JP2009502802A5 - - Google Patents
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- Publication number
- JP2009502802A5 JP2009502802A5 JP2008522959A JP2008522959A JP2009502802A5 JP 2009502802 A5 JP2009502802 A5 JP 2009502802A5 JP 2008522959 A JP2008522959 A JP 2008522959A JP 2008522959 A JP2008522959 A JP 2008522959A JP 2009502802 A5 JP2009502802 A5 JP 2009502802A5
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- JP
- Japan
- Prior art keywords
- compound
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- reagent
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- water
- Prior art date
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- 238000000034 method Methods 0.000 claims 28
- 239000003153 chemical reaction reagent Substances 0.000 claims 16
- ZMXDDKWLCZADIW-UHFFFAOYSA-N N,N-Dimethylformamide Chemical compound CN(C)C=O ZMXDDKWLCZADIW-UHFFFAOYSA-N 0.000 claims 12
- 150000001875 compounds Chemical class 0.000 claims 10
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 claims 10
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 10
- 229910052736 halogen Inorganic materials 0.000 claims 8
- CTSLXHKWHWQRSH-UHFFFAOYSA-N oxalyl chloride Chemical compound ClC(=O)C(Cl)=O CTSLXHKWHWQRSH-UHFFFAOYSA-N 0.000 claims 8
- 150000001412 amines Chemical class 0.000 claims 7
- 150000002367 halogens Chemical class 0.000 claims 7
- 230000003197 catalytic effect Effects 0.000 claims 6
- 238000006073 displacement reaction Methods 0.000 claims 6
- 239000003960 organic solvent Substances 0.000 claims 6
- 238000006243 chemical reaction Methods 0.000 claims 5
- 239000002904 solvent Substances 0.000 claims 5
- WYURNTSHIVDZCO-UHFFFAOYSA-N Tetrahydrofuran Chemical compound C1CCOC1 WYURNTSHIVDZCO-UHFFFAOYSA-N 0.000 claims 4
- 125000000753 cycloalkyl group Chemical group 0.000 claims 4
- 229910001415 sodium ion Inorganic materials 0.000 claims 4
- CSCPPACGZOOCGX-UHFFFAOYSA-N Acetone Chemical compound CC(C)=O CSCPPACGZOOCGX-UHFFFAOYSA-N 0.000 claims 3
- WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 claims 3
- YMWUJEATGCHHMB-UHFFFAOYSA-N Dichloromethane Chemical compound ClCCl YMWUJEATGCHHMB-UHFFFAOYSA-N 0.000 claims 3
- YXFVVABEGXRONW-UHFFFAOYSA-N Toluene Chemical compound CC1=CC=CC=C1 YXFVVABEGXRONW-UHFFFAOYSA-N 0.000 claims 3
- 125000003118 aryl group Chemical group 0.000 claims 3
- 125000000325 methylidene group Chemical group [H]C([H])=* 0.000 claims 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 3
- 229910001414 potassium ion Inorganic materials 0.000 claims 3
- -1 2-trifluoromethylphenyl Chemical group 0.000 claims 2
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 claims 2
- 229910052784 alkaline earth metal Inorganic materials 0.000 claims 2
- 230000015572 biosynthetic process Effects 0.000 claims 2
- 239000003054 catalyst Substances 0.000 claims 2
- 125000000623 heterocyclic group Chemical group 0.000 claims 2
- 125000000592 heterocycloalkyl group Chemical group 0.000 claims 2
- 150000002500 ions Chemical class 0.000 claims 2
- 229910052757 nitrogen Inorganic materials 0.000 claims 2
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 2
- 238000003786 synthesis reaction Methods 0.000 claims 2
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 claims 2
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 1
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 1
- WSLDOOZREJYCGB-UHFFFAOYSA-N 1,2-Dichloroethane Chemical compound ClCCCl WSLDOOZREJYCGB-UHFFFAOYSA-N 0.000 claims 1
- RYHBNJHYFVUHQT-UHFFFAOYSA-N 1,4-Dioxane Chemical compound C1COCCO1 RYHBNJHYFVUHQT-UHFFFAOYSA-N 0.000 claims 1
- VHUUQVKOLVNVRT-UHFFFAOYSA-N Ammonium hydroxide Chemical group [NH4+].[OH-] VHUUQVKOLVNVRT-UHFFFAOYSA-N 0.000 claims 1
- BZLVMXJERCGZMT-UHFFFAOYSA-N Methyl tert-butyl ether Chemical compound COC(C)(C)C BZLVMXJERCGZMT-UHFFFAOYSA-N 0.000 claims 1
- 125000003342 alkenyl group Chemical group 0.000 claims 1
- 125000000217 alkyl group Chemical group 0.000 claims 1
- 125000000304 alkynyl group Chemical group 0.000 claims 1
- QGZKDVFQNNGYKY-UHFFFAOYSA-N ammonia Natural products N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 claims 1
- 125000004093 cyano group Chemical group *C#N 0.000 claims 1
- 230000006378 damage Effects 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 125000001072 heteroaryl group Chemical group 0.000 claims 1
- 125000005842 heteroatom Chemical group 0.000 claims 1
- 229910021645 metal ion Inorganic materials 0.000 claims 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 1
- 125000001424 substituent group Chemical group 0.000 claims 1
- 238000006467 substitution reaction Methods 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US70115805P | 2005-07-21 | 2005-07-21 | |
| US60/701,158 | 2005-07-21 | ||
| PCT/US2006/028182 WO2007013974A2 (en) | 2005-07-21 | 2006-07-20 | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009502802A JP2009502802A (ja) | 2009-01-29 |
| JP2009502802A5 true JP2009502802A5 (enExample) | 2011-12-08 |
| JP4926172B2 JP4926172B2 (ja) | 2012-05-09 |
Family
ID=37571383
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008522959A Expired - Fee Related JP4926172B2 (ja) | 2005-07-21 | 2006-07-20 | スルホン酸塩よりスルホニルハライドおよびスルホンアミドを合成する方法 |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7842834B2 (enExample) |
| EP (1) | EP1907355B1 (enExample) |
| JP (1) | JP4926172B2 (enExample) |
| KR (1) | KR20080027868A (enExample) |
| CN (1) | CN101228118B (enExample) |
| AR (1) | AR057676A1 (enExample) |
| AU (1) | AU2006272886B2 (enExample) |
| BR (1) | BRPI0614005A2 (enExample) |
| CA (1) | CA2610228C (enExample) |
| CR (1) | CR9581A (enExample) |
| EC (1) | ECSP088116A (enExample) |
| ES (1) | ES2556620T3 (enExample) |
| GT (1) | GT200600325A (enExample) |
| IL (1) | IL187711A (enExample) |
| MX (1) | MX2008000816A (enExample) |
| NI (1) | NI200800018A (enExample) |
| NO (1) | NO20076358L (enExample) |
| PE (1) | PE20070245A1 (enExample) |
| RU (1) | RU2466983C2 (enExample) |
| SG (1) | SG163550A1 (enExample) |
| TW (1) | TW200728262A (enExample) |
| WO (1) | WO2007013974A2 (enExample) |
| ZA (1) | ZA200800557B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR048239A1 (es) | 2004-02-25 | 2006-04-12 | Wyeth Corp | Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo e intermediarios de sintesis de los mismos |
| SG163550A1 (en) | 2005-07-21 | 2010-08-30 | Wyeth Corp | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
| TW201036941A (en) * | 2009-03-30 | 2010-10-16 | Sumitomo Chemical Co | Method for producing sulfonamide compound |
| CN102887841A (zh) * | 2012-11-02 | 2013-01-23 | 天津希恩思生化科技有限公司 | 化合物丹磺酰氯的制备方法 |
| CN109722230B (zh) * | 2017-10-27 | 2021-07-23 | 中石化石油工程技术服务有限公司 | 一种油基钻井液用乳化剂及其制备方法和钻井液 |
| CN112110863A (zh) * | 2020-08-27 | 2020-12-22 | 中山大学 | 一种磺酰氟类化合物、其制备方法以及通过其制备磺酰胺类化合物的方法 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE48722C (de) | Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 | Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid | ||
| DE150313C (enExample) | ||||
| US2199568A (en) * | 1938-06-11 | 1940-05-07 | Gen Aniline & Film Corp | Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid |
| US2507408A (en) * | 1948-03-05 | 1950-05-09 | Rhone Poulenc Sa | 1-alkylsulfonyl-4-alkyl piperazines |
| US2888486A (en) * | 1953-11-20 | 1959-05-26 | Du Pont | Process for producing aromatic sulfonyl halides |
| US4885027A (en) * | 1985-04-05 | 1989-12-05 | Chevron Research Company | Herbicidal arylmethylenesulfonamido-acetamide and thioacetamide derivatives |
| JPS6310795A (ja) * | 1986-03-25 | 1988-01-18 | Takeda Chem Ind Ltd | 選択性除草化合物 |
| JP3814696B2 (ja) * | 1995-04-17 | 2006-08-30 | 住友精化株式会社 | 芳香族またはヘテロ芳香族スルホニルハライド類の製造方法 |
| JPH11292865A (ja) * | 1998-04-03 | 1999-10-26 | Ono Pharmaceut Co Ltd | 医薬品の中間体の製造方法 |
| JP4594574B2 (ja) * | 1999-08-03 | 2010-12-08 | 株式会社クレハ | Ｎ−（ベンジルスルホニル）ピコリン酸アミド誘導体、その製造方法及び除草剤 |
| FR2802121A1 (fr) * | 1999-12-14 | 2001-06-15 | Expansia Sa | Supports polymeriques organiques possedant des ligands mono- ou bi-dentates et leur utilisation en catalyse supportee |
| AU2002351182B2 (en) * | 2001-12-03 | 2009-01-15 | Novartis Ag | Inhibitors of cytosolic phospholipase A2 |
| EP1646617A2 (en) * | 2003-06-03 | 2006-04-19 | Rib-X Pharmaceuticals, Inc. | Sulfonamide compounds and methods of making and using the same |
| AR048239A1 (es) * | 2004-02-25 | 2006-04-12 | Wyeth Corp | Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo e intermediarios de sintesis de los mismos |
| SG163550A1 (en) | 2005-07-21 | 2010-08-30 | Wyeth Corp | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
| WO2010048122A1 (en) * | 2008-10-22 | 2010-04-29 | Cytec Technology Corp. | Improved processing of polymer matrix composites |
-
2006
- 2006-07-20 SG SG201004719-9A patent/SG163550A1/en unknown
- 2006-07-20 NI NI200800018A patent/NI200800018A/es unknown
- 2006-07-20 JP JP2008522959A patent/JP4926172B2/ja not_active Expired - Fee Related
- 2006-07-20 RU RU2007149184/04A patent/RU2466983C2/ru not_active Application Discontinuation
- 2006-07-20 WO PCT/US2006/028182 patent/WO2007013974A2/en not_active Ceased
- 2006-07-20 ES ES06800157.7T patent/ES2556620T3/es active Active
- 2006-07-20 CA CA2610228A patent/CA2610228C/en active Active
- 2006-07-20 TW TW095126535A patent/TW200728262A/zh unknown
- 2006-07-20 CN CN200680026736XA patent/CN101228118B/zh not_active Expired - Fee Related
- 2006-07-20 EP EP06800157.7A patent/EP1907355B1/en active Active
- 2006-07-20 BR BRPI0614005-0A patent/BRPI0614005A2/pt not_active Application Discontinuation
- 2006-07-20 AU AU2006272886A patent/AU2006272886B2/en not_active Ceased
- 2006-07-20 KR KR1020087001647A patent/KR20080027868A/ko not_active Ceased
- 2006-07-20 US US11/490,389 patent/US7842834B2/en active Active
- 2006-07-20 MX MX2008000816A patent/MX2008000816A/es active IP Right Grant
- 2006-07-21 AR ARP060103164A patent/AR057676A1/es unknown
- 2006-07-21 PE PE2006000883A patent/PE20070245A1/es not_active Application Discontinuation
- 2006-07-21 GT GT200600325A patent/GT200600325A/es unknown
-
2007
- 2007-11-28 IL IL187711A patent/IL187711A/en active IP Right Grant
- 2007-12-07 CR CR9581A patent/CR9581A/es not_active Application Discontinuation
- 2007-12-12 NO NO20076358A patent/NO20076358L/no not_active Application Discontinuation
-
2008
- 2008-01-17 EC EC2008008116A patent/ECSP088116A/es unknown
- 2008-01-18 ZA ZA2008/00557A patent/ZA200800557B/en unknown
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