JP2014509859A5 - - Google Patents

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JP2014509859A5
JP2014509859A5 JP2013558223A JP2013558223A JP2014509859A5 JP 2014509859 A5 JP2014509859 A5 JP 2014509859A5 JP 2013558223 A JP2013558223 A JP 2013558223A JP 2013558223 A JP2013558223 A JP 2013558223A JP 2014509859 A5 JP2014509859 A5 JP 2014509859A5
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JP
Japan
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methyl
arginine
nal
histidine
phenylalanine
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Pending
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JP2013558223A
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Japanese (ja)
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JP2014509859A (ja
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Priority claimed from PCT/US2012/029537 external-priority patent/WO2012125973A2/en
Publication of JP2014509859A publication Critical patent/JP2014509859A/ja
Publication of JP2014509859A5 publication Critical patent/JP2014509859A5/ja
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JP2013558223A 2011-03-16 2012-03-16 17nav1.3およびnav1.7の強力かつ選択的阻害剤 Pending JP2014509859A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161453492P 2011-03-16 2011-03-16
US61/453,492 2011-03-16
US201261608088P 2012-03-07 2012-03-07
US61/608,088 2012-03-07
PCT/US2012/029537 WO2012125973A2 (en) 2011-03-16 2012-03-16 Potent and selective inhibitors of nav1.3 and nav1.7

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016161682A Division JP2017031157A (ja) 2011-03-16 2016-08-22 17nav1.3およびnav1.7の強力かつ選択的阻害剤

Publications (2)

Publication Number Publication Date
JP2014509859A JP2014509859A (ja) 2014-04-24
JP2014509859A5 true JP2014509859A5 (enExample) 2015-04-30

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Family Applications (2)

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JP2013558223A Pending JP2014509859A (ja) 2011-03-16 2012-03-16 17nav1.3およびnav1.7の強力かつ選択的阻害剤
JP2016161682A Pending JP2017031157A (ja) 2011-03-16 2016-08-22 17nav1.3およびnav1.7の強力かつ選択的阻害剤

Family Applications After (1)

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JP2016161682A Pending JP2017031157A (ja) 2011-03-16 2016-08-22 17nav1.3およびnav1.7の強力かつ選択的阻害剤

Country Status (24)

Country Link
US (2) US9340590B2 (enExample)
EP (1) EP2686340A2 (enExample)
JP (2) JP2014509859A (enExample)
KR (1) KR20140145947A (enExample)
CN (1) CN103930437A (enExample)
AP (1) AP2013007173A0 (enExample)
AR (1) AR088413A1 (enExample)
AU (1) AU2012228990B2 (enExample)
BR (1) BR112013023674A2 (enExample)
CA (1) CA2830065A1 (enExample)
CL (1) CL2013002673A1 (enExample)
CO (1) CO6821886A2 (enExample)
CR (1) CR20130533A (enExample)
EA (1) EA201391331A1 (enExample)
HK (1) HK1198173A1 (enExample)
MA (1) MA35385B1 (enExample)
MX (1) MX2013010497A (enExample)
PE (1) PE20140593A1 (enExample)
PH (1) PH12013501865A1 (enExample)
SG (2) SG10201601789TA (enExample)
TW (1) TW201300407A (enExample)
UY (1) UY33959A (enExample)
WO (1) WO2012125973A2 (enExample)
ZA (1) ZA201306920B (enExample)

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CN120603815A (zh) 2022-12-06 2025-09-05 沃泰克斯药物股份有限公司 钠通道的取代四氢呋喃调节剂的合成方法
WO2025090480A1 (en) 2023-10-23 2025-05-01 Vertex Pharmaceuticals Incorporated Heteroaryl compounds for the treatment of pain
TW202523313A (zh) 2023-10-23 2025-06-16 美商維泰克斯製藥公司 用於治療疼痛之雜芳基化合物
TW202535867A (zh) 2023-10-23 2025-09-16 美商維泰克斯製藥公司 用於治療疼痛之鈉通道調節劑及其固體形式的製備方法
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