JP2013530957A5 - - Google Patents

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JP2013530957A5
JP2013530957A5 JP2013513348A JP2013513348A JP2013530957A5 JP 2013530957 A5 JP2013530957 A5 JP 2013530957A5 JP 2013513348 A JP2013513348 A JP 2013513348A JP 2013513348 A JP2013513348 A JP 2013513348A JP 2013530957 A5 JP2013530957 A5 JP 2013530957A5
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JP
Japan
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methyl
piperazin
benzamide
cyclohexyl
difluoro
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JP2013513348A
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Japanese (ja)
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JP5813101B2 (ja
JP2013530957A (ja
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Priority claimed from PCT/US2011/038939 external-priority patent/WO2011153359A1/en
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Publication of JP2013530957A5 publication Critical patent/JP2013530957A5/ja
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Publication of JP5813101B2 publication Critical patent/JP5813101B2/ja
Expired - Fee Related legal-status Critical Current
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JP2013513348A 2010-06-04 2011-06-02 グリシントランスポーター−1阻害剤、その作製方法および使用方法 Expired - Fee Related JP5813101B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35166210P 2010-06-04 2010-06-04
US61/351,662 2010-06-04
PCT/US2011/038939 WO2011153359A1 (en) 2010-06-04 2011-06-02 Glycine transporter-1 inhibitors, methods of making them, and uses thereof

Publications (3)

Publication Number Publication Date
JP2013530957A JP2013530957A (ja) 2013-08-01
JP2013530957A5 true JP2013530957A5 (enExample) 2014-07-10
JP5813101B2 JP5813101B2 (ja) 2015-11-17

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JP2013513348A Expired - Fee Related JP5813101B2 (ja) 2010-06-04 2011-06-02 グリシントランスポーター−1阻害剤、その作製方法および使用方法

Country Status (10)

Country Link
US (1) US9045445B2 (enExample)
EP (1) EP2575815A4 (enExample)
JP (1) JP5813101B2 (enExample)
KR (1) KR20130087002A (enExample)
CN (1) CN103096893B (enExample)
AU (1) AU2011261375B2 (enExample)
CA (1) CA2801074A1 (enExample)
NZ (1) NZ604035A (enExample)
SG (1) SG186885A1 (enExample)
WO (1) WO2011153359A1 (enExample)

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CA2821975A1 (en) 2010-12-17 2012-06-21 Shunqi Yan N-(4-(azetidine-1-carbonyl)phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase m2 pkm2 modulators
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