JP2015163632A5 - - Google Patents
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- JP2015163632A5 JP2015163632A5 JP2015096257A JP2015096257A JP2015163632A5 JP 2015163632 A5 JP2015163632 A5 JP 2015163632A5 JP 2015096257 A JP2015096257 A JP 2015096257A JP 2015096257 A JP2015096257 A JP 2015096257A JP 2015163632 A5 JP2015163632 A5 JP 2015163632A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- alkyl
- heteroaryl
- alkylene
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 14
- 125000000623 heterocyclic group Chemical group 0.000 claims 13
- 229910052757 nitrogen Inorganic materials 0.000 claims 10
- 125000006573 (C1-C10) heteroaryl group Chemical group 0.000 claims 8
- -1 —N (R a ) (R b ) Chemical class 0.000 claims 8
- 125000006376 (C3-C10) cycloalkyl group Chemical group 0.000 claims 6
- 229910052739 hydrogen Inorganic materials 0.000 claims 6
- 150000002431 hydrogen Chemical class 0.000 claims 6
- 239000001257 hydrogen Substances 0.000 claims 6
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 5
- 125000000041 C6-C10 aryl group Chemical group 0.000 claims 5
- YZCKVEUIGOORGS-OUBTZVSYSA-N Deuterium Chemical compound [2H] YZCKVEUIGOORGS-OUBTZVSYSA-N 0.000 claims 5
- 125000002993 cycloalkylene group Chemical group 0.000 claims 5
- 229910052805 deuterium Inorganic materials 0.000 claims 5
- 150000001875 compounds Chemical class 0.000 claims 4
- 125000005724 cycloalkenylene group Chemical group 0.000 claims 4
- 229910052736 halogen Inorganic materials 0.000 claims 4
- 150000002367 halogens Chemical class 0.000 claims 4
- 125000006585 (C6-C10) arylene group Chemical group 0.000 claims 3
- 125000000753 cycloalkyl group Chemical group 0.000 claims 3
- 125000005549 heteroarylene group Chemical group 0.000 claims 3
- 125000000008 (C1-C10) alkyl group Chemical group 0.000 claims 2
- 125000003161 (C1-C6) alkylene group Chemical group 0.000 claims 2
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 claims 2
- 125000006590 (C2-C6) alkenylene group Chemical group 0.000 claims 2
- 125000006591 (C2-C6) alkynylene group Chemical group 0.000 claims 2
- 125000006586 (C3-C10) cycloalkylene group Chemical group 0.000 claims 2
- 125000006553 (C3-C8) cycloalkenyl group Chemical group 0.000 claims 2
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 2
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 2
- 125000002947 alkylene group Chemical group 0.000 claims 2
- 229910052799 carbon Inorganic materials 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 2
- 125000006832 (C1-C10) alkylene group Chemical group 0.000 claims 1
- 125000006694 (C2-C10) heterocyclyl group Chemical group 0.000 claims 1
- 125000006374 C2-C10 alkenyl group Chemical group 0.000 claims 1
- 125000004450 alkenylene group Chemical group 0.000 claims 1
- 125000000304 alkynyl group Chemical group 0.000 claims 1
- 125000004419 alkynylene group Chemical group 0.000 claims 1
- 230000000975 bioactive effect Effects 0.000 claims 1
- 239000002207 metabolite Substances 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 125000004430 oxygen atom Chemical group O* 0.000 claims 1
- 229940002612 prodrug Drugs 0.000 claims 1
- 239000000651 prodrug Substances 0.000 claims 1
- 125000003226 pyrazolyl group Chemical group 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 229910052717 sulfur Inorganic materials 0.000 claims 1
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13160208P | 2008-06-10 | 2008-06-10 | |
| US13159908P | 2008-06-10 | 2008-06-10 | |
| US61/131,599 | 2008-06-10 | ||
| US61/131,602 | 2008-06-10 | ||
| US61/190,159 | 2008-08-25 | ||
| US19015908P | 2008-08-26 | 2008-08-26 | |
| US20106408P | 2008-12-05 | 2008-12-05 | |
| US61/201,064 | 2008-12-05 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011513627A Division JP5748659B2 (ja) | 2008-06-10 | 2009-06-09 | 新規な三環式化合物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2015163632A JP2015163632A (ja) | 2015-09-10 |
| JP2015163632A5 true JP2015163632A5 (cg-RX-API-DMAC7.html) | 2016-02-18 |
Family
ID=41415363
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011513627A Active JP5748659B2 (ja) | 2008-06-10 | 2009-06-09 | 新規な三環式化合物 |
| JP2015096257A Pending JP2015163632A (ja) | 2008-06-10 | 2015-05-11 | 新規な三環式化合物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011513627A Active JP5748659B2 (ja) | 2008-06-10 | 2009-06-09 | 新規な三環式化合物 |
Country Status (36)
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