ES2556620T3 - Proceso para la síntesis de haluros de sulfonilo y sulfonamidas a partir de sales de ácido sulfónico - Google Patents

Proceso para la síntesis de haluros de sulfonilo y sulfonamidas a partir de sales de ácido sulfónico Download PDF

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Publication number
ES2556620T3
ES2556620T3 ES06800157.7T ES06800157T ES2556620T3 ES 2556620 T3 ES2556620 T3 ES 2556620T3 ES 06800157 T ES06800157 T ES 06800157T ES 2556620 T3 ES2556620 T3 ES 2556620T3
Authority
ES
Spain
Prior art keywords
alkyl
compound
formula
group
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES06800157.7T
Other languages
English (en)
Spanish (es)
Inventor
Ronal Stanley Michalak
Jean Louise Helom
Joseph Zeldis
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ziarco Pharma Ltd
Original Assignee
Ziarco Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ziarco Pharma Ltd filed Critical Ziarco Pharma Ltd
Application granted granted Critical
Publication of ES2556620T3 publication Critical patent/ES2556620T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C07C303/38—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reaction of ammonia or amines with sulfonic acids, or with esters, anhydrides, or halides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/42—Separation; Purification; Stabilisation; Use of additives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/07—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
ES06800157.7T 2005-07-21 2006-07-20 Proceso para la síntesis de haluros de sulfonilo y sulfonamidas a partir de sales de ácido sulfónico Expired - Lifetime ES2556620T3 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70115805P 2005-07-21 2005-07-21
US701158P 2005-07-21
PCT/US2006/028182 WO2007013974A2 (en) 2005-07-21 2006-07-20 Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts

Publications (1)

Publication Number Publication Date
ES2556620T3 true ES2556620T3 (es) 2016-01-19

Family

ID=37571383

Family Applications (1)

Application Number Title Priority Date Filing Date
ES06800157.7T Expired - Lifetime ES2556620T3 (es) 2005-07-21 2006-07-20 Proceso para la síntesis de haluros de sulfonilo y sulfonamidas a partir de sales de ácido sulfónico

Country Status (23)

Country Link
US (1) US7842834B2 (enExample)
EP (1) EP1907355B1 (enExample)
JP (1) JP4926172B2 (enExample)
KR (1) KR20080027868A (enExample)
CN (1) CN101228118B (enExample)
AR (1) AR057676A1 (enExample)
AU (1) AU2006272886B2 (enExample)
BR (1) BRPI0614005A2 (enExample)
CA (1) CA2610228C (enExample)
CR (1) CR9581A (enExample)
EC (1) ECSP088116A (enExample)
ES (1) ES2556620T3 (enExample)
GT (1) GT200600325A (enExample)
IL (1) IL187711A (enExample)
MX (1) MX2008000816A (enExample)
NI (1) NI200800018A (enExample)
NO (1) NO20076358L (enExample)
PE (1) PE20070245A1 (enExample)
RU (1) RU2466983C2 (enExample)
SG (1) SG163550A1 (enExample)
TW (1) TW200728262A (enExample)
WO (1) WO2007013974A2 (enExample)
ZA (1) ZA200800557B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR048239A1 (es) 2004-02-25 2006-04-12 Wyeth Corp Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo e intermediarios de sintesis de los mismos
CA2610228C (en) 2005-07-21 2014-02-18 Wyeth Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts
TW201036941A (en) * 2009-03-30 2010-10-16 Sumitomo Chemical Co Method for producing sulfonamide compound
CN102887841A (zh) * 2012-11-02 2013-01-23 天津希恩思生化科技有限公司 化合物丹磺酰氯的制备方法
CN109722230B (zh) * 2017-10-27 2021-07-23 中石化石油工程技术服务有限公司 一种油基钻井液用乳化剂及其制备方法和钻井液
CN112110863A (zh) * 2020-08-27 2020-12-22 中山大学 一种磺酰氟类化合物、其制备方法以及通过其制备磺酰胺类化合物的方法
CN116514868A (zh) * 2022-01-20 2023-08-01 华创合成制药股份有限公司 一种用于治疗的磺酰胺类化合物其及制备方法和用途

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE150313C (enExample)
DE48722C (de) Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid
US2199568A (en) 1938-06-11 1940-05-07 Gen Aniline & Film Corp Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid
US2507408A (en) * 1948-03-05 1950-05-09 Rhone Poulenc Sa 1-alkylsulfonyl-4-alkyl piperazines
US2888486A (en) * 1953-11-20 1959-05-26 Du Pont Process for producing aromatic sulfonyl halides
US4885027A (en) * 1985-04-05 1989-12-05 Chevron Research Company Herbicidal arylmethylenesulfonamido-acetamide and thioacetamide derivatives
JPS6310795A (ja) * 1986-03-25 1988-01-18 Takeda Chem Ind Ltd 選択性除草化合物
JP3814696B2 (ja) * 1995-04-17 2006-08-30 住友精化株式会社 芳香族またはヘテロ芳香族スルホニルハライド類の製造方法
JPH11292865A (ja) * 1998-04-03 1999-10-26 Ono Pharmaceut Co Ltd 医薬品の中間体の製造方法
JP4594574B2 (ja) * 1999-08-03 2010-12-08 株式会社クレハ Ｎ−（ベンジルスルホニル）ピコリン酸アミド誘導体、その製造方法及び除草剤
FR2802121A1 (fr) * 1999-12-14 2001-06-15 Expansia Sa Supports polymeriques organiques possedant des ligands mono- ou bi-dentates et leur utilisation en catalyse supportee
HUP0402577A3 (en) * 2001-12-03 2011-05-30 Wyeth Corp Indole derivatives as inhibitors of cytosolic phospholipase a2, process for producing them and pharmaceutical compositions containing them
US20060270680A1 (en) * 2003-06-03 2006-11-30 Goldberg Joel A Sulfonamide compounds and methods of making and using the same
AR048239A1 (es) 2004-02-25 2006-04-12 Wyeth Corp Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo e intermediarios de sintesis de los mismos
CA2610228C (en) 2005-07-21 2014-02-18 Wyeth Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts
KR101680393B1 (ko) * 2008-10-22 2016-11-28 사이텍 테크놀러지 코포레이션 중합체 매트릭스 복합재의 개선된 가공성

Also Published As

Publication number Publication date
CR9581A (es) 2008-03-06
GT200600325A (es) 2007-02-26
ZA200800557B (en) 2011-06-26
US7842834B2 (en) 2010-11-30
BRPI0614005A2 (pt) 2011-03-01
IL187711A (en) 2016-04-21
AU2006272886B2 (en) 2012-03-01
AR057676A1 (es) 2007-12-12
JP4926172B2 (ja) 2012-05-09
IL187711A0 (en) 2008-08-07
KR20080027868A (ko) 2008-03-28
NO20076358L (no) 2008-04-16
TW200728262A (en) 2007-08-01
CA2610228C (en) 2014-02-18
RU2466983C2 (ru) 2012-11-20
WO2007013974A3 (en) 2007-04-12
EP1907355A2 (en) 2008-04-09
CA2610228A1 (en) 2007-02-01
SG163550A1 (en) 2010-08-30
PE20070245A1 (es) 2007-03-26
CN101228118A (zh) 2008-07-23
WO2007013974A2 (en) 2007-02-01
AU2006272886A1 (en) 2007-02-01
MX2008000816A (es) 2008-03-18
RU2007149184A (ru) 2009-08-27
EP1907355B1 (en) 2015-08-05
ECSP088116A (es) 2008-02-20
NI200800018A (es) 2009-03-03
JP2009502802A (ja) 2009-01-29
CN101228118B (zh) 2013-09-18
US20070021614A1 (en) 2007-01-25

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