JP2012505891A5 - - Google Patents

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Publication number
JP2012505891A5
JP2012505891A5 JP2011532175A JP2011532175A JP2012505891A5 JP 2012505891 A5 JP2012505891 A5 JP 2012505891A5 JP 2011532175 A JP2011532175 A JP 2011532175A JP 2011532175 A JP2011532175 A JP 2011532175A JP 2012505891 A5 JP2012505891 A5 JP 2012505891A5
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JP
Japan
Prior art keywords
alkyl
alkoxy
halogen
pyridinyl
alkoxycarbonyl
Prior art date
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JP2011532175A
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English (en)
Japanese (ja)
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JP2012505891A (ja
JP5529876B2 (ja
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Priority claimed from PCT/US2009/060436 external-priority patent/WO2010045188A1/en
Publication of JP2012505891A publication Critical patent/JP2012505891A/ja
Publication of JP2012505891A5 publication Critical patent/JP2012505891A5/ja
Application granted granted Critical
Publication of JP5529876B2 publication Critical patent/JP5529876B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011532175A 2008-10-17 2009-10-13 Ｍｍｐ−１３阻害剤として有用なヘテロアリール置換インドール化合物 Expired - Fee Related JP5529876B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10620708P 2008-10-17 2008-10-17
US61/106,207 2008-10-17
PCT/US2009/060436 WO2010045188A1 (en) 2008-10-17 2009-10-13 Heteroaryl substituted indole compounds useful as mmp-13 inhibitors

Publications (3)

Publication Number Publication Date
JP2012505891A JP2012505891A (ja) 2012-03-08
JP2012505891A5 true JP2012505891A5 (enExample) 2012-11-29
JP5529876B2 JP5529876B2 (ja) 2014-06-25

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ID=41508906

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011532175A Expired - Fee Related JP5529876B2 (ja) 2008-10-17 2009-10-13 Ｍｍｐ−１３阻害剤として有用なヘテロアリール置換インドール化合物

Country Status (5)

Country Link
US (1) US8785489B2 (enExample)
EP (1) EP2340243B1 (enExample)
JP (1) JP5529876B2 (enExample)
CA (1) CA2738929A1 (enExample)
WO (1) WO2010045188A1 (enExample)

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US8785489B2 (en) 2008-10-17 2014-07-22 Boehringer Ingelheim International Gmbh Heteroaryl substituted indole compounds useful as MMP-13 inhibitors
CA2743146A1 (en) 2008-11-17 2010-05-20 Boehringer Ingelheim International Gmbh Heteroaryl diamide compounds useful as mmp-13 inhibitors

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