JP2016512243A5 - - Google Patents

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JP2016512243A5
JP2016512243A5 JP2016500154A JP2016500154A JP2016512243A5 JP 2016512243 A5 JP2016512243 A5 JP 2016512243A5 JP 2016500154 A JP2016500154 A JP 2016500154A JP 2016500154 A JP2016500154 A JP 2016500154A JP 2016512243 A5 JP2016512243 A5 JP 2016512243A5
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JP6479749B2 (ja
JP2016512243A (ja
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Priority claimed from PCT/US2014/000058 external-priority patent/WO2014149139A2/en
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JP2016500154A 2013-03-15 2014-03-17 トロンビン阻害剤としてのハロゲノピラゾール Active JP6479749B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361789358P 2013-03-15 2013-03-15
US61/789,358 2013-03-15
US201361899588P 2013-11-04 2013-11-04
US61/899,588 2013-11-04
PCT/US2014/000058 WO2014149139A2 (en) 2013-03-15 2014-03-17 Halogenopyrazoles as inhibitors of thrombin

Related Child Applications (1)

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JP2019019308A Division JP2019081782A (ja) 2013-03-15 2019-02-06 トロンビン阻害剤としてのハロゲノピラゾール

Publications (3)

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JP2016512243A JP2016512243A (ja) 2016-04-25
JP2016512243A5 true JP2016512243A5 (enExample) 2017-04-20
JP6479749B2 JP6479749B2 (ja) 2019-03-06

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JP2016500154A Active JP6479749B2 (ja) 2013-03-15 2014-03-17 トロンビン阻害剤としてのハロゲノピラゾール
JP2019019308A Pending JP2019081782A (ja) 2013-03-15 2019-02-06 トロンビン阻害剤としてのハロゲノピラゾール
JP2020103499A Pending JP2020158522A (ja) 2013-03-15 2020-06-16 トロンビン阻害剤としてのハロゲノピラゾール

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JP2019019308A Pending JP2019081782A (ja) 2013-03-15 2019-02-06 トロンビン阻害剤としてのハロゲノピラゾール
JP2020103499A Pending JP2020158522A (ja) 2013-03-15 2020-06-16 トロンビン阻害剤としてのハロゲノピラゾール

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US (2) US9951025B2 (enExample)
EP (1) EP2970141B1 (enExample)
JP (3) JP6479749B2 (enExample)
KR (1) KR20150130405A (enExample)
CN (2) CN105209440B (enExample)
AU (2) AU2014238478B2 (enExample)
BR (1) BR112015023214A8 (enExample)
CA (1) CA2902431A1 (enExample)
ES (1) ES2791749T3 (enExample)
HK (1) HK1214252A1 (enExample)
IL (1) IL240763B (enExample)
MX (1) MX373646B (enExample)
RU (1) RU2015144193A (enExample)
SG (2) SG11201506757TA (enExample)
WO (2) WO2014149139A2 (enExample)
ZA (1) ZA201506440B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2970141B1 (en) 2013-03-15 2020-02-26 Verseon Corporation Halogenopyrazoles as inhibitors of thrombin
ES2853483T3 (es) 2013-03-15 2021-09-16 Verseon Int Corporation Compuestos aromáticos multisustituidos como inhibidores de la serina proteasa
US10532995B2 (en) * 2015-02-27 2020-01-14 Verseon Corporation Substituted pyrazole compounds as serine protease inhibitors
JP2022526827A (ja) 2019-04-11 2022-05-26 アンジオン バイオメディカ コーポレーション （ｅ）－３－［２－（２－チエニル）ビニル］－１ｈ－ピラゾールの固体形態
CN112062692A (zh) * 2019-06-11 2020-12-11 太仓市茜泾化工有限公司 一种乙氧甲叉氰基乙酸乙酯的制备方法
CN112986065B (zh) * 2021-02-08 2021-08-31 杭州同创医学检验实验室有限公司 一种用于血细胞分析仪的全血质控品及其制备方法

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