JP2010507641A5 - - Google Patents

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Publication number
JP2010507641A5
JP2010507641A5 JP2009533939A JP2009533939A JP2010507641A5 JP 2010507641 A5 JP2010507641 A5 JP 2010507641A5 JP 2009533939 A JP2009533939 A JP 2009533939A JP 2009533939 A JP2009533939 A JP 2009533939A JP 2010507641 A5 JP2010507641 A5 JP 2010507641A5
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JP
Japan
Prior art keywords
methylpyrazin
difluoromethoxy
propan
pyrazine
oxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009533939A
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English (en)
Japanese (ja)
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JP4673429B2 (ja
JP2010507641A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/GB2007/004057 external-priority patent/WO2008050117A1/en
Publication of JP2010507641A publication Critical patent/JP2010507641A/ja
Publication of JP2010507641A5 publication Critical patent/JP2010507641A5/ja
Application granted granted Critical
Publication of JP4673429B2 publication Critical patent/JP4673429B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009533939A 2006-10-26 2007-10-25 グルコキナーゼ（ｇｌｋ）活性化剤としてのベンゾイルアミノヘテロシクリル化合物 Expired - Fee Related JP4673429B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US86305606P 2006-10-26 2006-10-26
US95737007P 2007-08-22 2007-08-22
PCT/GB2007/004057 WO2008050117A1 (en) 2006-10-26 2007-10-25 Benzoyl amino heterocyclyl compounds as glucokinase (glk) activators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010228109A Division JP2011046724A (ja) 2006-10-26 2010-10-08 グルコキナーゼ（ｇｌｋ）活性化剤としてのベンゾイルアミノヘテロシクリル化合物

Publications (3)

Publication Number Publication Date
JP2010507641A JP2010507641A (ja) 2010-03-11
JP2010507641A5 true JP2010507641A5 (enExample) 2010-11-25
JP4673429B2 JP4673429B2 (ja) 2011-04-20

Family

ID=38925536

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009533939A Expired - Fee Related JP4673429B2 (ja) 2006-10-26 2007-10-25 グルコキナーゼ（ｇｌｋ）活性化剤としてのベンゾイルアミノヘテロシクリル化合物
JP2010228109A Withdrawn JP2011046724A (ja) 2006-10-26 2010-10-08 グルコキナーゼ（ｇｌｋ）活性化剤としてのベンゾイルアミノヘテロシクリル化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010228109A Withdrawn JP2011046724A (ja) 2006-10-26 2010-10-08 グルコキナーゼ（ｇｌｋ）活性化剤としてのベンゾイルアミノヘテロシクリル化合物

Country Status (20)

Country Link
US (2) US7671060B2 (enExample)
EP (2) EP2272834A1 (enExample)
JP (2) JP4673429B2 (enExample)
KR (1) KR20090084880A (enExample)
CN (1) CN101805299A (enExample)
AR (1) AR063393A1 (enExample)
AU (1) AU2007310624B2 (enExample)
BR (1) BRPI0718155A2 (enExample)
CA (1) CA2667316A1 (enExample)
CL (1) CL2007003061A1 (enExample)
CO (1) CO6160314A2 (enExample)
IL (1) IL198143A0 (enExample)
MX (1) MX2009004467A (enExample)
NO (1) NO20091596L (enExample)
PE (1) PE20080927A1 (enExample)
RU (1) RU2440992C2 (enExample)
SA (1) SA07280576B1 (enExample)
TW (1) TW200825060A (enExample)
UY (1) UY30659A1 (enExample)
WO (1) WO2008050117A1 (enExample)

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GB0902406D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Crystalline polymorphic form
GB0902434D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
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TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
GB201714777D0 (en) 2017-09-14 2017-11-01 Univ London Queen Mary Agent
CN110128352A (zh) 2018-02-02 2019-08-16 青岛清原化合物有限公司 哒嗪醇类化合物及其衍生物、制备方法、除草组合物和应用

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TW200600086A (en) * 2004-06-05 2006-01-01 Astrazeneca Ab Chemical compound
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WO2010116177A1 (en) 2009-04-09 2010-10-14 Astrazeneca Ab A pyrazolo [4,5-e] pyrimidine derivative and its use to treat diabetes and obesity
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