JP2010540426A5 - - Google Patents

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JP2010540426A5
JP2010540426A5 JP2010525442A JP2010525442A JP2010540426A5 JP 2010540426 A5 JP2010540426 A5 JP 2010540426A5 JP 2010525442 A JP2010525442 A JP 2010525442A JP 2010525442 A JP2010525442 A JP 2010525442A JP 2010540426 A5 JP2010540426 A5 JP 2010540426A5
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formula
compound
under conditions
conditions suitable
reacting
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JP2010525442A
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JP2010540426A (ja
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Priority claimed from PCT/GB2008/003226 external-priority patent/WO2009040517A2/en
Publication of JP2010540426A publication Critical patent/JP2010540426A/ja
Publication of JP2010540426A5 publication Critical patent/JP2010540426A5/ja
Pending legal-status Critical Current

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JP2010525442A 2007-09-25 2008-09-23 特定のヒドロキサム酸化合物の合成方法 Pending JP2010540426A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US97488007P 2007-09-25 2007-09-25
PCT/GB2008/003226 WO2009040517A2 (en) 2007-09-25 2008-09-23 Methods of synthesis of certain hydroxamic acid compounds

Publications (2)

Publication Number Publication Date
JP2010540426A JP2010540426A (ja) 2010-12-24
JP2010540426A5 true JP2010540426A5 (https=) 2011-11-10

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JP2010525442A Pending JP2010540426A (ja) 2007-09-25 2008-09-23 特定のヒドロキサム酸化合物の合成方法

Country Status (7)

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US (1) US8642809B2 (https=)
EP (1) EP2203421B1 (https=)
JP (1) JP2010540426A (https=)
CN (1) CN101868446A (https=)
CA (1) CA2700173C (https=)
MX (1) MX2010003230A (https=)
WO (1) WO2009040517A2 (https=)

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RU2748835C1 (ru) 2017-11-27 2021-05-31 Совет Научных И Прикладных Исследований Индол(сульфонил)-n-гидроксибензамидные производные в качестве селективных ингибиторов hdac
CN108033902B (zh) * 2017-12-26 2020-07-07 深圳万乐药业有限公司 一种高纯度贝利司他顺式异构体的制备方法
CN109265377B (zh) * 2018-10-25 2021-01-22 瑞阳制药股份有限公司 贝利司他的绿色合成方法
CN109336788A (zh) * 2018-10-31 2019-02-15 安徽省庆云医药股份有限公司 一种贝利司他的制备方法
CN111848591B (zh) * 2019-04-25 2022-03-18 成都先导药物开发股份有限公司 Hdac抑制剂及其制备方法和用途
CN115636774B (zh) * 2022-12-01 2023-12-22 南开大学 一种贝利司他的合成方法
CN119456224B (zh) * 2024-10-31 2025-11-28 郑州大学 一种矿物的预处理方法协同浮选药剂的分离工艺

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