JP2011528020A5 - - Google Patents

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Publication number
JP2011528020A5
JP2011528020A5 JP2011517911A JP2011517911A JP2011528020A5 JP 2011528020 A5 JP2011528020 A5 JP 2011528020A5 JP 2011517911 A JP2011517911 A JP 2011517911A JP 2011517911 A JP2011517911 A JP 2011517911A JP 2011528020 A5 JP2011528020 A5 JP 2011528020A5
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JP
Japan
Prior art keywords
pain
methyl
compound
compound according
pyridinyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2011517911A
Other languages
English (en)
Japanese (ja)
Other versions
JP2011528020A (ja
JP5543966B2 (ja
Filing date
Publication date
Priority claimed from GBGB0813142.7A external-priority patent/GB0813142D0/en
Application filed filed Critical
Publication of JP2011528020A publication Critical patent/JP2011528020A/ja
Publication of JP2011528020A5 publication Critical patent/JP2011528020A5/ja
Application granted granted Critical
Publication of JP5543966B2 publication Critical patent/JP5543966B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2011517911A 2008-07-17 2009-07-15 Cav2.2カルシウムチャネルモジュレーターとして使用されるピペラジン誘導体 Expired - Fee Related JP5543966B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0813142.7 2008-07-17
GBGB0813142.7A GB0813142D0 (en) 2008-07-17 2008-07-17 Novel compounds
PCT/EP2009/059012 WO2010007073A1 (en) 2008-07-17 2009-07-15 Piperazine derivatives used as cav2.2 calcium channel modulators

Publications (3)

Publication Number Publication Date
JP2011528020A JP2011528020A (ja) 2011-11-10
JP2011528020A5 true JP2011528020A5 (enExample) 2012-08-30
JP5543966B2 JP5543966B2 (ja) 2014-07-09

Family

ID=39737239

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2011517910A Expired - Fee Related JP5688850B2 (ja) 2008-07-17 2009-07-15 Cav2.2カルシウムチャネルモジュレーターとして使用されるピペラジン誘導体
JP2011517911A Expired - Fee Related JP5543966B2 (ja) 2008-07-17 2009-07-15 Cav2.2カルシウムチャネルモジュレーターとして使用されるピペラジン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2011517910A Expired - Fee Related JP5688850B2 (ja) 2008-07-17 2009-07-15 Cav2.2カルシウムチャネルモジュレーターとして使用されるピペラジン誘導体

Country Status (19)

Country Link
US (3) US8288388B2 (enExample)
EP (2) EP2300432B1 (enExample)
JP (2) JP5688850B2 (enExample)
KR (1) KR101599087B1 (enExample)
CN (1) CN102099337B (enExample)
AR (1) AR072809A1 (enExample)
AU (1) AU2009272762B2 (enExample)
BR (1) BRPI0916622A2 (enExample)
CA (1) CA2730471C (enExample)
EA (1) EA018621B1 (enExample)
ES (2) ES2396962T3 (enExample)
GB (1) GB0813142D0 (enExample)
IL (1) IL210446A (enExample)
MX (1) MX2011000600A (enExample)
PL (1) PL2300432T3 (enExample)
TW (1) TW201016677A (enExample)
UY (1) UY31990A (enExample)
WO (2) WO2010007073A1 (enExample)
ZA (1) ZA201100014B (enExample)

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GB0813142D0 (en) * 2008-07-17 2008-08-27 Glaxo Group Ltd Novel compounds
GB201000685D0 (en) * 2010-01-15 2010-03-03 Glaxo Group Ltd Novel compounds
JP6058556B2 (ja) * 2011-01-19 2017-01-11 クオンベルゲンセ プハルマセウトイカルス リミテッド CaV2.2カルシウムチャンネルブロッカーとしてのピペラジン誘導体
EA022973B1 (ru) 2011-06-27 2016-03-31 Ньюрон Фармасьютикалс С.П.А. Фторированные арилалкиламинокарбоксамидные производные
CN106458955B (zh) * 2014-04-14 2019-07-19 格吕伦塔尔有限公司 芳基取代的杂环基砜
AR100073A1 (es) * 2014-04-14 2016-09-07 Gruenenthal Gmbh Sulfonas heterocíclicas sustituidas con heteroarilos
GB201516183D0 (en) * 2015-09-14 2015-10-28 Calchan Ltd Novel pharmaceutical composition
TW201718557A (zh) 2015-10-08 2017-06-01 歌林達有限公司 經吡唑基取代之四氫吡喃基碸
TW201726128A (zh) 2015-10-08 2017-08-01 歌林達有限公司 經吡唑基取代之四氫哌喃基碸
KR102654466B1 (ko) * 2017-04-26 2024-04-08 카비온, 인코포레이티드 기억 및 인지 개선 방법 및 기억 및 인지 장애 치료 방법
CN118085389B (zh) * 2024-03-11 2024-11-05 伟建实业(苏州)有限公司 一种环保型抗菌海绵及其制备方法

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