6285090B2/ja active Active
- 2010-03-03 PT PT107071870T patent/PT2403834E/pt unknown
- 2010-03-03 CN CN2010800198065A patent/CN102421756A/zh active Pending
- 2010-03-03 WO PCT/US2010/026003 patent/WO2010101973A1/en not_active Ceased
- 2010-03-03 DK DK10707187.0T patent/DK2403834T3/en active
- 2010-03-03 CN CN201710017930.1A patent/CN107011326B/zh active Active
- 2010-03-03 ME MEP-2016-26A patent/ME02349B/me unknown
- 2010-03-03 TW TW099106178A patent/TWI548344B/zh active
- 2010-03-03 EP EP10707187.0A patent/EP2403834B1/en active Active
- 2010-03-03 US US13/254,205 patent/US9062005B2/en active Active
- 2010-03-03 RS RS20160051A patent/RS54531B1/sr unknown
- 2010-03-03 AU AU2010221440A patent/AU2010221440B2/en active Active
- 2010-03-03 RU RU2011139893/04A patent/RU2577247C2/ru active
- 2010-03-03 HU HUE10707187A patent/HUE026926T2/en unknown
- 2010-03-03 EP EP15178327.1A patent/EP2966063A1/en not_active Withdrawn
- 2010-03-03 ES ES10707187.0T patent/ES2562178T3/es active Active
- 2010-03-03 SI SI201031129T patent/SI2403834T1/sl unknown
- 2010-03-03 GE GEAP201012393A patent/GEP20156211B/en unknown
- 2010-03-03 UA UAA201109619A patent/UA124518C2/uk unknown
- 2010-03-03 PL PL10707187T patent/PL2403834T3/pl unknown
- 2010-03-03 PE PE2011001568A patent/PE20120101A1/es not_active Application Discontinuation
- 2010-03-03 KR KR1020117023011A patent/KR101752925B1/ko active Active
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2011
- 2011-07-19 IL IL214184A patent/IL214184A/en active IP Right Grant
- 2011-07-21 ZA ZA2011/05391A patent/ZA201105391B/en unknown
- 2011-09-01 CO CO11112622A patent/CO6361933A2/es active IP Right Grant
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2015
- 2015-04-24 US US14/695,689 patent/US9655361B2/en active Active
- 2015-05-20 JP JP2015102333A patent/JP2015172062A/ja not_active Withdrawn
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2016
- 2016-12-27 JP JP2016252244A patent/JP2017081965A/ja not_active Withdrawn
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2017
- 2017-04-25 US US15/496,048 patent/US20170223959A1/en not_active Abandoned
- 2017-07-24 JP JP2017142601A patent/JP6641326B2/ja active Active
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2018
- 2018-10-29 US US16/173,167 patent/US10448639B2/en active Active
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2019
- 2019-09-17 US US16/572,759 patent/US20200008425A1/en not_active Abandoned