CL2007003061A1 - Compuestos derivados de 3,5-dioxi-benzamida; proceso de preparacion; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar una enfermedad mediada a traves de glk, tal como la diabetes tipo 2. - Google Patents
Compuestos derivados de 3,5-dioxi-benzamida; proceso de preparacion; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar una enfermedad mediada a traves de glk, tal como la diabetes tipo 2.Info
- Publication number
- CL2007003061A1 CL2007003061A1 CL200703061A CL2007003061A CL2007003061A1 CL 2007003061 A1 CL2007003061 A1 CL 2007003061A1 CL 200703061 A CL200703061 A CL 200703061A CL 2007003061 A CL2007003061 A CL 2007003061A CL 2007003061 A1 CL2007003061 A1 CL 2007003061A1
- Authority
- CL
- Chile
- Prior art keywords
- compounds
- benzamida
- dioxi
- glk
- diabetes
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US86305606P | 2006-10-26 | 2006-10-26 | |
US95737007P | 2007-08-22 | 2007-08-22 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2007003061A1 true CL2007003061A1 (es) | 2008-08-01 |
Family
ID=38925536
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL200703061A CL2007003061A1 (es) | 2006-10-26 | 2007-10-24 | Compuestos derivados de 3,5-dioxi-benzamida; proceso de preparacion; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar una enfermedad mediada a traves de glk, tal como la diabetes tipo 2. |
Country Status (20)
Country | Link |
---|---|
US (2) | US7671060B2 (es) |
EP (2) | EP2272834A1 (es) |
JP (2) | JP4673429B2 (es) |
KR (1) | KR20090084880A (es) |
CN (1) | CN101805299A (es) |
AR (1) | AR063393A1 (es) |
AU (1) | AU2007310624B2 (es) |
BR (1) | BRPI0718155A2 (es) |
CA (1) | CA2667316A1 (es) |
CL (1) | CL2007003061A1 (es) |
CO (1) | CO6160314A2 (es) |
IL (1) | IL198143A0 (es) |
MX (1) | MX2009004467A (es) |
NO (1) | NO20091596L (es) |
PE (1) | PE20080927A1 (es) |
RU (1) | RU2440992C2 (es) |
SA (1) | SA07280576B1 (es) |
TW (1) | TW200825060A (es) |
UY (1) | UY30659A1 (es) |
WO (1) | WO2008050117A1 (es) |
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TW200600086A (en) * | 2004-06-05 | 2006-01-01 | Astrazeneca Ab | Chemical compound |
TW200714597A (en) * | 2005-05-27 | 2007-04-16 | Astrazeneca Ab | Chemical compounds |
EP2305674A1 (en) * | 2005-07-09 | 2011-04-06 | AstraZeneca AB | Heteroaryl benzamide derivatives for use as GLK activators in the treatment of diabetes |
TW200825060A (en) * | 2006-10-26 | 2008-06-16 | Astrazeneca Ab | Chemical compounds |
EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
MY180558A (en) | 2007-09-21 | 2020-12-02 | Array Biopharma Inc | Pyridin-2-yl-amino-1,2,4- theiadiazole derivatives as glucokinase activators for the treatment of diabetes mellitus |
BRPI0917589A2 (pt) | 2008-08-04 | 2015-11-17 | Astrazeneca Ab | composto, composição farmacêutica, uso de um composto, método para tratar doenças, processo, combinação farmacêutica, e, reação de metiloxirano-2-carboxilato (ix) com um álcool roh |
GB0902434D0 (en) * | 2009-02-13 | 2009-04-01 | Astrazeneca Ab | Chemical process |
GB0902406D0 (en) * | 2009-02-13 | 2009-04-01 | Astrazeneca Ab | Crystalline polymorphic form |
WO2010116177A1 (en) | 2009-04-09 | 2010-10-14 | Astrazeneca Ab | A pyrazolo [4,5-e] pyrimidine derivative and its use to treat diabetes and obesity |
WO2010116176A1 (en) * | 2009-04-09 | 2010-10-14 | Astrazeneca Ab | Pyrazolo [4, 5-e] pyrimidine derivative and its use to treat diabetes and obesity |
GB0919757D0 (en) * | 2009-11-12 | 2009-12-30 | Johnson Matthey Plc | Polymorphs of bromfenac sodium and methods for preparing bromfenac sodium polymorphs |
US8299295B2 (en) | 2009-10-15 | 2012-10-30 | Johnson Matthey Public Limited Company | Polymorphs of bromfenac sodium and methods for preparing bromfenac sodium polymorphs |
WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
US8933024B2 (en) | 2010-06-18 | 2015-01-13 | Sanofi | Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
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TW200825060A (en) | 2006-10-26 | 2008-06-16 | Astrazeneca Ab | Chemical compounds |
UY30822A1 (es) | 2006-12-21 | 2008-07-31 | Astrazeneca Ab | Fnueva forma cristalina de 3-{[5-azetidin-1-ylcabonyl)pyrazin-2-yl]oxy}-5-[1-methylethyloxy]-n-1h-pyrazol-3-ylbenzamida, composiciones conteniéndola, procesos de preparacion y aplicaciones |
BRPI0917589A2 (pt) * | 2008-08-04 | 2015-11-17 | Astrazeneca Ab | composto, composição farmacêutica, uso de um composto, método para tratar doenças, processo, combinação farmacêutica, e, reação de metiloxirano-2-carboxilato (ix) com um álcool roh |
GB0902434D0 (en) * | 2009-02-13 | 2009-04-01 | Astrazeneca Ab | Chemical process |
GB0902406D0 (en) * | 2009-02-13 | 2009-04-01 | Astrazeneca Ab | Crystalline polymorphic form |
WO2010116176A1 (en) * | 2009-04-09 | 2010-10-14 | Astrazeneca Ab | Pyrazolo [4, 5-e] pyrimidine derivative and its use to treat diabetes and obesity |
WO2010116177A1 (en) * | 2009-04-09 | 2010-10-14 | Astrazeneca Ab | A pyrazolo [4,5-e] pyrimidine derivative and its use to treat diabetes and obesity |
-
2007
- 2007-10-24 TW TW096139912A patent/TW200825060A/zh unknown
- 2007-10-24 CL CL200703061A patent/CL2007003061A1/es unknown
- 2007-10-24 SA SA07280576A patent/SA07280576B1/ar unknown
- 2007-10-25 AR ARP070104727A patent/AR063393A1/es not_active Application Discontinuation
- 2007-10-25 RU RU2009114802/04A patent/RU2440992C2/ru not_active IP Right Cessation
- 2007-10-25 CA CA002667316A patent/CA2667316A1/en not_active Abandoned
- 2007-10-25 KR KR1020097010497A patent/KR20090084880A/ko not_active Application Discontinuation
- 2007-10-25 BR BRPI0718155-8A2A patent/BRPI0718155A2/pt not_active IP Right Cessation
- 2007-10-25 MX MX2009004467A patent/MX2009004467A/es active IP Right Grant
- 2007-10-25 WO PCT/GB2007/004057 patent/WO2008050117A1/en active Application Filing
- 2007-10-25 AU AU2007310624A patent/AU2007310624B2/en not_active Ceased
- 2007-10-25 EP EP10181670A patent/EP2272834A1/en not_active Withdrawn
- 2007-10-25 JP JP2009533939A patent/JP4673429B2/ja not_active Expired - Fee Related
- 2007-10-25 EP EP07824303A patent/EP2078000A1/en not_active Withdrawn
- 2007-10-25 CN CN201010118676A patent/CN101805299A/zh active Pending
- 2007-10-26 US US11/924,888 patent/US7671060B2/en not_active Expired - Fee Related
- 2007-10-26 PE PE2007001462A patent/PE20080927A1/es not_active Application Discontinuation
- 2007-10-29 UY UY30659A patent/UY30659A1/es not_active Application Discontinuation
-
2009
- 2009-04-16 IL IL198143A patent/IL198143A0/en unknown
- 2009-04-21 CO CO09040125A patent/CO6160314A2/es unknown
- 2009-04-22 NO NO20091596A patent/NO20091596L/no not_active Application Discontinuation
- 2009-12-22 US US12/644,249 patent/US7964725B2/en not_active Expired - Fee Related
-
2010
- 2010-10-08 JP JP2010228109A patent/JP2011046724A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
PE20080927A1 (es) | 2008-09-20 |
CO6160314A2 (es) | 2010-05-20 |
JP4673429B2 (ja) | 2011-04-20 |
CN101805299A (zh) | 2010-08-18 |
JP2010507641A (ja) | 2010-03-11 |
AR063393A1 (es) | 2009-01-28 |
AU2007310624A1 (en) | 2008-05-02 |
UY30659A1 (es) | 2008-05-31 |
US7671060B2 (en) | 2010-03-02 |
AU2007310624A8 (en) | 2009-05-14 |
BRPI0718155A2 (pt) | 2013-11-19 |
TW200825060A (en) | 2008-06-16 |
EP2272834A1 (en) | 2011-01-12 |
CA2667316A1 (en) | 2008-05-02 |
SA07280576B1 (ar) | 2011-06-22 |
KR20090084880A (ko) | 2009-08-05 |
JP2011046724A (ja) | 2011-03-10 |
IL198143A0 (en) | 2009-12-24 |
MX2009004467A (es) | 2009-07-27 |
RU2009114802A (ru) | 2010-12-10 |
AU2007310624B2 (en) | 2011-09-01 |
NO20091596L (no) | 2009-06-30 |
US20080318968A1 (en) | 2008-12-25 |
WO2008050117A1 (en) | 2008-05-02 |
RU2440992C2 (ru) | 2012-01-27 |
US7964725B2 (en) | 2011-06-21 |
US20100173825A1 (en) | 2010-07-08 |
EP2078000A1 (en) | 2009-07-15 |
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