JP2013544786A5 - - Google Patents
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- Publication number
- JP2013544786A5 JP2013544786A5 JP2013533941A JP2013533941A JP2013544786A5 JP 2013544786 A5 JP2013544786 A5 JP 2013544786A5 JP 2013533941 A JP2013533941 A JP 2013533941A JP 2013533941 A JP2013533941 A JP 2013533941A JP 2013544786 A5 JP2013544786 A5 JP 2013544786A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- chch
- isobutyl
- alkyl
- propylthio
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39245110P | 2010-10-12 | 2010-10-12 | |
| US61/392,451 | 2010-10-12 | ||
| PCT/US2011/055788 WO2012051193A1 (en) | 2010-10-12 | 2011-10-11 | Cyclosporin analogs |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013544786A JP2013544786A (ja) | 2013-12-19 |
| JP2013544786A5 true JP2013544786A5 (enExample) | 2014-02-06 |
| JP5805773B2 JP5805773B2 (ja) | 2015-11-10 |
Family
ID=44883796
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013533941A Expired - Fee Related JP5805773B2 (ja) | 2010-10-12 | 2011-10-11 | シクロスポリンアナログ |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US9175042B2 (enExample) |
| EP (1) | EP2627663B1 (enExample) |
| JP (1) | JP5805773B2 (enExample) |
| KR (1) | KR20140026328A (enExample) |
| CN (1) | CN103261212A (enExample) |
| AU (1) | AU2011316689B2 (enExample) |
| BR (1) | BR112013008749A2 (enExample) |
| CA (1) | CA2814191A1 (enExample) |
| IL (1) | IL225616A0 (enExample) |
| MX (1) | MX2013004062A (enExample) |
| RU (1) | RU2013120927A (enExample) |
| WO (1) | WO2012051193A1 (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010138422A1 (en) * | 2009-05-27 | 2010-12-02 | Allergan, Inc. | Cyclosporin derivatives for enhancing the growth of hair |
| JP6144627B2 (ja) * | 2010-12-15 | 2017-06-07 | コントラヴィア ファーマシューティカルズ、インク． | アミノ酸１および３で修飾されたシクロスポリン類似体分子 |
| EP2855508B1 (en) | 2012-06-01 | 2018-02-14 | Allergan, Inc. | Cyclosporin a analogs |
| CN105025929A (zh) | 2013-03-08 | 2015-11-04 | 阿勒根公司 | 环孢菌素a-类固醇缀合物 |
| WO2016112321A1 (en) | 2015-01-08 | 2016-07-14 | Allergan, Inc. | Cyclosporin derivatives wherein the mebmt sidechain has been cyclized |
| EP3551034A1 (en) | 2016-12-07 | 2019-10-16 | Progenity, Inc. | Gastrointestinal tract detection methods, devices and systems |
| WO2018112255A1 (en) | 2016-12-14 | 2018-06-21 | Progenity Inc. | Treatment of a disease of the gastrointestinal tract with an immunosuppressant |
| WO2019246312A1 (en) | 2018-06-20 | 2019-12-26 | Progenity, Inc. | Treatment of a disease of the gastrointestinal tract with an immunomodulator |
| CN115028681B (zh) * | 2022-08-11 | 2022-11-15 | 中国科学院微生物研究所 | 一种降解亲环素a的嵌合体化合物及其制备方法与应用 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4649047A (en) | 1985-03-19 | 1987-03-10 | University Of Georgia Research Foundation, Inc. | Ophthalmic treatment by topical administration of cyclosporin |
| US5474979A (en) | 1994-05-17 | 1995-12-12 | Allergan, Inc. | Nonirritating emulsions for sensitive tissue |
| FR2757521B1 (fr) * | 1996-12-24 | 1999-01-29 | Rhone Poulenc Rorer Sa | Nouveaux derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR2757522B1 (fr) * | 1996-12-24 | 1999-01-29 | Rhone Poulenc Rorer Sa | Derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR2762843B1 (fr) | 1997-04-30 | 1999-12-10 | Rhone Poulenc Rorer Sa | Nouveaux derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR2772768B1 (fr) * | 1997-12-19 | 2000-01-14 | Rhone Poulenc Rorer Sa | Nouveau procede de preparation de derives de cyclosporine |
| ES2212583T3 (es) | 1998-06-12 | 2004-07-16 | C-Chem Ag | Nuevas ciclosporinas. |
| US6254860B1 (en) * | 1999-04-13 | 2001-07-03 | Allergan Sales, Inc. | Ocular treatment using cyclosporin-A derivatives |
| CN100478025C (zh) * | 2005-03-25 | 2009-04-15 | 中国科学院上海药物研究所 | 一种环孢菌素a眼用微乳制剂及其制备方法 |
| ATE502633T1 (de) * | 2006-05-19 | 2011-04-15 | Scynexis Inc | Cyclosporins zur behandlung und vorbeugung von augenerkrankungen |
| CA2686234A1 (en) | 2007-05-04 | 2008-11-13 | Allergan, Inc. | Use of cyclosporines in the treatment of patients with intraocular lenses |
| AU2009268549B2 (en) | 2008-07-10 | 2015-07-16 | Allergan, Inc. | Cyclosporin derivatives for treating ocular and dermal diseases and conditions |
| WO2012009715A2 (en) * | 2010-07-16 | 2012-01-19 | S&T Global Inc. | Novel cyclosporin derivatives for the treatment and prevention of a viral infection |
| WO2012021796A2 (en) | 2010-08-12 | 2012-02-16 | S&T Global, Inc. | Novel cyclosporin derivatives for the treatment and prevention of a viral infection |
| RU2013119869A (ru) | 2010-10-12 | 2014-11-20 | Аллерган, Инк. | Аналоги циклоспорина |
| JP6093307B2 (ja) * | 2010-12-03 | 2017-03-08 | エス アンド ティー グローバル インク． | ウイルス感染の治療および予防のための新規シクロスポリン誘導体 |
| US9890198B2 (en) | 2010-12-03 | 2018-02-13 | S&T Global Inc. | Cyclosporin derivatives and uses thereof |
-
2011
- 2011-10-11 US US13/270,929 patent/US9175042B2/en active Active
- 2011-10-11 CN CN201180059696XA patent/CN103261212A/zh active Pending
- 2011-10-11 EP EP11770984.0A patent/EP2627663B1/en not_active Not-in-force
- 2011-10-11 CA CA2814191A patent/CA2814191A1/en not_active Abandoned
- 2011-10-11 AU AU2011316689A patent/AU2011316689B2/en not_active Ceased
- 2011-10-11 KR KR1020137012144A patent/KR20140026328A/ko not_active Withdrawn
- 2011-10-11 BR BR112013008749A patent/BR112013008749A2/pt not_active IP Right Cessation
- 2011-10-11 MX MX2013004062A patent/MX2013004062A/es unknown
- 2011-10-11 JP JP2013533941A patent/JP5805773B2/ja not_active Expired - Fee Related
- 2011-10-11 WO PCT/US2011/055788 patent/WO2012051193A1/en not_active Ceased
- 2011-10-11 RU RU2013120927/04A patent/RU2013120927A/ru not_active Application Discontinuation
-
2013
- 2013-04-07 IL IL225616A patent/IL225616A0/en unknown
-
2015
- 2015-10-02 US US14/873,908 patent/US9561259B2/en not_active Expired - Fee Related
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