CN101228118B - 由磺酸盐合成磺酰卤和磺酰胺的方法 - Google Patents
由磺酸盐合成磺酰卤和磺酰胺的方法 Download PDFInfo
- Publication number
- CN101228118B CN101228118B CN200680026736XA CN200680026736A CN101228118B CN 101228118 B CN101228118 B CN 101228118B CN 200680026736X A CN200680026736X A CN 200680026736XA CN 200680026736 A CN200680026736 A CN 200680026736A CN 101228118 B CN101228118 B CN 101228118B
- Authority
- CN
- China
- Prior art keywords
- compound
- alkyl
- formula
- reagent
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 0 *Cc1c(C*)[n](*)c2c1cccc2 Chemical compound *Cc1c(C*)[n](*)c2c1cccc2 0.000 description 3
- DPDRNZHWQDQFSQ-UHFFFAOYSA-N CCNCS(C)(=O)=O Chemical compound CCNCS(C)(=O)=O DPDRNZHWQDQFSQ-UHFFFAOYSA-N 0.000 description 1
- ABTFCSFEAMEIGN-UHFFFAOYSA-N CN(N)S(C)(=O)=O Chemical compound CN(N)S(C)(=O)=O ABTFCSFEAMEIGN-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
- C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
- C07C303/38—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reaction of ammonia or amines with sulfonic acids, or with esters, anhydrides, or halides thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/42—Separation; Purification; Stabilisation; Use of additives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/07—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US70115805P | 2005-07-21 | 2005-07-21 | |
| US60/701,158 | 2005-07-21 | ||
| PCT/US2006/028182 WO2007013974A2 (en) | 2005-07-21 | 2006-07-20 | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN101228118A CN101228118A (zh) | 2008-07-23 |
| CN101228118B true CN101228118B (zh) | 2013-09-18 |
Family
ID=37571383
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN200680026736XA Expired - Fee Related CN101228118B (zh) | 2005-07-21 | 2006-07-20 | 由磺酸盐合成磺酰卤和磺酰胺的方法 |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7842834B2 (enExample) |
| EP (1) | EP1907355B1 (enExample) |
| JP (1) | JP4926172B2 (enExample) |
| KR (1) | KR20080027868A (enExample) |
| CN (1) | CN101228118B (enExample) |
| AR (1) | AR057676A1 (enExample) |
| AU (1) | AU2006272886B2 (enExample) |
| BR (1) | BRPI0614005A2 (enExample) |
| CA (1) | CA2610228C (enExample) |
| CR (1) | CR9581A (enExample) |
| EC (1) | ECSP088116A (enExample) |
| ES (1) | ES2556620T3 (enExample) |
| GT (1) | GT200600325A (enExample) |
| IL (1) | IL187711A (enExample) |
| MX (1) | MX2008000816A (enExample) |
| NI (1) | NI200800018A (enExample) |
| NO (1) | NO20076358L (enExample) |
| PE (1) | PE20070245A1 (enExample) |
| RU (1) | RU2466983C2 (enExample) |
| SG (1) | SG163550A1 (enExample) |
| TW (1) | TW200728262A (enExample) |
| WO (1) | WO2007013974A2 (enExample) |
| ZA (1) | ZA200800557B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR048239A1 (es) | 2004-02-25 | 2006-04-12 | Wyeth Corp | Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo e intermediarios de sintesis de los mismos |
| SG163550A1 (en) | 2005-07-21 | 2010-08-30 | Wyeth Corp | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
| TW201036941A (en) * | 2009-03-30 | 2010-10-16 | Sumitomo Chemical Co | Method for producing sulfonamide compound |
| CN102887841A (zh) * | 2012-11-02 | 2013-01-23 | 天津希恩思生化科技有限公司 | 化合物丹磺酰氯的制备方法 |
| CN109722230B (zh) * | 2017-10-27 | 2021-07-23 | 中石化石油工程技术服务有限公司 | 一种油基钻井液用乳化剂及其制备方法和钻井液 |
| CN112110863A (zh) * | 2020-08-27 | 2020-12-22 | 中山大学 | 一种磺酰氟类化合物、其制备方法以及通过其制备磺酰胺类化合物的方法 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN87102275A (zh) * | 1986-03-25 | 1988-02-17 | 武田药品工业株式会社 | 选择性除草剂及其制造和使用 |
| CN1150796A (zh) * | 1995-04-17 | 1997-05-28 | 住友精化株式会社 | 芳香族或杂芳族磺酰卤类的制备方法 |
| CN1617855A (zh) * | 2001-12-03 | 2005-05-18 | 惠氏公司 | 细胞溶质磷脂酶a2抑制剂 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE48722C (de) | Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 | Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid | ||
| DE150313C (enExample) | ||||
| US2199568A (en) * | 1938-06-11 | 1940-05-07 | Gen Aniline & Film Corp | Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid |
| US2507408A (en) * | 1948-03-05 | 1950-05-09 | Rhone Poulenc Sa | 1-alkylsulfonyl-4-alkyl piperazines |
| US2888486A (en) * | 1953-11-20 | 1959-05-26 | Du Pont | Process for producing aromatic sulfonyl halides |
| US4885027A (en) * | 1985-04-05 | 1989-12-05 | Chevron Research Company | Herbicidal arylmethylenesulfonamido-acetamide and thioacetamide derivatives |
| JPH11292865A (ja) * | 1998-04-03 | 1999-10-26 | Ono Pharmaceut Co Ltd | 医薬品の中間体の製造方法 |
| JP4594574B2 (ja) * | 1999-08-03 | 2010-12-08 | 株式会社クレハ | Ｎ−（ベンジルスルホニル）ピコリン酸アミド誘導体、その製造方法及び除草剤 |
| FR2802121A1 (fr) * | 1999-12-14 | 2001-06-15 | Expansia Sa | Supports polymeriques organiques possedant des ligands mono- ou bi-dentates et leur utilisation en catalyse supportee |
| EP1646617A2 (en) * | 2003-06-03 | 2006-04-19 | Rib-X Pharmaceuticals, Inc. | Sulfonamide compounds and methods of making and using the same |
| AR048239A1 (es) * | 2004-02-25 | 2006-04-12 | Wyeth Corp | Procesos para la preparacion de haluros de aril- y heteroaril-alquilsulfonilo e intermediarios de sintesis de los mismos |
| SG163550A1 (en) | 2005-07-21 | 2010-08-30 | Wyeth Corp | Process for the synthesis of sulfonyl halides and sulfonamides from sulfonic acid salts |
| WO2010048122A1 (en) * | 2008-10-22 | 2010-04-29 | Cytec Technology Corp. | Improved processing of polymer matrix composites |
-
2006
- 2006-07-20 SG SG201004719-9A patent/SG163550A1/en unknown
- 2006-07-20 NI NI200800018A patent/NI200800018A/es unknown
- 2006-07-20 JP JP2008522959A patent/JP4926172B2/ja not_active Expired - Fee Related
- 2006-07-20 RU RU2007149184/04A patent/RU2466983C2/ru not_active Application Discontinuation
- 2006-07-20 WO PCT/US2006/028182 patent/WO2007013974A2/en not_active Ceased
- 2006-07-20 ES ES06800157.7T patent/ES2556620T3/es active Active
- 2006-07-20 CA CA2610228A patent/CA2610228C/en active Active
- 2006-07-20 TW TW095126535A patent/TW200728262A/zh unknown
- 2006-07-20 CN CN200680026736XA patent/CN101228118B/zh not_active Expired - Fee Related
- 2006-07-20 EP EP06800157.7A patent/EP1907355B1/en active Active
- 2006-07-20 BR BRPI0614005-0A patent/BRPI0614005A2/pt not_active Application Discontinuation
- 2006-07-20 AU AU2006272886A patent/AU2006272886B2/en not_active Ceased
- 2006-07-20 KR KR1020087001647A patent/KR20080027868A/ko not_active Ceased
- 2006-07-20 US US11/490,389 patent/US7842834B2/en active Active
- 2006-07-20 MX MX2008000816A patent/MX2008000816A/es active IP Right Grant
- 2006-07-21 AR ARP060103164A patent/AR057676A1/es unknown
- 2006-07-21 PE PE2006000883A patent/PE20070245A1/es not_active Application Discontinuation
- 2006-07-21 GT GT200600325A patent/GT200600325A/es unknown
-
2007
- 2007-11-28 IL IL187711A patent/IL187711A/en active IP Right Grant
- 2007-12-07 CR CR9581A patent/CR9581A/es not_active Application Discontinuation
- 2007-12-12 NO NO20076358A patent/NO20076358L/no not_active Application Discontinuation
-
2008
- 2008-01-17 EC EC2008008116A patent/ECSP088116A/es unknown
- 2008-01-18 ZA ZA2008/00557A patent/ZA200800557B/en unknown
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN87102275A (zh) * | 1986-03-25 | 1988-02-17 | 武田药品工业株式会社 | 选择性除草剂及其制造和使用 |
| CN1150796A (zh) * | 1995-04-17 | 1997-05-28 | 住友精化株式会社 | 芳香族或杂芳族磺酰卤类的制备方法 |
| CN1617855A (zh) * | 2001-12-03 | 2005-05-18 | 惠氏公司 | 细胞溶质磷脂酶a2抑制剂 |
Non-Patent Citations (1)
| Title |
|---|
| Derek Brundish等.Design and Synthesis of Thrombin Inhibitors: Analogues of MD-805 with Reduced Stereogenicity and Improved Potency.《J. Med. Chem.》.1999,第42卷(第22期), * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1907355B1 (en) | 2015-08-05 |
| IL187711A (en) | 2016-04-21 |
| GT200600325A (es) | 2007-02-26 |
| CN101228118A (zh) | 2008-07-23 |
| ECSP088116A (es) | 2008-02-20 |
| AU2006272886A1 (en) | 2007-02-01 |
| CA2610228A1 (en) | 2007-02-01 |
| KR20080027868A (ko) | 2008-03-28 |
| ZA200800557B (en) | 2011-06-26 |
| JP4926172B2 (ja) | 2012-05-09 |
| AR057676A1 (es) | 2007-12-12 |
| US20070021614A1 (en) | 2007-01-25 |
| NI200800018A (es) | 2009-03-03 |
| WO2007013974A3 (en) | 2007-04-12 |
| BRPI0614005A2 (pt) | 2011-03-01 |
| EP1907355A2 (en) | 2008-04-09 |
| AU2006272886B2 (en) | 2012-03-01 |
| CA2610228C (en) | 2014-02-18 |
| WO2007013974A2 (en) | 2007-02-01 |
| ES2556620T3 (es) | 2016-01-19 |
| NO20076358L (no) | 2008-04-16 |
| MX2008000816A (es) | 2008-03-18 |
| JP2009502802A (ja) | 2009-01-29 |
| IL187711A0 (en) | 2008-08-07 |
| RU2007149184A (ru) | 2009-08-27 |
| SG163550A1 (en) | 2010-08-30 |
| TW200728262A (en) | 2007-08-01 |
| US7842834B2 (en) | 2010-11-30 |
| RU2466983C2 (ru) | 2012-11-20 |
| CR9581A (es) | 2008-03-06 |
| PE20070245A1 (es) | 2007-03-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| ASS | Succession or assignment of patent right |
Owner name: QIAIKE CORP. Free format text: FORMER OWNER: WYETH CORP. Effective date: 20130911 |
|
| C41 | Transfer of patent application or patent right or utility model | ||
| TR01 | Transfer of patent right |
Effective date of registration: 20130911 Address after: California, USA Patentee after: Chieko Co. Address before: New jersey, USA Patentee before: WYETH |
|
| CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20130918 |
|
| CF01 | Termination of patent right due to non-payment of annual fee |