JP2011518836A - 大環状化合物およびそれらのキナーゼ阻害剤としての使用 - Google Patents
大環状化合物およびそれらのキナーゼ阻害剤としての使用 Download PDFInfo
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- JP2011518836A JP2011518836A JP2011506453A JP2011506453A JP2011518836A JP 2011518836 A JP2011518836 A JP 2011518836A JP 2011506453 A JP2011506453 A JP 2011506453A JP 2011506453 A JP2011506453 A JP 2011506453A JP 2011518836 A JP2011518836 A JP 2011518836A
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- Prior art keywords
- chloro
- docosa
- nonaen
- tetraazatetracyclo
- pentaazatetracyclo
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| PCT/US2009/041555 WO2009132202A2 (en) | 2008-04-24 | 2009-04-23 | Macrocyclic compounds and their use as kinase inhibitors |
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| JP2016041709A (ja) * | 2012-03-06 | 2016-03-31 | ファイザー・インク | 増殖性疾患の治療のための大環状誘導体 |
| JP2016540824A (ja) * | 2013-12-20 | 2016-12-28 | インスティテュート オブ ファーマコロジー アンド トキシコロジー アカデミー オブ ミリタリー メディカル サイエンシズ ピー．エル．エー．チャイナ | 新規ピペリジンカルボキサミド化合物、その調製方法及び使用 |
| JP2023513793A (ja) * | 2020-02-14 | 2023-04-03 | ソーク インスティテュート フォー バイオロジカル スタディーズ | 大環状ｕｌｋ１／２阻害剤 |
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| JP2016041709A (ja) * | 2012-03-06 | 2016-03-31 | ファイザー・インク | 増殖性疾患の治療のための大環状誘導体 |
| JP2016505069A (ja) * | 2013-01-25 | 2016-02-18 | ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ | Ｃ型肝炎の治療用のアンモニウム誘導体 |
| JP2016540824A (ja) * | 2013-12-20 | 2016-12-28 | インスティテュート オブ ファーマコロジー アンド トキシコロジー アカデミー オブ ミリタリー メディカル サイエンシズ ピー．エル．エー．チャイナ | 新規ピペリジンカルボキサミド化合物、その調製方法及び使用 |
| JP2023513793A (ja) * | 2020-02-14 | 2023-04-03 | ソーク インスティテュート フォー バイオロジカル スタディーズ | 大環状ｕｌｋ１／２阻害剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009132202A3 (en) | 2010-11-25 |
| US8871753B2 (en) | 2014-10-28 |
| CA2722326A1 (en) | 2009-10-29 |
| WO2009132202A2 (en) | 2009-10-29 |
| EP2274288A2 (en) | 2011-01-19 |
| US20090286778A1 (en) | 2009-11-19 |
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